Evaluation of the sensitivities of six triple-negative breast cancer (TNBC) cell lines to 23 different PI3K/AKT/mTOR inhibitors or to a MEK inhibitor (trametinib). Dataset 2 of 2: GR metrics. - Dataset (ID:20365)

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Cell line Drug name Experimental replicate Timepoint Curve type (GR values) Curve type (relative cell counts) Experiment name Number of concentrations Cell doublings (DMSO control) GR50 GRmax GR_AOC GEC50 GRinf Hill slope (GR values) R-squared sigmoid fit (GR values) P-value sigmoid fit (GR values) R-squared flat fit (GR values) IC50 Emax AUC EC50 Einf Hill slope (relative cell counts) R-squared sigmoid fit (relative cell counts) P-value sigmoid fit (relative cell counts) R-squared flat fit (relative cell counts)
BT-549 Dactolisib 3 72
sigmoid
sigmoid
BT549 dactolisib 0 3 72
8 1.801
0.0058
-0.00929
0.751
0.00579
0.000747
0.866
0.994
2.41e-07
NA
0.011
0.282
0.442
0.00425
0.29
0.909
0.995
1.54e-07
NA
HCC38 AZD8055 3 72
sigmoid
sigmoid
HCC38 AZD8055 0 3 72
8 1.417
0.0464
0.0327
0.53
0.0463
0.000983
1.04
0.997
4.27e-08
NA
0.157
0.392
0.658
0.041
0.372
1.02
0.996
5.78e-08
NA
HCC38 Dactolisib 2 72
sigmoid
sigmoid
HCC38 dactolisib 0 2 72
8 2.120
0.0118
-0.0557
0.668
0.0118
-0.00134
0.785
0.98
7.61e-06
NA
0.0145
0.204
0.447
0.00701
0.245
0.927
0.988
1.88e-06
NA
BT-549 ZSTK474 1 72
sigmoid
sigmoid
BT549 ZSTK474 0 1 72
8 1.861
0.58
0.213
0.256
0.583
-0.00205
0.771
0.992
5.43e-07
NA
1.12
0.394
0.788
0.428
0.261
0.767
0.989
1.49e-06
NA
HCC38 Trametinib 2 72
sigmoid
sigmoid
HCC38 trametinib 0 2 72
8 2.133
0.219
0.267
0.389
0.222
-0.00324
0.424
0.987
2.39e-06
NA
0.391
0.377
0.644
0.127
0.183
0.404
0.988
1.91e-06
NA
HCC70 BX-912 2 72
sigmoid
sigmoid
HCC70 BX-912 0 2 72
8 1.693
1.25
0.00257
0.0619
1.25
-0.00649
5.0
0.971
2.55e-05
NA
1.44
0.311
0.961
1.2
0.306
5.0
0.956
8.35e-05
NA
Hs 578T Dactolisib 2
sigmoid
sigmoid
Hs578T dactolisib 2
8 2.509
0.0128
-0.0617
0.655
0.0126
0.00741
0.79
0.974
1.78e-05
NA
0.0105
0.15
0.405
0.00638
0.203
1.04
0.985
3.67e-06
NA
BT-549 GDC-0980 2 72
sigmoid
sigmoid
BT549 apitolisib 0 2 72
8 1.939
0.189
0.0264
0.357
0.193
-0.011
1.04
0.997
2.98e-08
NA
0.278
0.274
0.71
0.142
0.257
1.07
0.997
3.64e-08
NA
Hs 578T AS605240 2
sigmoid
sigmoid
Hs578T AS-605240 2
8 2.547
1.89
0.43
0.194
1.81
0.011
0.541
0.988
1.81e-06
NA
1.6
0.426
0.784
0.971
0.117
0.532
0.983
4.67e-06
NA
HCC38 WYE-125132 3 72
sigmoid
sigmoid
HCC38 WYE-132 0 3 72
8 1.449
0.0494
-0.0216
0.518
0.0504
-0.0117
1.18
0.998
9.69e-09
NA
0.128
0.355
0.662
0.0441
0.361
1.2
0.998
9.53e-09
NA
Hs 578T Dactolisib 1
sigmoid
sigmoid
