Evaluation of the sensitivities of six triple-negative breast cancer (TNBC) cell lines to 23 different PI3K/AKT/mTOR inhibitors or to a MEK inhibitor (trametinib). Dataset 2 of 2: GR metrics. - Dataset (ID:20365)

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Cell line Drug name Experimental replicate Timepoint Curve type (GR values) Curve type (relative cell counts) Experiment name Number of concentrations Cell doublings (DMSO control) GR50 GRmax GR_AOC GEC50 GRinf Hill slope (GR values) R-squared sigmoid fit (GR values) P-value sigmoid fit (GR values) R-squared flat fit (GR values) IC50 Emax AUC EC50 Einf Hill slope (relative cell counts) R-squared sigmoid fit (relative cell counts) P-value sigmoid fit (relative cell counts) R-squared flat fit (relative cell counts)
HCC70 PI103 1 72
sigmoid
sigmoid
HCC70 PI-103 0 1 72
8 1.305
1.04
-0.0102
0.104
1.14
-0.107
2.26
0.957
7.9e-05
NA
1.83
0.399
0.938
1.08
0.349
2.28
0.949
0.000133
NA
HCC70 ZSTK474 1 72
sigmoid
sigmoid
HCC70 ZSTK474 0 1 72
8 1.332
0.167
-0.265
0.366
0.201
-0.206
1.85
0.975
1.56e-05
NA
0.289
0.264
0.782
0.182
0.299
1.96
0.971
2.35e-05
NA
HCC70 AZD8055 1 72
sigmoid
sigmoid
HCC70 AZD8055 0 1 72
8 1.339
0.0485
0.242
0.442
0.0243
0.26
1.06
0.976
1.32e-05
NA
Inf
0.529
0.721
0.0222
0.54
1.08
0.974
1.81e-05
NA
HCC38 AS605240 3 72
flat
flat
HCC38 AS-605240 0 3 72
8 1.343
Inf
0.958
-0.0162
0.0
0.958
0.01
-0.233
1.0
1.01
Inf
0.972
1.01
0.0
0.972
0.01
-0.235
1.0
1.01
HCC70 Torin1 1 72
sigmoid
sigmoid
HCC70 Torin1 0 1 72
8 1.345
0.0472
0.15
0.487
0.0311
0.149
0.849
0.973
1.89e-05
NA
0.93
0.475
0.693
0.0276
0.475
0.854
0.973
2.05e-05
NA
HCC70 KIN001-244 1 72
flat
flat
HCC70 KIN001-244 0 1 72
8 1.350
Inf
0.889
0.00722
0.0
0.889
0.01
0.616
0.0568
0.988
Inf
0.926
0.995
0.0
0.926
0.01
0.612
0.0584
0.992
HCC70 GDC-0980 1 72
sigmoid
sigmoid
HCC70 apitolisib 0 1 72
8 1.350
0.211
-0.312
0.362
0.339
-0.362
1.15
0.985
3.24e-06
NA
0.441
0.237
0.779
0.266
0.236
1.26
0.985
3.31e-06
NA
HCC70 Omipalisib 1 72
sigmoid
sigmoid
HCC70 omipalisib 0 1 72
8 1.358
0.00496
-0.785
1.14
0.0157
-0.775
0.812
0.989
1.34e-06
NA
0.0123
0.0486
0.349
0.011
0.0462
0.833
0.984
3.73e-06
NA
HCC70 Torin2 1 72
sigmoid
sigmoid
HCC70 Torin2 0 1 72
8 1.364
0.0288
-0.732
0.772
0.183
-1.0
0.594
0.991
6.58e-07
NA
0.088
0.0644
0.539
0.088
0.0
0.622
0.988
1.95e-06
NA
HCC70 Everolimus 1 72
flat
flat
HCC70 everolimus 0 1 72
8 1.366
Inf
0.569
0.354
0.0
0.569
0.01
0.623
0.0534
0.643
Inf
0.718
0.766
0.0
0.718
0.01
0.62
0.0547
0.765
HCC70 AZD-6482 1 72
sigmoid
sigmoid
HCC70 AZD6482 0 1 72
