Evaluation of the sensitivities of six triple-negative breast cancer (TNBC) cell lines to 23 different PI3K/AKT/mTOR inhibitors or to a MEK inhibitor (trametinib). Dataset 2 of 2: GR metrics. - Dataset (ID:20365)

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Cell line Drug name Experimental replicate Timepoint Curve type (GR values) Curve type (relative cell counts) Experiment name Number of concentrations Cell doublings (DMSO control) GR50 GRmax GR_AOC GEC50 GRinf Hill slope (GR values) R-squared sigmoid fit (GR values) P-value sigmoid fit (GR values) R-squared flat fit (GR values) IC50 Emax AUC EC50 Einf Hill slope (relative cell counts) R-squared sigmoid fit (relative cell counts) P-value sigmoid fit (relative cell counts) R-squared flat fit (relative cell counts)
BT-20 ZSTK474 3 72
sigmoid
sigmoid
BT20 ZSTK474 0 3 72
8 2.609
0.457
-0.00222
0.296
0.783
-0.31
0.895
0.982
5.76e-06
NA
0.422
0.163
0.702
0.422
0.0
0.82
0.971
2.52e-05
NA
BT-549 PI103 3 72
sigmoid
sigmoid
BT549 PI-103 0 3 72
8 1.758
0.16
0.00249
0.391
0.166
-0.0225
1.12
0.989
1.19e-06
NA
0.279
0.297
0.704
0.134
0.28
1.12
0.985
3.23e-06
NA
HCC70 BX-912 2 72
sigmoid
sigmoid
HCC70 BX-912 0 2 72
8 1.693
1.25
0.00257
0.0619
1.25
-0.00649
5.0
0.971
2.55e-05
NA
1.44
0.311
0.961
1.2
0.306
5.0
0.956
8.35e-05
NA
BT-549 Dactolisib 1 72
sigmoid
sigmoid
BT549 dactolisib 0 1 72
8 1.840
0.00961
-0.00769
0.683
0.00888
0.0384
1.01
0.985
3.53e-06
NA
0.0161
0.275
0.482
0.0068
0.303
1.09
0.987
2.38e-06
NA
BT-549 Dactolisib 2 72
sigmoid
sigmoid
BT549 dactolisib 0 2 72
8 1.889
0.00968
-0.00862
0.677
0.00884
0.0542
1.27
0.985
3.3e-06
NA
0.0134
0.266
0.48
0.00701
0.305
1.45
0.988
1.53e-06
NA
Hs 578T Trametinib 1
sigmoid
sigmoid
Hs578T trametinib 1
8 2.044
0.00353
-0.00904
0.765
0.00516
-0.0906
0.437
0.992
4.85e-07
NA
0.00661
0.238
0.385
0.00213
0.201
0.456
0.993
3e-07
NA
BT-549 Dactolisib 3 72
sigmoid
sigmoid
BT549 dactolisib 0 3 72
8 1.801
0.0058
-0.00929
0.751
0.00579
0.000747
0.866
0.994
2.41e-07
NA
0.011
0.282
0.442
0.00425
0.29
0.909
0.995
1.54e-07
NA
HCC70 PI103 1 72
sigmoid
sigmoid
HCC70 PI-103 0 1 72
8 1.305
1.04
-0.0102
0.104
1.14
-0.107
2.26
0.957
7.9e-05
NA
1.83
0.399
0.938
1.08
0.349
2.28
0.949
0.000133
NA
HCC38 Torin1 1 72
sigmoid
sigmoid
HCC38 Torin1 0 1 72
8 1.688
0.0287
-0.0113
0.569
0.0278
0.013
0.843
0.993
4.14e-07
NA
0.0653
0.304
0.585
0.0204
0.325
0.9
0.992
4.53e-07
NA
BT-20 PI103 1 72
sigmoid
sigmoid
BT20 PI-103 0 1 72
8 1.924
0.646
-0.0114
0.16
0.659
-0.0268
2.6
0.978
1.1e-05
NA
0.753
0.258
0.883
0.579
0.252
2.68
0.964
4.79e-05
NA
Hs 578T BX-912 3
sigmoid
sigmoid
