Evaluation of the sensitivities of six triple-negative breast cancer (TNBC) cell lines to 23 different PI3K/AKT/mTOR inhibitors or to a MEK inhibitor (trametinib). Dataset 2 of 2: GR metrics. - Dataset (ID:20365)

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Cell line Drug name Experimental replicate Timepoint Curve type (GR values) Curve type (relative cell counts) Experiment name Number of concentrations Cell doublings (DMSO control) GR50 GRmax GR_AOC GEC50 GRinf Hill slope (GR values) R-squared sigmoid fit (GR values) P-value sigmoid fit (GR values) R-squared flat fit (GR values) IC50 Emax AUC EC50 Einf Hill slope (relative cell counts) R-squared sigmoid fit (relative cell counts) P-value sigmoid fit (relative cell counts) R-squared flat fit (relative cell counts)
BT-20 Omipalisib 2 72
sigmoid
sigmoid
BT20 omipalisib 0 2 72
8 1.717
0.00324
-0.799
1.1
0.00361
-0.354
4.99
0.808
0.00704
NA
0.00518
0.0194
0.291
0.00429
0.111
1.34
0.968
3.16e-05
NA
BT-20 Omipalisib 3 72
sigmoid
sigmoid
BT20 omipalisib 0 3 72
8 2.586
0.00689
-0.587
0.893
0.044
-0.714
0.478
0.958
7.32e-05
NA
0.00572
0.017
0.281
0.00491
0.0669
0.945
0.983
4.7e-06
NA
Hs 578T Trametinib 2
sigmoid
sigmoid
Hs578T trametinib 2
8 2.483
0.00633
0.074
0.701
0.00558
0.0362
0.593
0.998
1.32e-08
NA
0.0058
0.214
0.361
0.00257
0.193
0.602
0.998
3.66e-09
NA
Hs 578T Trametinib 1
sigmoid
sigmoid
Hs578T trametinib 1
8 2.044
0.00353
-0.00904
0.765
0.00516
-0.0906
0.437
0.992
4.85e-07
NA
0.00661
0.238
0.385
0.00213
0.201
0.456
0.993
3e-07
NA
Hs 578T Dactolisib 3
sigmoid
sigmoid
Hs578T dactolisib 3
8 2.837
0.0118
0.0569
0.624
0.00848
0.115
0.799
0.96
6.53e-05
NA
0.00728
0.164
0.377
0.0043
0.212
1.05
0.968
3.34e-05
NA
BT-20 Omipalisib 1 72
sigmoid
sigmoid
BT20 omipalisib 0 1 72
8 2.078
0.00617
-0.729
0.985
0.0283
-0.739
0.596
0.97
2.83e-05
NA
0.00781
0.0157
0.306
0.00685
0.0597
0.96
0.988
1.57e-06
NA
Hs 578T Omipalisib 1
sigmoid
sigmoid
Hs578T omipalisib 1
8 2.079
0.00552
-0.546
0.842
0.17
-1.0
0.321
0.98
8.1e-06
NA
0.0079
0.0459
0.351
0.0079
0.0
0.369
0.984
4.12e-06
NA
BT-20 Dactolisib 2 72
sigmoid
sigmoid
BT20 dactolisib 0 2 72
8 1.727
0.00497
-0.212
0.896
0.00652
-0.186
1.17
0.995
1.45e-07
NA
0.00801
0.2
0.382
0.00505
0.211
1.19
0.994
2.07e-07
NA
BT-20 Torin2 2 72
sigmoid
sigmoid
BT20 Torin2 0 2 72
8 1.733
0.00315
-0.761
0.992
0.0484
-0.95
0.389
0.949
0.000131
NA
0.00804
0.0252
0.336
0.00642
0.0613
0.583
0.974
1.77e-05
NA
Hs 578T Trametinib 3
sigmoid
sigmoid
Hs578T trametinib 3
8 2.830
0.0128
0.0657
0.644
0.0112
0.0447
0.702
0.998
4.02e-09
NA
0.00864
0.168
0.366
0.00512
0.157
0.722
0.998
5.57e-09
NA
Hs 578T Dactolisib 2
sigmoid
sigmoid
Hs578T dactolisib 2
8 2.509
0.0128
-0.0617
