Breast Cancer Deubiquitinating Enzyme (DUB) Inhibitor Profiling: Fixed-cell GR measures of 21 breast cell lines to 32 small molecule perturbagens. Dataset 2 of 2: Calculated dose response metrics. - Dataset (ID:20351)
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Cell | Small Molecule | Treatment Duration | GR50 | GRmax | GR_AOC | GEC50 | GRinf | hGR |
---|---|---|---|---|---|---|---|---|
PDX1328 | z-VAE(OMe)-fmk | 72 | inf | 1.0551 | 0.0297 | 0.0000 | 0.9884 | 0.0100 |
MDA-MB-231 | z-VAE(OMe)-fmk | 72 | inf | 0.9382 | 0.0024 | 0.0000 | 0.9922 | 0.0100 |
MCF7 | z-VAE(OMe)-fmk | 72 | inf | 1.0118 | -0.0177 | 0.0000 | 1.0000 | 0.0100 |
PDX1258 | z-VAE(OMe)-fmk | 72 | inf | 0.9262 | 0.0692 | 0.0000 | 0.9516 | 0.0100 |
SK-BR-3 | z-VAE(OMe)-fmk | 72 | inf | 0.9573 | 0.0430 | 0.0000 | 0.9575 | 0.0100 |
HCC1806 | z-VAE(OMe)-fmk | 72 | inf | 0.9581 | 0.0231 | 0.0000 | 0.9783 | 0.0100 |
MCF 10A | z-VAE(OMe)-fmk | 72 | inf | 0.9979 | 0.0012 | 0.0000 | 0.9999 | 0.0100 |
HCC202 | z-VAE(OMe)-fmk | 72 | inf | 1.0085 | 0.0421 | 0.0000 | 0.9739 | 0.0100 |
HCC1954 | z-VAE(OMe)-fmk | 72 | inf | 1.0513 | 0.0385 | 0.0000 | 0.9751 | 0.0100 |
MDA-MB-361 | z-VAE(OMe)-fmk | 72 | inf | 0.9096 | 0.0284 | 0.0000 | 0.9738 | 0.0100 |
PDXHCI002 | z-VAE(OMe)-fmk | 72 | inf | 0.9278 | 0.0585 | 0.0000 | 0.9445 | 0.0100 |
BT-549 | z-VAE(OMe)-fmk | 72 | inf | 0.9727 | 0.0182 | 0.0000 | 0.9828 | 0.0100 |
Hs 578T | z-VAE(OMe)-fmk | 72 | inf | 0.9948 | 0.0176 | 0.0000 | 0.9832 | 0.0100 |
T47D | z-VAE(OMe)-fmk | 72 | inf | 0.9468 | 0.0261 | 0.0000 | 0.9749 | 0.0100 |
HCC1500 | z-VAE(OMe)-fmk | 72 | inf | 1.1021 | 0.0136 | 0.0000 | 1.0000 | 0.0100 |
CAMA-1 | z-VAE(OMe)-fmk | 72 | inf | 0.9619 | 0.0262 | 0.0000 | 0.9726 | 0.0100 |
BT-20 | z-VAE(OMe)-fmk | 72 | inf | 0.9762 | 0.0198 | 0.0000 | 0.9890 | 0.0100 |
HCC1937 | z-VAE(OMe)-fmk | 72 | inf | 0.9933 | -0.0106 | 0.0000 | 1.0000 | 0.0100 |
HCC1419 | z-VAE(OMe)-fmk | 72 | inf | 0.9275 | 0.0463 | 0.0000 | 0.9622 | 0.0100 |
HCC1428 | z-VAE(OMe)-fmk | 72 | inf | 0.9944 | 0.0566 | 0.0000 | 0.9577 | 0.0100 |
MDA-MB-134-VI | z-VAE(OMe)-fmk | 72 | inf | 0.9937 | 0.1205 | 0.0000 | 0.8924 | 0.0100 |
HCC1428 | Vialinin A | 72 | 7.02266916467 | -0.5218 | 0.2922 | 19.4033 | -1.0000 | 1.0810 |
CAMA-1 | Vialinin A | 72 | 8.96202630369 | -0.5255 | 0.2577 | 13.2114 | -0.6248 | 2.0890 |
MCF7 | Vialinin A | 72 | 6.03216171414 | -0.2574 | 0.2814 | 7.1157 | -0.2692 | 2.6069 |
MCF 10A | Vialinin A | 72 | 12.7930209016 | -0.2051 | 0.1740 | 13.7221 | -0.2088 | 4.9768 |