Hs578T BX-912 3
8 2.805
1.04
0.0121
0.125
1.09
-0.0661
2.36
0.992
4.22e-07
NA
0.936
0.148
0.883
0.841
0.116
2.45
0.982
5.7e-06
NA
HCC70 AZD-6482 1 72
sigmoid
sigmoid
HCC70 AZD6482 0 1 72
8 1.368
0.0982
0.0128
0.462
0.205
-0.212
0.481
0.975
1.49e-05
NA
0.767
0.394
0.704
0.121
0.305
0.509
0.973
1.9e-05
NA
BT-20 PI103 3 72
sigmoid
sigmoid
BT20 PI-103 0 3 72
8 2.496
0.373
0.0139
0.282
0.387
-0.0286
1.52
0.994
1.99e-07
NA
0.359
0.183
0.735
0.279
0.162
1.56
0.988
1.71e-06
NA
Hs 578T Torin1 1
sigmoid
sigmoid
Hs578T Torin1 1
8 1.956
0.0217
0.0183
0.598
0.0203
0.0286
0.911
0.994
1.81e-07
NA
0.0321
0.267
0.524
0.0141
0.28
0.995
0.996
8.78e-08
NA
HCC38 GDC-0980 3 72
sigmoid
sigmoid
HCC38 apitolisib 0 3 72
8 1.437
0.371
-0.0189
0.29
0.513
-0.179
0.946
0.993
3.35e-07
NA
0.96
0.359
0.808
0.393
0.295
0.998
0.993
3.51e-07
NA
Hs 578T BX-912 2
sigmoid
sigmoid
Hs578T BX-912 2
8 2.540
1.07
-0.019
0.174
1.79
-0.489
1.33
0.998
6.37e-09
NA
1.01
0.164
0.828
1.01
0.0
1.4
0.996
7.64e-08
NA
BT-549 PI103 2 72
sigmoid
sigmoid
BT549 PI-103 0 2 72
8 1.893
0.218
0.0201
0.344
0.229
-0.0262
1.08
0.997
2.55e-08
NA
0.326
0.28
0.725
0.169
0.261
1.13
0.996
6.2e-08
NA
Hs 578T PI103 2
sigmoid
sigmoid
Hs578T PI-103 2
8 2.503
0.223
-0.0213
0.356
0.303
-0.15
0.858
0.999
7.33e-10
NA
0.206
0.167
0.661
0.152
0.121
0.921
0.999
1.9e-09
NA
HCC38 WYE-125132 3 72
sigmoid
sigmoid
HCC38 WYE-132 0 3 72
8 1.449
0.0494
-0.0216
0.518
0.0504
-0.0117
1.18
0.998
9.69e-09
NA
0.128
0.355
0.662
0.0441
0.361
1.2
0.998
9.53e-09
NA
BT-20 ZSTK474 1 72
sigmoid
sigmoid
BT20 ZSTK474 0 1 72
8 1.940
0.788
0.0217
0.122
0.819
-0.0395
1.99
0.957
7.76e-05
NA
0.942
0.272
0.913
0.677
0.249
2.09
0.934
0.000293
NA
HCC70 PI103 2 72
sigmoid
sigmoid
HCC70 PI-103 0 2 72
8 1.739
1.19
0.0238
0.151
2.67
-0.766
1.15
0.997
2.59e-08
NA
1.68
0.312
0.885
1.68
0.0
1.21
0.996
6.86e-08
NA
BT-20 Dactolisib 3 72
sigmoid
sigmoid
BT20 dactolisib 0 3 72
8 2.420
0.0111
0.024
0.639
0.00921
0.0987
1.17
0.982
6.27e-06
NA
0.0106
0.198
0.427
0.00645
0.241
1.32
0.99
9.14e-07
NA
BT-20 AZD-6482 2 72
sigmoid
sigmoid
BT20 AZD6482 0 2 72
8 1.645
0.581
0.0253
0.303
3.86
-1.0
0.58
0.904
0.000884
NA
1.34
0.333
0.772
1.34
0.0
0.582
0.864
0.0025
NA
BT-549 Torin1 3 72
sigmoid
sigmoid
BT549 Torin1 0 3 72
8 1.757
0.0123
0.026
0.659
0.0112
0.0466
1.02
0.997
3.77e-08
NA
0.0235
0.309
0.513
0.00878
0.322
1.05
0.997
1.65e-08
NA
BT-549 GDC-0980 2 72
sigmoid
sigmoid
BT549 apitolisib 0 2 72
8 1.939
0.189
0.0264
0.357
0.193
-0.011
1.04
0.997
2.98e-08
NA
0.278
0.274
0.71
0.142
0.257
1.07
0.997
3.64e-08
NA
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