Breast Cancer Deubiquitinating Enzyme (DUB) Inhibitor Profiling: Fixed-cell GR measures of 21 breast cell lines to 32 small molecule perturbagens. Dataset 2 of 2: Calculated dose response metrics. - Dataset (ID:20351)

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Cell Small Molecule Treatment Duration GR50 GRmax GR_AOC GEC50 GRinf hGR
HCC1428 5-(4-fluorophenyl)-3-hydroxy-4-(5-methyl-2-furoyl)-1-(3-pyridinylmethyl)-1,5-dihydro-2H-pyrrol-2-one 72
inf
0.9183 0.0941 0.0000 0.9165 0.0100
CAMA-1 z-VAE(OMe)-fmk 72
inf
0.9619 0.0262 0.0000 0.9726 0.0100
HCC1428 IU1 72
inf
0.7506 0.0316 0.0000 0.9483 0.0100
HCC1419 z-VAE(OMe)-fmk 72
inf
0.9275 0.0463 0.0000 0.9622 0.0100
HCC1428 USP7-IN-1 72
inf
0.6846 0.0667 0.0000 0.9252 0.0100
CAMA-1 STK547622 72
inf
0.8258 0.0467 0.0000 0.9496 0.0100
HCC1428 GW7647 72
inf
0.6988 -0.0012 0.0000 0.9685 0.0100
HCC1428 HY-17542 72
inf
0.7557 0.0179 0.0000 0.9697 0.0100
BT-549 z-VAE(OMe)-fmk 72
inf
0.9727 0.0182 0.0000 0.9828 0.0100
HCC1419 STK547622 72
inf
1.0781 0.0128 0.0000 1.0000 0.0100
HCC1419 5-(4-fluorophenyl)-3-hydroxy-4-(5-methyl-2-furoyl)-1-(3-pyridinylmethyl)-1,5-dihydro-2H-pyrrol-2-one 72
inf
0.9816 -0.0058 0.0000 1.0000 0.0100
BT-549 5-(4-fluorophenyl)-3-hydroxy-4-(5-methyl-2-furoyl)-1-(3-pyridinylmethyl)-1,5-dihydro-2H-pyrrol-2-one 72
inf
0.9516 0.0187 0.0000 0.9793 0.0100
BT-20 HY-17542 72
inf
1.0099 -0.0181 0.0000 1.0000 0.0100
CAMA-1 HY-17542 72
inf
0.8374 0.0179 0.0000 0.9681 0.0100
BT-20 5-(4-fluorophenyl)-3-hydroxy-4-(5-methyl-2-furoyl)-1-(3-pyridinylmethyl)-1,5-dihydro-2H-pyrrol-2-one 72
inf
1.0460 0.0369 0.0000 0.9732 0.0100
CAMA-1 5-(4-fluorophenyl)-3-hydroxy-4-(5-methyl-2-furoyl)-1-(3-pyridinylmethyl)-1,5-dihydro-2H-pyrrol-2-one 72
inf
0.9375 0.0403 0.0000 0.9497 0.0100
BT-20 SB1-F-22 72
inf
0.8486 -0.0325 0.0000 1.0000 0.0100
BT-20 Doxycycline 72
inf
0.5650 0.0355 0.0000 0.9177 0.0100
BT-20 IU1 72
inf
1.1490 -0.1850 0.0000 1.0000 0.0100
BT-20 STK547622 72
inf
1.1526 -0.0532 0.0000 1.0000 0.0100
BT-20 z-VAE(OMe)-fmk 72
inf
0.9762 0.0198 0.0000 0.9890 0.0100
BT-549 STK547622 72
inf
0.9826 0.0068 0.0000 0.9966 0.0100
BT-20 GW7647 72
inf
0.7093 -0.0625 0.0000 1.0000 0.0100
HCC1428 Doxycycline 72
inf
0.5312 0.1526 0.0000 0.8018 0.0100
HCC1428 STK547622 72
inf
0.8677 0.0634 0.0000 0.9587 0.0100
  • Page 1 of 27
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