Breast Cancer Deubiquitinating Enzyme (DUB) Inhibitor Profiling: Fixed-cell GR measures of 21 breast cell lines to 32 small molecule perturbagens. Dataset 2 of 2: Calculated dose response metrics. - Dataset (ID:20351)
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Cell | Small Molecule | Treatment Duration | GR50 | GRmax | GR_AOC | GEC50 | GRinf | hGR |
---|---|---|---|---|---|---|---|---|
PDX1328 | Pevonedistat | 72 | inf | -0.7089 | -0.4505 | 0.0000 | 1.0000 | 0.0100 |
PDX1328 | SB1-F-22 | 72 | inf | 1.0347 | -0.2404 | 0.0000 | 1.0000 | 0.0100 |
BT-20 | IU1 | 72 | inf | 1.1490 | -0.1850 | 0.0000 | 1.0000 | 0.0100 |
MDA-MB-361 | STK547622 | 72 | inf | 1.0471 | -0.1279 | 0.0000 | 1.0000 | 0.0100 |
MDA-MB-134-VI | GW7647 | 72 | inf | 1.0004 | -0.0983 | 0.0000 | 1.0000 | 0.0100 |
PDX1328 | GW7647 | 72 | inf | 0.8376 | -0.0784 | 0.0000 | 1.0000 | 0.0100 |
HCC202 | GW7647 | 72 | inf | 0.8031 | -0.0688 | 0.0000 | 1.0000 | 0.0100 |
PDX1258 | GW7647 | 72 | inf | 1.0702 | -0.0651 | 0.0000 | 1.0000 | 0.0100 |
BT-20 | GW7647 | 72 | inf | 0.7093 | -0.0625 | 0.0000 | 1.0000 | 0.0100 |
MDA-MB-361 | HY-17542 | 72 | inf | 0.8632 | -0.0548 | 0.0000 | 1.0000 | 0.0100 |
BT-20 | STK547622 | 72 | inf | 1.1526 | -0.0532 | 0.0000 | 1.0000 | 0.0100 |
HCC1937 | STK547622 | 72 | inf | 1.0316 | -0.0512 | 0.0000 | 1.0000 | 0.0100 |
MDA-MB-361 | IU1 | 72 | inf | 0.7838 | -0.0464 | 0.0000 | 1.0000 | 0.0100 |
HCC1937 | HY-17542 | 72 | inf | 0.9422 | -0.0439 | 0.0000 | 1.0000 | 0.0100 |
HCC1954 | GW7647 | 72 | 53.2192077737 | 0.5700 | -0.0367 | 66.2968 | -1.0000 | 5.0000 |
BT-20 | SB1-F-22 | 72 | inf | 0.8486 | -0.0325 | 0.0000 | 1.0000 | 0.0100 |
Hs 578T | GW7647 | 72 | inf | 0.8977 | -0.0280 | 0.0000 | 1.0000 | 0.0100 |
PDXHCI002 | GW7647 | 72 | inf | 0.7629 | -0.0251 | 0.0000 | 0.9997 | 0.0100 |
HCC202 | IU1 | 72 | inf | 0.7641 | -0.0242 | 0.0000 | 0.9954 | 0.0100 |
Hs 578T | Doxycycline | 72 | inf | 1.3436 | -0.0222 | 0.0000 | 1.0000 | 0.0100 |
HCC1500 | GW7647 | 72 | 42.1427904431 | 0.1820 | -0.0218 | 72.6766 | -0.9087 | 1.9008 |
Hs 578T | HY-17542 | 72 | inf | 0.9246 | -0.0205 | 0.0000 | 1.0000 | 0.0100 |
HCC202 | USP7-IN-1 | 72 | inf | 0.8501 | -0.0200 | 0.0000 | 1.0000 | 0.0100 |
MDA-MB-231 | GW7647 | 72 | inf | 0.9369 | -0.0195 | 0.0000 | 1.0000 | 0.0100 |
BT-20 | HY-17542 | 72 | inf | 1.0099 | -0.0181 | 0.0000 | 1.0000 | 0.0100 |