Evaluation of the sensitivities of six triple-negative breast cancer (TNBC) cell lines to 23 different PI3K/AKT/mTOR inhibitors or to a MEK inhibitor (trametinib). Dataset 2 of 2: GR metrics. - Dataset (ID:20365)

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Cell line Drug name Experimental replicate Timepoint Curve type (GR values) Curve type (relative cell counts) Experiment name Number of concentrations Cell doublings (DMSO control) GR50 GRmax GR_AOC GEC50 GRinf Hill slope (GR values) R-squared sigmoid fit (GR values) P-value sigmoid fit (GR values) R-squared flat fit (GR values) IC50 Emax AUC EC50 Einf Hill slope (relative cell counts) R-squared sigmoid fit (relative cell counts) P-value sigmoid fit (relative cell counts) R-squared flat fit (relative cell counts)
BT-549 MK2206 3 72
sigmoid
sigmoid
BT549 MK-2206 0 3 72
8 1.685
Inf
0.714
0.131
0.123
0.711
3.44
0.953
0.000102
NA
Inf
0.771
0.895
0.123
0.768
3.25
0.949
0.000136
NA
BT-549 AZD-6482 2 72
sigmoid
sigmoid
BT549 AZD6482 0 2 72
8 1.973
9.15
0.635
0.112
120.0
-1.0
0.426
0.951
0.000115
NA
19.4
0.672
0.895
19.4
0.0
0.437
0.946
0.000154
NA
HCC70 Trametinib 3 72
sigmoid
sigmoid
HCC70 trametinib 0 3 72
8 2.463
Inf
0.56
0.361
0.00419
0.548
0.954
0.95
0.000123
NA
Inf
0.542
0.618
0.00342
0.533
0.965
0.958
7.33e-05
NA
BT-20 Torin2 2 72
sigmoid
sigmoid
BT20 Torin2 0 2 72
8 1.733
0.00315
-0.761
0.992
0.0484
-0.95
0.389
0.949
0.000131
NA
0.00804
0.0252
0.336
0.00642
0.0613
0.583
0.974
1.77e-05
NA
HCC38 Trametinib 1 72
sigmoid
sigmoid
HCC38 trametinib 0 1 72
8 1.733
0.162
0.196
0.407
0.173
-0.0184
0.559
0.948
0.000139
NA
0.568
0.41
0.686
0.161
0.234
0.501
0.947
0.000151
NA
HCC70 TGX221 2 72
sigmoid
sigmoid
HCC70 TGX-221 0 2 72
8 1.786
1.77
0.467
0.233
0.531
0.227
0.503
0.948
0.000139
NA
5.85
0.575
0.806
3.44
0.0897
0.372
0.937
0.000249
NA
Hs 578T CAL-101 1
sigmoid
sigmoid
Hs578T idelalisib 1
8 2.050
27.9
0.72
0.0764
4.56
0.356
0.688
0.945
0.000168
NA
18.7
0.734
0.925
18.7
0.0
0.568
0.941
0.000203
NA
HCC70 Trametinib 2 72
sigmoid
sigmoid
HCC70 trametinib 0 2 72
8 1.721
0.506
0.504
0.395
0.00469
0.467
0.581
0.944
0.000179
NA
Inf
0.612
0.687
0.00389
0.585
0.57
0.948
0.000138
NA
BT-549 Pictilisib 2 72
sigmoid
sigmoid
BT549 pictilisib 0 2 72
8 1.960
1.84
0.365
0.166
11.5
-1.0
0.599
0.943
0.000187
NA
2.82
0.473
0.851
2.82
0.0
0.647
0.924
0.000432
NA
BT-549 AZD8055 3 72
sigmoid
sigmoid
BT549 AZD8055 0 3 72
8 1.757
0.0178
0.159
0.59
0.0122
0.145
0.913
0.942
0.000193
NA
0.0479
0.383
0.555
0.00973
0.372
0.854
0.954
9.74e-05
NA
BT-549 Trametinib 3 72
sigmoid
sigmoid
BT549 trametinib 0 3 72
