Evaluation of the sensitivities of six triple-negative breast cancer (TNBC) cell lines to 23 different PI3K/AKT/mTOR inhibitors or to a MEK inhibitor (trametinib). Dataset 2 of 2: GR metrics. - Dataset (ID:20365)

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  • Page 1 of 18
  • 1 to 25 of 432 records
Cell line Drug name Experimental replicate Timepoint Curve type (GR values) Curve type (relative cell counts) Experiment name Number of concentrations Cell doublings (DMSO control) GR50 GRmax GR_AOC GEC50 GRinf Hill slope (GR values) R-squared sigmoid fit (GR values) P-value sigmoid fit (GR values) R-squared flat fit (GR values) IC50 Emax AUC EC50 Einf Hill slope (relative cell counts) R-squared sigmoid fit (relative cell counts) P-value sigmoid fit (relative cell counts) R-squared flat fit (relative cell counts)
Hs 578T Alpelisib 3
sigmoid
sigmoid
Hs578T alpelisib 3
8 2.856
Inf
0.712
0.0759
0.872
0.616
0.828
0.963
5.21e-05
NA
Inf
0.641
0.901
0.65
0.553
0.853
0.955
8.85e-05
NA
BT-20 Alpelisib 2 72
sigmoid
sigmoid
BT20 alpelisib 0 2 72
8 1.692
0.253
-0.0994
0.405
2.25
-1.0
0.503
0.835
0.00451
NA
0.612
0.259
0.698
0.612
0.0
0.507
0.764
0.0131
NA
HCC1806 Alpelisib 1 72
flat
flat
HCC1806 alpelisib 0 1 72
8 2.771
Inf
0.918
0.0583
0.0
0.918
0.01
-0.337
1.0
0.94
Inf
0.891
0.921
0.0
0.891
0.01
-0.351
1.0
0.919
Hs 578T Alpelisib 2
flat
flat
Hs578T alpelisib 2
8 2.513
Inf
0.668
0.131
0.0
0.668
0.01
0.599
0.0647
0.856
Inf
0.634
0.847
0.0
0.634
0.01
0.541
0.0969
0.833
HCC1806 Alpelisib 2 72
flat
flat
HCC1806 alpelisib 0 2 72
8 2.856
Inf
0.921
0.0566
0.0
0.921
0.01
-0.336
1.0
0.941
Inf
0.891
0.921
0.0
0.891
0.01
-0.351
1.0
0.919
BT-20 Alpelisib 3 72
sigmoid
sigmoid
BT20 alpelisib 0 3 72
8 2.541
1.21
0.199
0.21
5.83
-1.0
0.697
0.881
0.00167
NA
1.12
0.272
0.775
1.12
0.0
0.764
0.791
0.00916
NA
HCC38 Alpelisib 3 72
flat
flat
HCC38 alpelisib 0 3 72
8 1.398
Inf
0.75
0.0995
0.0
0.75
0.01
0.141
0.634
0.883
Inf
0.829
0.932
0.0
0.829
0.01
0.113
0.698
0.92
HCC70 Alpelisib 2 72
flat
flat
HCC70 alpelisib 0 2 72
8 1.799
Inf
0.748
0.0777
0.0
0.748
0.01
0.00864
0.974
0.907
Inf
0.785
0.932
0.0
0.785
0.01
0.00534
0.984
0.919
HCC38 Alpelisib 2 72
flat
flat
HCC38 alpelisib 0 2 72
8 2.086
Inf
0.848
0.0559
0.0
0.848
0.01
-0.0371
1.0
0.931
Inf
0.848
0.944
0.0
0.848
0.01
-0.0359
1.0
0.932
Hs 578T Alpelisib 1
sigmoid
sigmoid
Hs578T alpelisib 1
8 2.097
2.3
0.449
0.205
42.0
-1.0
0.378
0.954
9.56e-05
NA
3.9
0.508
0.803
3.9
0.0
0.401
0.94
0.000216
NA
BT-549 Alpelisib 2 72
sigmoid
sigmoid
