Evaluation of the sensitivities of six triple-negative breast cancer (TNBC) cell lines to 23 different PI3K/AKT/mTOR inhibitors or to a MEK inhibitor (trametinib). Dataset 2 of 2: GR metrics. - Dataset (ID:20365)

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Cell line Drug name Experimental replicate Timepoint Curve type (GR values) Curve type (relative cell counts) Experiment name Number of concentrations Cell doublings (DMSO control) GR50 GRmax GR_AOC GEC50 GRinf Hill slope (GR values) R-squared sigmoid fit (GR values) P-value sigmoid fit (GR values) R-squared flat fit (GR values) IC50 Emax AUC EC50 Einf Hill slope (relative cell counts) R-squared sigmoid fit (relative cell counts) P-value sigmoid fit (relative cell counts) R-squared flat fit (relative cell counts)
BT-549 Omipalisib 2 72
sigmoid
sigmoid
BT549 omipalisib 0 2 72
8 1.990
0.0104
-0.291
0.751
0.026
-0.32
0.542
0.966
4.09e-05
NA
0.0175
0.127
0.422
0.011
0.118
0.58
0.953
0.000102
NA
Hs 578T TGX221 3
sigmoid
sigmoid
Hs578T TGX-221 3
8 2.818
24.2
0.885
0.0148
88.9
-1.0
0.843
0.958
7.66e-05
NA
23.4
0.846
0.98
23.4
0.0
0.862
0.953
0.000103
NA
HCC38 MK2206 1 72
sigmoid
sigmoid
HCC38 MK-2206 0 1 72
8 1.789
19.4
0.698
0.0995
320.0
-0.949
0.38
0.956
8.33e-05
NA
61.8
0.746
0.914
61.8
0.0
0.386
0.951
0.000115
NA
HCC70 PI103 1 72
sigmoid
sigmoid
HCC70 PI-103 0 1 72
8 1.305
1.04
-0.0102
0.104
1.14
-0.107
2.26
0.957
7.9e-05
NA
1.83
0.399
0.938
1.08
0.349
2.28
0.949
0.000133
NA
BT-549 PIK-93 2 72
sigmoid
sigmoid
BT549 PIK-93 0 2 72
8 1.983
7.03
0.687
0.0641
29.9
-1.0
0.759
0.956
8.81e-05
NA
10.4
0.713
0.939
10.4
0.0
0.788
0.949
0.000136
NA
BT-549 MK2206 3 72
sigmoid
sigmoid
BT549 MK-2206 0 3 72
8 1.685
Inf
0.714
0.131
0.123
0.711
3.44
0.953
0.000102
NA
Inf
0.771
0.895
0.123
0.768
3.25
0.949
0.000136
NA
HCC70 Trametinib 2 72
sigmoid
sigmoid
HCC70 trametinib 0 2 72
8 1.721
0.506
0.504
0.395
0.00469
0.467
0.581
0.944
0.000179
NA
Inf
0.612
0.687
0.00389
0.585
0.57
0.948
0.000138
NA
BT-20 Buparlisib 2 72
sigmoid
sigmoid
BT20 buparlisib 0 2 72
8 1.743
0.334
-0.45
0.391
0.844
-0.82
1.05
0.972
2.21e-05
NA
0.487
0.105
0.718
0.487
0.0
1.12
0.948
0.000142
NA
BT-20 MK2206 2 72
sigmoid
sigmoid
BT20 MK-2206 0 2 72
8 1.739
0.823
0.0896
0.246
4.34
-1.0
0.661
0.965
4.36e-05
NA
1.47
0.348
0.806
1.47
0.0
0.715
0.947
0.000145
NA
HCC38 Trametinib 1 72
sigmoid
sigmoid
HCC38 trametinib 0 1 72
8 1.733
0.162
0.196
0.407
0.173
-0.0184
0.559
0.948
0.000139
NA
0.568
0.41
0.686
0.161
0.234
0.501
0.947
0.000151
NA
BT-549 AZD-6482 2 72
sigmoid
sigmoid
BT549 AZD6482 0 2 72
8 1.973