8 1.368
0.0982
0.0128
0.462
0.205
-0.212
0.481
0.975
1.49e-05
NA
0.767
0.394
0.704
0.121
0.305
0.509
0.973
1.9e-05
NA
HCC70 Buparlisib 1 72
sigmoid
sigmoid
HCC70 buparlisib 0 1 72
8 1.374
0.608
-0.494
0.231
1.27
-0.9
1.4
0.98
7.6e-06
NA
0.988
0.151
0.861
0.98
0.00578
1.46
0.973
1.91e-05
NA
HCC70 TGX221 1 72
sigmoid
sigmoid
HCC70 TGX-221 0 1 72
8 1.381
0.539
0.344
0.244
0.245
0.278
1.03
0.986
2.58e-06
NA
Inf
0.578
0.84
0.229
0.536
1.02
0.986
2.87e-06
NA
HCC38 PIK-93 3 72
sigmoid
sigmoid
HCC38 PIK-93 0 3 72
8 1.382
5.05
0.598
0.061
2.34
0.358
1.63
0.919
0.000533
NA
Inf
0.734
0.959
2.23
0.586
1.64
0.914
0.000645
NA
HCC70 WYE-125132 1 72
sigmoid
sigmoid
HCC70 WYE-132 0 1 72
8 1.382
0.0518
0.346
0.418
0.0175
0.348
1.1
0.985
3.58e-06
NA
Inf
0.579
0.727
0.0165
0.579
1.09
0.983
4.63e-06
NA
HCC70 Alpelisib 1 72
sigmoid
sigmoid
HCC70 alpelisib 0 1 72
8 1.383
4.4
0.574
0.105
20.4
-1.0
0.717
0.78
0.0106
NA
11.9
0.718
0.929
11.9
0.0
0.732
0.768
0.0124
NA
HCC70 CAL-101 1 72
sigmoid
sigmoid
HCC70 idelalisib 0 1 72
8 1.384
2.78
0.485
0.0894
0.883
0.424
1.65
0.972
2.11e-05
NA
Inf
0.662
0.941
0.846
0.626
1.66
0.97
2.79e-05
NA
HCC38 Torin2 3 72
sigmoid
sigmoid
HCC38 Torin2 0 3 72
8 1.385
0.013
-0.624
0.855
0.0547
-0.706
0.615
0.996
8.13e-08
NA
0.0407
0.0986
0.484
0.0311
0.0829
0.669
0.997
3.31e-08
NA
HCC70 AS605240 1 72
sigmoid
sigmoid
HCC70 AS-605240 0 1 72
8 1.387
10.4
0.487
0.159
0.247
0.497
1.34
0.963
5.14e-05
NA
Inf
0.663
0.894
0.23
0.672
1.39
0.961
6.01e-05
NA
HCC70 XL147 1 72
flat
flat
HCC70 pilaralisib 0 1 72
8 1.396
Inf
1.05
-0.0406
0.0
1.05
0.01
-0.285
1.0
1.03
Inf
1.04
1.03
0.0
1.04
0.01
-0.295
1.0
1.02
HCC38 Alpelisib 3 72
flat
flat
HCC38 alpelisib 0 3 72
8 1.398
Inf
0.75
0.0995
0.0
0.75
0.01
0.141
0.634
0.883
Inf
0.829
0.932
0.0
0.829
0.01
0.113
0.698
0.92
HCC70 Dactolisib 1 72
sigmoid
sigmoid
HCC70 dactolisib 0 1 72
8 1.400
0.0808
-0.0667
0.501
3.34
-1.0
0.295
0.963
5.02e-05
NA
0.753
0.344
0.673
0.753
0.0
0.308
0.962
5.37e-05
NA
HCC70 Pictilisib 1 72
sigmoid
sigmoid
HCC70 pictilisib 0 1 72
8 1.409
0.408
-0.099
0.284
0.578
-0.245
1.14
0.996
7.62e-08
NA
0.888
0.325
0.816
0.477
0.261
1.19
0.995
1.2e-07
NA
HCC70 Sirolimus 1 72
sigmoid
sigmoid
HCC70 rapamycin 0 1 72
8 1.416
37.6
0.533
0.397
0.00426
0.298
0.1
0.742
0.0172
NA
125000000.0
0.687
0.732
0.00186
0.541
0.1
0.74
0.0175
NA
HCC38 AZD8055 3 72
sigmoid
sigmoid
HCC38 AZD8055 0 3 72
8 1.417
0.0464
0.0327
0.53
0.0463
0.000983
1.04
0.997
4.27e-08
NA
0.157
0.392
0.658
0.041
0.372
1.02
0.996
5.78e-08
NA
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