Evaluation of the sensitivity of two triple-negative breast cancer cell lines (HCC1806, HCC70) to a collection of dual mTOR and PI3K-like kinase (PIKK) inhibitors. Dataset 2 of 2: GR metrics. - Dataset (ID:20367)
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Cell line | Drug name | Experimental replicate | Curve type (GR values) | Curve type (relative cell counts) | Experiment name | Number of concentrations | Cell doublings (DMSO control) | GR50 | GRmax | GR_AOC | GEC50 | GRinf | Hill slope (GR values) | R-squared curve fit (GR values) | P-value curve fit (GR values) | IC50 | Emax | AUC | EC50 | Einf | Hill slope (relative cell counts) | R-squared curve fit (relative cell counts) | P-value curve fit (relative cell counts) |
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HCC70 | QL-X-138 | 2 | sigmoid | sigmoid | HCC70 QL-X-138 0 2 | 9 | 1.573 | 1.62 | -0.286 | 0.211 | 3.74 | -0.725 | 1.07 | 0.966 | 1.18e-25 | 2.65 | 0.198 | 0.859 | 2.44 | 0.045 | 1.14 | 0.953 | 3.05e-23 |
HCC70 | QL-VI-86 | 2 | sigmoid | sigmoid | HCC70 QL-VI-86 0 2 | 9 | 1.573 | 0.266 | -0.695 | 0.519 | 0.899 | -0.926 | 0.861 | 0.989 | 1.06e-33 | 0.467 | 0.052 | 0.672 | 0.467 | 0.0 | 0.934 | 0.983 | 9.31e-31 |
HCC70 | Torin1 | 2 | sigmoid | sigmoid | HCC70 Torin1 0 2 | 9 | 1.573 | 0.0399 | -0.322 | 0.653 | 0.107 | -0.343 | 0.53 | 0.962 | 7.04e-25 | 0.123 | 0.183 | 0.557 | 0.0522 | 0.201 | 0.6 | 0.964 | 3.46e-25 |
HCC70 | QL-IV-100 | 2 | sigmoid | sigmoid | HCC70 QL-IV-100 0 2 | 9 | 1.573 | 0.0891 | -0.75 | 0.716 | 0.451 | -1.0 | 0.678 | 0.986 | 2.16e-32 | 0.18 | 0.0381 | 0.549 | 0.18 | 0.0 | 0.729 | 0.977 | 1.02e-28 |
HCC70 | QL-VIII-58 | 2 | sigmoid | sigmoid | HCC70 QL-VIII-58 0 2 | 9 | 1.573 | 0.0674 | -0.973 | 0.806 | 0.287 | -1.0 | 0.759 | 0.972 | 3.07e-27 | 0.12 | 0.00122 | 0.517 | 0.12 | 0.0 | 0.752 | 0.975 | 6.9e-28 |
HCC70 | QL-V-107 | 2 | sigmoid | sigmoid | HCC70 QL-V-107 0 2 | 9 | 1.573 | 0.0752 | -0.655 | 0.721 | 0.361 | -0.895 | 0.653 | 0.99 | 7.55e-35 | 0.163 | 0.0632 | 0.541 | 0.163 | 0.0 | 0.682 | 0.987 | 1.08e-32 |
HCC70 | QL-XII-47 | 2 | sigmoid | sigmoid | HCC70 QL-XII-47 0 2 | 9 | 1.573 | 0.728 | -0.818 | 0.401 | 1.07 | -0.805 | 2.49 | 0.991 | 6.84e-36 | 0.901 | 0.0231 | 0.771 | 0.883 | 0.029 | 2.89 | 0.985 | 1.44e-31 |
HCC70 | Torin2 | 2 | sigmoid | sigmoid | HCC70 Torin2 0 2 | 9 | 1.573 | 0.0124 | -0.955 | 1.11 | 0.0639 | -1.0 | 0.669 | 0.99 | 1.92e-34 | 0.0242 | 0.00262 | 0.351 | 0.0242 | 0.0 | 0.695 | 0.987 | 7.52e-33 |
HCC70 | QL-XII-108 | 2 | sigmoid | sigmoid | HCC70 QL-XII-108 0 2 | 9 | 1.573 | 1.64 | 0.0651 | 0.189 | 1.78 | -0.0491 | 1.11 | 0.948 | 1.42e-22 | 3.36 | 0.371 | 0.867 | 1.34 | 0.336 | 1.2 | 0.936 | 4.76e-21 |
HCC70 | QL-V-73 | 2 | sigmoid | sigmoid | HCC70 QL-V-73 0 2 | 9 | 1.573 | 0.397 | -0.619 | 0.474 | 1.71 | -1.0 | 0.751 | 0.983 | 7.11e-31 | 0.749 | 0.0739 | 0.686 | 0.749 | 0.0 | 0.776 | 0.972 | 4.32e-27 |
HCC70 | QL-XII-61 | 2 | sigmoid | sigmoid | HCC70 QL-XII-61 0 2 | 9 | 1.573 | 4.5 | 0.179 | 0.0498 | 4.14 | 0.169 | 5.0 | 0.928 | 3.35e-20 | 5.98 | 0.436 | 0.967 | 4.03 | 0.43 | 5.0 | 0.913 | 1.01e-18 |