0.655
0.0126
0.00741
0.79
0.974
1.78e-05
NA
0.0105
0.15
0.405
0.00638
0.203
1.04
0.985
3.67e-06
NA
BT-20 Dactolisib 3 72
sigmoid
sigmoid
BT20 dactolisib 0 3 72
8 2.420
0.0111
0.024
0.639
0.00921
0.0987
1.17
0.982
6.27e-06
NA
0.0106
0.198
0.427
0.00645
0.241
1.32
0.99
9.14e-07
NA
BT-549 Dactolisib 3 72
sigmoid
sigmoid
BT549 dactolisib 0 3 72
8 1.801
0.0058
-0.00929
0.751
0.00579
0.000747
0.866
0.994
2.41e-07
NA
0.011
0.282
0.442
0.00425
0.29
0.909
0.995
1.54e-07
NA
Hs 578T Omipalisib 2
sigmoid
sigmoid
Hs578T omipalisib 2
8 2.507
0.0155
-0.52
0.766
0.239
-1.0
0.402
0.993
3.45e-07
NA
0.0114
0.028
0.355
0.0114
0.0
0.468
0.981
6.9e-06
NA
Hs 578T Torin2 2
sigmoid
sigmoid
Hs578T Torin2 2
8 2.528
0.0153
-0.467
0.778
0.112
-0.771
0.47
0.986
2.55e-06
NA
0.0122
0.0353
0.352
0.0109
0.036
0.668
0.984
4.09e-06
NA
HCC70 Omipalisib 1 72
sigmoid
sigmoid
HCC70 omipalisib 0 1 72
8 1.358
0.00496
-0.785
1.14
0.0157
-0.775
0.812
0.989
1.34e-06
NA
0.0123
0.0486
0.349
0.011
0.0462
0.833
0.984
3.73e-06
NA
Hs 578T Dactolisib 1
sigmoid
sigmoid
Hs578T dactolisib 1
8 2.047
0.00952
-0.0606
0.691
0.00928
0.0117
0.91
0.977
1.27e-05
NA
0.0124
0.213
0.443
0.00621
0.259
1.06
0.985
3.61e-06
NA
BT-20 Torin1 2 72
sigmoid
sigmoid
BT20 Torin1 0 2 72
8 1.793
0.00766
-0.152
0.806
0.00992
-0.146
0.986
0.986
2.59e-06
NA
0.0131
0.215
0.421
0.00727
0.212
0.936
0.988
1.92e-06
NA
BT-549 Dactolisib 2 72
sigmoid
sigmoid
BT549 dactolisib 0 2 72
8 1.889
0.00968
-0.00862
0.677
0.00884
0.0542
1.27
0.985
3.3e-06
NA
0.0134
0.266
0.48
0.00701
0.305
1.45
0.988
1.53e-06
NA
HCC70 Omipalisib 2 72
sigmoid
sigmoid
HCC70 omipalisib 0 2 72
8 1.682
0.00746
-0.705
1.01
0.0241
-0.703
0.749
0.991
6.69e-07
NA
0.0135
0.0399
0.359
0.0121
0.0458
0.852
0.989
1.45e-06
NA
HCC38 Dactolisib 2 72
sigmoid
sigmoid
HCC38 dactolisib 0 2 72
8 2.120
0.0118
-0.0557
0.668
0.0118
-0.00134
0.785
0.98
7.61e-06
NA
0.0145
0.204
0.447
0.00701
0.245
0.927
0.988
1.88e-06
NA
Hs 578T Omipalisib 3
sigmoid
sigmoid
Hs578T omipalisib 3
8 2.869
0.0255
-0.107
0.615
0.0533
-0.22
0.494
0.99
8.79e-07
NA
0.0145
0.0989
0.392
0.0102
0.0968
0.62
0.993
3.4e-07
NA
BT-20 Torin2 3 72
sigmoid
sigmoid
BT20 Torin2 0 3 72
8 2.458
0.019
-0.64
0.751
0.234
-1.0
0.438
0.959
6.92e-05
NA
0.0147
0.0148
0.379
0.0123
0.0598
0.727
0.977
1.28e-05
NA
HCC70 Omipalisib 3 72
sigmoid
sigmoid
HCC70 omipalisib 0 3 72
8 2.458
0.0158
-0.404
0.771
0.0319
-0.379
0.8
0.99
8.95e-07
NA
0.0148
0.051
0.376
0.0127
0.0733
1.02
0.996
4.59e-08
NA
BT-549 Dactolisib 1 72
sigmoid
sigmoid
BT549 dactolisib 0 1 72
8 1.840
0.00961
-0.00769
0.683
0.00888
0.0384
1.01
0.985
3.53e-06
NA
0.0161
0.275
0.482
0.0068
0.303
1.09
0.987
2.38e-06
NA
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