8 1.755
Inf
0.553
0.223
0.107
0.505
0.899
0.942
0.000194
NA
Inf
0.642
0.817
0.104
0.595
0.804
0.938
0.000236
NA
HCC1806 AS605240 3 72
sigmoid
sigmoid
HCC1806 AS-605240 0 3 72
8 3.181
Inf
0.923
0.011
0.57
0.923
2.81
0.936
0.000257
NA
Inf
0.883
0.983
0.559
0.882
2.81
0.931
0.000333
NA
BT-20 AZD8055 2 72
sigmoid
sigmoid
BT20 AZD8055 0 2 72
8 1.951
0.00909
0.155
0.651
0.00651
0.115
0.785
0.936
0.000258
NA
0.0185
0.343
0.477
0.00469
0.311
0.706
0.934
0.000289
NA
HCC1806 AS605240 2 72
sigmoid
sigmoid
HCC1806 AS-605240 0 2 72
8 2.813
Inf
0.913
0.0124
0.569
0.913
2.8
0.936
0.000261
NA
Inf
0.883
0.983
0.559
0.882
2.81
0.931
0.000333
NA
HCC1806 AS605240 1 72
sigmoid
sigmoid
HCC1806 AS-605240 0 1 72
8 2.728
Inf
0.911
0.0128
0.569
0.91
2.8
0.936
0.000262
NA
Inf
0.883
0.983
0.559
0.882
2.81
0.931
0.000333
NA
HCC38 AS605240 2 72
sigmoid
sigmoid
HCC38 AS-605240 0 2 72
8 2.200
17.4
0.642
0.114
4.07
0.256
0.493
0.936
0.000265
NA
46.2
0.648
0.882
1.68
0.411
0.522
0.929
0.000356
NA
HCC38 Everolimus 3 72
sigmoid
sigmoid
HCC38 everolimus 0 3 72
8 1.437
5.11
0.511
0.429
0.000567
0.299
0.1
0.934
0.000284
NA
573000000.0
0.668
0.707
0.000349
0.53
0.1
0.932
0.000308
NA
BT-20 AZD8055 3 72
sigmoid
sigmoid
BT20 AZD8055 0 3 72
8 2.694
0.0351
0.345
0.472
0.0116
0.313
0.89
0.934
0.000286
NA
0.0291
0.343
0.506
0.00813
0.306
0.743
0.922
0.000471
NA
HCC38 Pictilisib 2 72
sigmoid
sigmoid
HCC38 pictilisib 0 2 72
8 2.112
Inf
0.622
0.0838
0.644
0.58
1.32
0.933
0.000298
NA
Inf
0.642
0.918
0.568
0.612
1.36
0.922
0.000475
NA
BT-549 CAL-101 2 72
sigmoid
sigmoid
BT549 idelalisib 0 2 72
8 1.975
Inf
0.792
0.0561
4.65
0.526
0.693
0.933
0.000307
NA
43.0
0.805
0.946
43.0
0.0
0.548
0.932
0.000314
NA
BT-549 CAL-101 1 72
sigmoid
sigmoid
BT549 idelalisib 0 1 72
8 1.791
Inf
0.836
0.041
4.8
0.605
0.778
0.924
0.00044
NA
Inf
0.858
0.964
4.79
0.659
0.767
0.92
0.000518
NA
BT-20 WYE-125132 3 72
sigmoid
sigmoid
BT20 WYE-132 0 3 72
8 2.654
0.0504
0.282
0.465
0.0254
0.236
0.929
0.922
0.000468
NA
0.048
0.307
0.526
0.0182
0.246
0.698
0.918
0.000553
NA
HCC38 PIK-93 2 72
sigmoid
sigmoid
HCC38 PIK-93 0 2 72
8 2.107
31.9
0.661
0.0151
2.16
0.497
1.86
0.922
0.000468
NA
Inf
0.676
0.987
1.97
0.545
1.87
0.907
0.000813
NA
BT-549 KIN001-244 3 72
sigmoid
sigmoid
BT549 KIN001-244 0 3 72
8 1.740
Inf
0.861
0.0287
4.69
0.681
0.74
0.922
0.00047
NA
Inf
0.882
0.975
4.7
0.729
0.732
0.919
0.000531
NA
HCC38 PIK-93 3 72
sigmoid
sigmoid
HCC38 PIK-93 0 3 72
8 1.382
5.05
0.598
0.061
2.34
0.358
1.63
0.919
0.000533
NA
Inf
0.734
0.959
2.23
0.586
1.64
0.914
0.000645
NA
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