9.15
0.635
0.112
120.0
-1.0
0.426
0.951
0.000115
NA
19.4
0.672
0.895
19.4
0.0
0.437
0.946
0.000154
NA
BT-20 Alpelisib 1 72
sigmoid
sigmoid
BT20 alpelisib 0 1 72
8 2.077
1.14
0.046
0.196
3.52
-1.0
0.977
0.966
4.1e-05
NA
1.32
0.26
0.825
1.32
0.0
1.13
0.942
0.000194
NA
Hs 578T CAL-101 1
sigmoid
sigmoid
Hs578T idelalisib 1
8 2.050
27.9
0.72
0.0764
4.56
0.356
0.688
0.945
0.000168
NA
18.7
0.734
0.925
18.7
0.0
0.568
0.941
0.000203
NA
Hs 578T Alpelisib 1
sigmoid
sigmoid
Hs578T alpelisib 1
8 2.097
2.3
0.449
0.205
42.0
-1.0
0.378
0.954
9.56e-05
NA
3.9
0.508
0.803
3.9
0.0
0.401
0.94
0.000216
NA
BT-549 Trametinib 3 72
sigmoid
sigmoid
BT549 trametinib 0 3 72
8 1.755
Inf
0.553
0.223
0.107
0.505
0.899
0.942
0.000194
NA
Inf
0.642
0.817
0.104
0.595
0.804
0.938
0.000236
NA
HCC70 TGX221 2 72
sigmoid
sigmoid
HCC70 TGX-221 0 2 72
8 1.786
1.77
0.467
0.233
0.531
0.227
0.503
0.948
0.000139
NA
5.85
0.575
0.806
3.44
0.0897
0.372
0.937
0.000249
NA
BT-20 AZD8055 2 72
sigmoid
sigmoid
BT20 AZD8055 0 2 72
8 1.951
0.00909
0.155
0.651
0.00651
0.115
0.785
0.936
0.000258
NA
0.0185
0.343
0.477
0.00469
0.311
0.706
0.934
0.000289
NA
BT-20 ZSTK474 1 72
sigmoid
sigmoid
BT20 ZSTK474 0 1 72
8 1.940
0.788
0.0217
0.122
0.819
-0.0395
1.99
0.957
7.76e-05
NA
0.942
0.272
0.913
0.677
0.249
2.09
0.934
0.000293
NA
BT-549 Trametinib 1 72
sigmoid
sigmoid
BT549 trametinib 0 1 72
8 1.812
Inf
0.596
0.202
0.131
0.523
0.61
0.959
6.65e-05
NA
28.3
0.664
0.828
3.47
0.254
0.337
0.933
0.000305
NA
HCC38 Everolimus 3 72
sigmoid
sigmoid
HCC38 everolimus 0 3 72
8 1.437
5.11
0.511
0.429
0.000567
0.299
0.1
0.934
0.000284
NA
573000000.0
0.668
0.707
0.000349
0.53
0.1
0.932
0.000308
NA
BT-549 CAL-101 2 72
sigmoid
sigmoid
BT549 idelalisib 0 2 72
8 1.975
Inf
0.792
0.0561
4.65
0.526
0.693
0.933
0.000307
NA
43.0
0.805
0.946
43.0
0.0
0.548
0.932
0.000314
NA
HCC1806 AS605240 2 72
sigmoid
sigmoid
HCC1806 AS-605240 0 2 72
8 2.813
Inf
0.913
0.0124
0.569
0.913
2.8
0.936
0.000261
NA
Inf
0.883
0.983
0.559
0.882
2.81
0.931
0.000333
NA
HCC1806 AS605240 1 72
sigmoid
sigmoid
HCC1806 AS-605240 0 1 72
8 2.728
Inf
0.911
0.0128
0.569
0.91
2.8
0.936
0.000262
NA
Inf
0.883
0.983
0.559
0.882
2.81
0.931
0.000333
NA
HCC1806 AS605240 3 72
sigmoid
sigmoid
HCC1806 AS-605240 0 3 72
8 3.181
Inf
0.923
0.011
0.57
0.923
2.81
0.936
0.000257
NA
Inf
0.883
0.983
0.559
0.882
2.81
0.931
0.000333
NA
HCC38 AS605240 2 72
sigmoid
sigmoid
HCC38 AS-605240 0 2 72
8 2.200
17.4
0.642
0.114
4.07
0.256
0.493
0.936
0.000265
NA
46.2
0.648
0.882
1.68
0.411
0.522
0.929
0.000356
NA
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