Breast Cancer Deubiquitinating Enzyme (DUB) Inhibitor Profiling: Fixed-cell GR measures of 21 breast cell lines to 32 small molecule perturbagens. Dataset 2 of 2: Calculated dose response metrics. - Dataset (ID:20351)
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Cell | Small Molecule | Treatment Duration | GR50 | GRmax | GR_AOC | GEC50 | GRinf | hGR |
---|---|---|---|---|---|---|---|---|
Hs 578T | ML-323 | 72 | 133.678939825 | 0.6153 | 0.1131 | 2077.0523 | -1.0000 | 0.4005 |
BT-20 | ML-323 | 72 | 211.396631725 | 0.7311 | 0.0653 | 1563.4058 | -1.0000 | 0.5491 |
HCC1954 | ML-323 | 72 | 85.295133896 | 0.5808 | 0.1325 | 985.9258 | -1.0000 | 0.4489 |
PDX1258 | SB1-F-22 | 72 | 141.822011334 | 0.6791 | 0.0519 | 862.0159 | -1.0000 | 0.6088 |
BT-549 | ML-323 | 72 | 74.3999913582 | 0.5763 | 0.0892 | 442.2433 | -1.0000 | 0.6164 |
HCC1806 | USP7-IN-1 | 72 | 154.815652356 | 0.8197 | 0.0286 | 421.1954 | -1.0000 | 1.0977 |
MCF 10A | USP7-IN-1 | 72 | 130.869645041 | 0.7420 | 0.0432 | 404.8308 | -0.8498 | 0.8794 |
HCC1937 | ML-323 | 72 | 86.9696327252 | 0.6194 | 0.0517 | 375.1322 | -0.9832 | 0.7439 |
MCF 10A | ML-323 | 72 | 66.3873318694 | 0.5514 | 0.0860 | 333.5126 | -1.0000 | 0.6806 |
PDX1328 | Spautin-1 | 72 | 43.5833222905 | 0.4636 | 0.1399 | 310.0635 | -1.0000 | 0.5599 |
T47D | USP7-IN-1 | 72 | 35.2358506575 | 0.3921 | 0.1491 | 300.7608 | -1.0000 | 0.5124 |
MDA-MB-231 | ML-323 | 72 | 60.8635339383 | 0.5091 | 0.0928 | 299.6220 | -1.0000 | 0.6893 |
T47D | SB1-F-22 | 72 | 156.804339896 | 0.7134 | 0.0621 | 286.2396 | -0.2481 | 0.6696 |
MCF 10A | 5-(4-fluorophenyl)-3-hydroxy-4-(5-methyl-2-furoyl)-1-(3-pyridinylmethyl)-1,5-dihydro-2H-pyrrol-2-one | 72 | 738.9217363 | 0.8943 | 0.0150 | 255.4365 | 0.3311 | 1.0216 |
SK-BR-3 | ML-323 | 72 | 71.5457262907 | 0.6083 | 0.0659 | 250.9976 | -1.0000 | 0.8753 |
CAMA-1 | USP7-IN-1 | 72 | 90.407874652 | 0.7005 | 0.0265 | 239.6012 | -1.0000 | 1.1272 |
MCF 10A | HY-17542 | 72 | 122.726417103 | 0.9130 | 0.0108 | 200.5533 | -1.0000 | 2.2369 |
HCC1806 | IU1 | 72 | 116.251943958 | 0.8831 | 0.0051 | 197.1530 | -0.9493 | 2.0147 |
BT-549 | USP7-IN-1 | 72 | 94.531181628 | 0.8209 | 0.0177 | 166.1357 | -1.0000 | 1.9483 |
CAMA-1 | SB1-F-22 | 72 | 43.6088606735 | 0.4408 | 0.0565 | 156.5267 | -1.0000 | 0.8597 |
MCF7 | ML-323 | 72 | 34.9041902184 | 0.3934 | 0.1213 | 138.0045 | -1.0000 | 0.7992 |
SK-BR-3 | USP7-IN-1 | 72 | 62.2210904101 | 0.5764 | 0.0588 | 133.0943 | -1.0000 | 1.4449 |
HCC1500 | USP7-IN-1 | 72 | 51.9923039456 | 0.4861 | 0.0630 | 130.5080 | -1.0000 | 1.1937 |
T47D | HY-17542 | 72 | 60.7583842474 | 0.5918 | 0.0384 | 120.2191 | -1.0000 | 1.6099 |
SK-BR-3 | GW7647 | 72 | 63.3177975853 | 0.6434 | 0.0223 | 112.2791 | -1.0000 | 1.9179 |