BT549 alpelisib 0 2 72
8 1.927
Inf
0.832
0.0409
4.24
0.663
0.548
0.706
0.0254
NA
Inf
0.844
0.962
4.26
0.686
0.542
0.696
0.0282
NA
HCC1806 Alpelisib 3 72
flat
flat
HCC1806 alpelisib 0 3 72
8 3.224
Inf
0.93
0.0502
0.0
0.93
0.01
-0.335
1.0
0.948
Inf
0.891
0.921
0.0
0.891
0.01
-0.351
1.0
0.919
BT-549 Alpelisib 1 72
flat
flat
BT549 alpelisib 0 1 72
8 1.822
Inf
0.747
0.0781
0.0
0.747
0.01
0.439
0.176
0.914
Inf
0.782
0.931
0.0
0.782
0.01
0.415
0.2
0.925
HCC70 Alpelisib 1 72
sigmoid
sigmoid
HCC70 alpelisib 0 1 72
8 1.383
4.4
0.574
0.105
20.4
-1.0
0.717
0.78
0.0106
NA
11.9
0.718
0.929
11.9
0.0
0.732
0.768
0.0124
NA
BT-549 Alpelisib 3 72
flat
flat
BT549 alpelisib 0 3 72
8 1.743
Inf
0.817
0.068
0.0
0.817
0.01
-0.0192
1.0
0.915
Inf
0.846
0.942
0.0
0.846
0.01
-0.0162
1.0
0.928
HCC38 Alpelisib 1 72
flat
flat
HCC38 alpelisib 0 1 72
8 1.738
Inf
0.757
0.0835
0.0
0.757
0.01
0.593
0.0674
0.909
Inf
0.798
0.929
0.0
0.798
0.01
0.579
0.0744
0.923
HCC70 Alpelisib 3 72
flat
flat
HCC70 alpelisib 0 3 72
8 2.465
Inf
0.859
0.027
0.0
0.859
0.01
0.407
0.209
0.961
Inf
0.835
0.968
0.0
0.835
0.01
0.394
0.222
0.954
BT-20 Alpelisib 1 72
sigmoid
sigmoid
BT20 alpelisib 0 1 72
8 2.077
1.14
0.046
0.196
3.52
-1.0
0.977
0.966
4.1e-05
NA
1.32
0.26
0.825
1.32
0.0
1.13
0.942
0.000194
NA
HCC70 AS605240 3 72
sigmoid
sigmoid
HCC70 AS-605240 0 3 72
8 2.447
Inf
0.58
0.112
0.427
0.549
1.18
0.985
3.24e-06
NA
Inf
0.562
0.877
0.345
0.544
1.24
0.982
6.14e-06
NA
BT-549 AS605240 2 72
flat
flat
BT549 AS-605240 0 2 72
8 1.961
Inf
0.91
0.0479
0.0
0.91
0.01
0.414
0.201
0.949
Inf
0.914
0.954
0.0
0.914
0.01
0.418
0.197
0.951
HCC1806 AS605240 1 72
sigmoid
sigmoid
HCC1806 AS-605240 0 1 72
8 2.728
Inf
0.911
0.0128
0.569
0.91
2.8
0.936
0.000262
NA
Inf
0.883
0.983
0.559
0.882
2.81
0.931
0.000333
NA
HCC70 AS605240 1 72
sigmoid
sigmoid
HCC70 AS-605240 0 1 72
8 1.387
10.4
0.487
0.159
0.247
0.497
1.34
0.963
5.14e-05
NA
Inf
0.663
0.894
0.23
0.672
1.39
0.961
6.01e-05
NA
HCC70 AS605240 2 72
sigmoid
sigmoid
HCC70 AS-605240 0 2 72
8 1.771
6.13
0.558
0.126
1.21
0.339
0.698
0.981
7.24e-06
NA
785.0
0.643
0.894
0.946
0.496
0.708
0.978
1.04e-05
NA
HCC38 AS605240 1 72
sigmoid
sigmoid
HCC38 AS-605240 0 1 72
8 1.744
Inf
0.734
0.0803
0.448
0.691
0.881
0.969
2.92e-05
NA
Inf
0.78
0.932
0.405
0.748
0.895
0.967
3.48e-05
NA
BT-549 AS605240 3 72
sigmoid
sigmoid
BT549 AS-605240 0 3 72
8 1.796
Inf
0.863
0.066
4.3
0.721
0.307
0.896
0.00112
NA
Inf
0.881
0.942
4.35
0.756
0.302
0.894
0.00118
NA
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