HCC70 | AZD8055 | 2 | sigmoid | sigmoid | HCC70 AZD8055 0 2 | 9 | 1.573 | 0.029 | -0.0375 | 0.612 | 0.0272 | 0.0241 | 0.792 | 0.972 | 3.37e-27 | 0.0959 | 0.317 | 0.576 | 0.0216 | 0.35 | 0.808 | 0.974 | 9.92e-28 |
HCC70 | QL-V-107 | 1 | sigmoid | sigmoid | HCC70 QL-V-107 0 1 | 9 | 1.598 | 0.0994 | -0.612 | 0.672 | 0.409 | -0.834 | 0.694 | 0.988 | 3.47e-33 | 0.206 | 0.0727 | 0.566 | 0.206 | 0.0 | 0.712 | 0.984 | 4.79e-31 |
HCC70 | Torin2 | 1 | sigmoid | sigmoid | HCC70 Torin2 0 1 | 9 | 1.598 | 0.014 | -0.946 | 1.07 | 0.0747 | -1.0 | 0.657 | 0.991 | 3.28e-35 | 0.0269 | 0.00323 | 0.362 | 0.0269 | 0.0 | 0.682 | 0.988 | 1.64e-33 |
HCC70 | QL-VI-86 | 1 | sigmoid | sigmoid | HCC70 QL-VI-86 0 1 | 9 | 1.598 | 0.299 | -0.674 | 0.511 | 1.21 | -1.0 | 0.786 | 0.987 | 7.69e-33 | 0.529 | 0.0552 | 0.668 | 0.529 | 0.0 | 0.854 | 0.981 | 5.86e-30 |
HCC70 | QL-XII-47 | 1 | sigmoid | sigmoid | HCC70 QL-XII-47 0 1 | 9 | 1.598 | 0.767 | -0.806 | 0.406 | 1.22 | -0.822 | 2.11 | 0.994 | 3.85e-38 | 0.971 | 0.0243 | 0.758 | 0.954 | 0.0199 | 2.33 | 0.989 | 7.52e-34 |
HCC70 | AZD8055 | 1 | sigmoid | sigmoid | HCC70 AZD8055 0 1 | 9 | 1.598 | 0.0382 | 0.0624 | 0.564 | 0.0292 | 0.0882 | 0.722 | 0.969 | 1.75e-26 | 0.158 | 0.364 | 0.601 | 0.0229 | 0.379 | 0.734 | 0.965 | 1.44e-25 |
HCC70 | Torin1 | 1 | sigmoid | sigmoid | HCC70 Torin1 0 1 | 9 | 1.598 | 0.061 | -0.147 | 0.573 | 0.0884 | -0.134 | 0.64 | 0.954 | 1.68e-23 | 0.182 | 0.256 | 0.601 | 0.057 | 0.275 | 0.684 | 0.957 | 6.27e-24 |
HCC70 | QL-XII-108 | 1 | sigmoid | sigmoid | HCC70 QL-XII-108 0 1 | 9 | 1.598 | 1.64 | 0.0903 | 0.226 | 2.06 | -0.115 | 0.914 | 0.963 | 5.57e-25 | 3.65 | 0.379 | 0.836 | 1.5 | 0.287 | 0.962 | 0.954 | 1.98e-23 |
HCC70 | QL-V-73 | 1 | sigmoid | sigmoid | HCC70 QL-V-73 0 1 | 9 | 1.598 | 0.538 | -0.558 | 0.42 | 2.22 | -1.0 | 0.774 | 0.987 | 5.03e-33 | 0.973 | 0.0898 | 0.716 | 0.973 | 0.0 | 0.812 | 0.98 | 1.98e-29 |
HCC70 | QL-XII-61 | 1 | sigmoid | sigmoid | HCC70 QL-XII-61 0 1 | 9 | 1.598 | 6.18 | 0.125 | 0.0875 | 11.5 | -1.0 | 1.76 | 0.946 | 2.8e-22 | 8.07 | 0.399 | 0.937 | 8.07 | 0.0 | 1.9 | 0.932 | 1.35e-20 |
HCC70 | QL-X-138 | 1 | sigmoid | sigmoid | HCC70 QL-X-138 0 1 | 9 | 1.598 | 1.41 | -0.213 | 0.248 | 3.83 | -0.724 | 0.893 | 0.983 | 5.84e-31 | 2.51 | 0.225 | 0.827 | 2.38 | 0.025 | 0.931 | 0.978 | 8.59e-29 |
HCC70 | QL-IV-100 | 1 | sigmoid | sigmoid | HCC70 QL-IV-100 0 1 | 9 | 1.598 | 0.115 | -0.713 | 0.67 | 0.502 | -0.951 | 0.723 | 0.992 | 2.58e-36 | 0.219 | 0.045 | 0.574 | 0.219 | 0.0 | 0.776 | 0.989 | 2.4e-34 |
HCC70 | QL-VIII-58 | 1 | sigmoid | sigmoid | HCC70 QL-VIII-58 0 1 | 9 | 1.598 | 0.0739 | -0.976 | 0.791 | 0.319 | -1.0 | 0.752 | 0.972 | 4.08e-27 | 0.127 | 0.000989 | 0.519 | 0.127 | 0.0 | 0.723 | 0.981 | 6.68e-30 |
HCC70 | QL-VI-86 | 3 | sigmoid | sigmoid | HCC70 QL-VI-86 0 3 | 9 | 1.750 | 0.305 | -0.639 | 0.508 | 1.34 | -1.0 | 0.742 | 0.989 | 4.41e-34 | 0.478 | 0.0501 | 0.649 | 0.478 | 0.0 | 0.81 | 0.981 | 5.26e-30 |