Hs578T dactolisib 1
8 2.047
0.00952
-0.0606
0.691
0.00928
0.0117
0.91
0.977
1.27e-05
NA
0.0124
0.213
0.443
0.00621
0.259
1.06
0.985
3.61e-06
NA
HCC38 Torin1 1 72
sigmoid
sigmoid
HCC38 Torin1 0 1 72
8 1.688
0.0287
-0.0113
0.569
0.0278
0.013
0.843
0.993
4.14e-07
NA
0.0653
0.304
0.585
0.0204
0.325
0.9
0.992
4.53e-07
NA
BT-549 GDC-0980 3 72
sigmoid
sigmoid
BT549 apitolisib 0 3 72
8 1.802
0.162
0.0283
0.377
0.158
0.0179
1.2
0.994
2.53e-07
NA
0.268
0.302
0.709
0.128
0.294
1.2
0.992
4.85e-07
NA
HCC38 Trametinib 1 72
sigmoid
sigmoid
HCC38 trametinib 0 1 72
8 1.733
0.162
0.196
0.407
0.173
-0.0184
0.559
0.948
0.000139
NA
0.568
0.41
0.686
0.161
0.234
0.501
0.947
0.000151
NA
HCC38 Dactolisib 1 72
sigmoid
sigmoid
HCC38 dactolisib 0 1 72
8 1.821
0.0109
-0.0403
0.672
0.0104
0.0212
0.892
0.985
3.44e-06
NA
0.0194
0.263
0.492
0.00757
0.301
0.975
0.988
1.65e-06
NA
BT-549 PI103 3 72
sigmoid
sigmoid
BT549 PI-103 0 3 72
8 1.758
0.16
0.00249
0.391
0.166
-0.0225
1.12
0.989
1.19e-06
NA
0.279
0.297
0.704
0.134
0.28
1.12
0.985
3.23e-06
NA
HCC70 AZD-6482 2 72
sigmoid
sigmoid
HCC70 AZD6482 0 2 72
8 1.772
0.267
0.256
0.366
0.237
0.0255
0.43
0.987
2.27e-06
NA
1.16
0.438
0.706
0.133
0.306
0.437
0.986
3.03e-06
NA
BT-549 PI103 2 72
sigmoid
sigmoid
BT549 PI-103 0 2 72
8 1.893
0.218
0.0201
0.344
0.229
-0.0262
1.08
0.997
2.55e-08
NA
0.326
0.28
0.725
0.169
0.261
1.13
0.996
6.2e-08
NA
BT-20 PI103 1 72
sigmoid
sigmoid
BT20 PI-103 0 1 72
8 1.924
0.646
-0.0114
0.16
0.659
-0.0268
2.6
0.978
1.1e-05
NA
0.753
0.258
0.883
0.579
0.252
2.68
0.964
4.79e-05
NA
BT-20 PI103 3 72
sigmoid
sigmoid
BT20 PI-103 0 3 72
8 2.496
0.373
0.0139
0.282
0.387
-0.0286
1.52
0.994
1.99e-07
NA
0.359
0.183
0.735
0.279
0.162
1.56
0.988
1.71e-06
NA
Hs 578T Torin1 1
sigmoid
sigmoid
Hs578T Torin1 1
8 1.956
0.0217
0.0183
0.598
0.0203
0.0286
0.911
0.994
1.81e-07
NA
0.0321
0.267
0.524
0.0141
0.28
0.995
0.996
8.78e-08
NA
HCC70 PI103 3 72
sigmoid
sigmoid
HCC70 PI-103 0 3 72
8 2.446
1.51
0.227
0.0983
1.57
-0.0288
1.54
0.986
2.66e-06
NA
1.48
0.303
0.906
1.15
0.168
1.59
0.976
1.42e-05
NA
HCC38 GDC-0980 1 72
sigmoid
sigmoid
HCC38 apitolisib 0 1 72
8 1.777
0.317
0.114
0.305
0.295
0.0315
0.91
0.99
9.47e-07
NA
0.623
0.354
0.761
0.219
0.315
0.951
0.989
1.26e-06
NA
Hs 578T PIK-93 3
sigmoid
sigmoid
Hs578T PIK-93 3
8 2.816
2.36
0.412
0.0884
2.23
0.033
1.2
0.994
1.87e-07
NA
1.89
0.375
0.897
1.42
0.149
1.24
0.991
8.33e-07
NA
Hs 578T Trametinib 2
sigmoid
sigmoid
Hs578T trametinib 2
8 2.483
0.00633
0.074
0.701
0.00558
0.0362
0.593
0.998
1.32e-08
NA
0.0058
0.214
0.361
0.00257
0.193
0.602
0.998
3.66e-09
NA
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