GRK1 - Protein (ID:)
| Name: | GRK1 |
| HMS LINCS ID: | 200180 |
| UniProt ID: | Q15835 |
| Alternative Names: | G protein-coupled receptor kinase 1; GPRK1; GRK1; RHODK; RHODK/GRK1; RHOK; RK |
| Provider: | KINOMEscan |
| Provider Catalog ID: | |
| Amino Acid Sequence: | |
| Gene Symbol: | GRK1 |
| Gene ID: | 6011 |
| Protein Source: | Mammalian expression system |
| Mutation: | |
| Phosphlorylation State: | |
| Domain: | |
| Protein Description: | Wild Type; Full length |
| Protein Purity: | |
| Protein Complex: | |
| Isoform: | |
| Protein Type: | |
| Source Organism: | Homo sapiens |
| Reference: | |
| Comments: | |
| Date Publicly Available: | 2012-11-15 |
| Most Recent Update: | 2016-09-14 |
Datasets:
| HMS Dataset ID | Dataset Title | HMS Dataset Type |
|---|---|---|
| 20020 | Sorafenib KINOMEscan | KINOMEscan |
| 20021 | HG-6-64-1 KINOMEscan | KINOMEscan |
| 20022 | GW-5074 KINOMEscan | KINOMEscan |
| 20023 | SB590885 KINOMEscan | KINOMEscan |
| 20024 | PLX-4720 KINOMEscan | KINOMEscan |
| 20025 | AZ-628 KINOMEscan | KINOMEscan |
| 20026 | PLX4032 KINOMEscan | KINOMEscan |
| 20027 | AZD7762 KINOMEscan | KINOMEscan |
| 20028 | CP466722 KINOMEscan | KINOMEscan |
| 20029 | CP724714 KINOMEscan | KINOMEscan |
| 20030 | GSK429286A KINOMEscan | KINOMEscan |
| 20031 | GSK461364 KINOMEscan | KINOMEscan |
| 20032 | GW843682 KINOMEscan | KINOMEscan |
| 20033 | PF02341066 KINOMEscan | KINOMEscan |
| 20034 | BMS345541 KINOMEscan | KINOMEscan |
| 20035 | AS601245 KINOMEscan | KINOMEscan |
| 20036 | WH-4-023 KINOMEscan | KINOMEscan |
| 20037 | BX-912 KINOMEscan | KINOMEscan |
| 20038 | AZD-6482 KINOMEscan | KINOMEscan |
| 20039 | TAK-715 KINOMEscan | KINOMEscan |
| 20040 | NU7441 KINOMEscan | KINOMEscan |
| 20041 | KIN001-220 KINOMEscan | KINOMEscan |
| 20042 | MLN8054 KINOMEscan | KINOMEscan |
| 20043 | AZD1152-HQPA KINOMEscan | KINOMEscan |
| 20044 | PD0332991 KINOMEscan | KINOMEscan |
| 20045 | THZ-2-98-01 KINOMEscan | KINOMEscan |
| 20046 | JWE-035 KINOMEscan | KINOMEscan |
| 20047 | ZM-447439 KINOMEscan | KINOMEscan |
| 20048 | JNK-9L KINOMEscan | KINOMEscan |
| 20049 | ALW-II-38-3 KINOMEscan | KINOMEscan |
| 20053 | HKI-272 KINOMEscan | KINOMEscan |
| 20054 | CGP60474 KINOMEscan | KINOMEscan |
| 20060 | GDC-0941 KINOMEscan | KINOMEscan |
| 20062 | QL-X-138 KINOMEscan | KINOMEscan |
| 20063 | QL-XI-92 KINOMEscan | KINOMEscan |
| 20064 | Torin1 KINOMEscan | KINOMEscan |
| 20065 | Torin2 KINOMEscan | KINOMEscan |
| 20067 | WZ-7043 KINOMEscan | KINOMEscan |
| 20068 | WZ3105 KINOMEscan | KINOMEscan |
| 20070 | XMD11-50 KINOMEscan | KINOMEscan |
| 20071 | XMD11-85h KINOMEscan | KINOMEscan |
| 20072 | XMD13-2 KINOMEscan | KINOMEscan |
| 20073 | XMD14-99 KINOMEscan | KINOMEscan |
| 20074 | XMD15-27 KINOMEscan | KINOMEscan |
| 20075 | XMD16-144 KINOMEscan | KINOMEscan |
| 20076 | XMD8-85 KINOMEscan | KINOMEscan |
| 20077 | XMD8-92 KINOMEscan | KINOMEscan |
| 20078 | ZG-10 KINOMEscan | KINOMEscan |
| 20079 | WYE-125132 KINOMEscan | KINOMEscan |
| 20080 | PD0325901 KINOMEscan | KINOMEscan |
| 20081 | JNK-IN-5A KINOMEscan | KINOMEscan |
| 20082 | CYT387 KINOMEscan | KINOMEscan |
| 20083 | Sigma A6730 KINOMEscan | KINOMEscan |
| 20084 | GSK2126458 KINOMEscan | KINOMEscan |
| 20085 | GSK1059615 KINOMEscan | KINOMEscan |
| 20086 | AG1478 KINOMEscan | KINOMEscan |
| 20096 | BEZ235 KINOMEscan | KINOMEscan |
| 20107 | Lapatinib KINOMEscan | KINOMEscan |
| 20114 | CG-930 KINOMEscan | KINOMEscan |
| 20115 | XMD-12 KINOMEscan | KINOMEscan |
| 20116 | Bosutinib KINOMEscan | KINOMEscan |
| 20117 | KU63794 KINOMEscan | KINOMEscan |
| 20124 | (R)-Roscovitine KINOMEscan | KINOMEscan |
| 20125 | PHA-793887 KINOMEscan | KINOMEscan |
| 20126 | PHA-767491 KINOMEscan | KINOMEscan |
| 20127 | BS-181 KINOMEscan | KINOMEscan |
| 20128 | Dinaciclib KINOMEscan | KINOMEscan |
| 20129 | AZD4547 KINOMEscan | KINOMEscan |
| 20130 | OTSSP167 KINOMEscan | KINOMEscan |
| 20131 | Dabrafenib KINOMEscan | KINOMEscan |
| 20132 | HG-9-91-01 KINOMEscan | KINOMEscan |
| 20133 | HG-14-8-02 KINOMEscan | KINOMEscan |
| 20134 | HG-14-10-04 KINOMEscan | KINOMEscan |
| 20135 | AZD 5438 KINOMEscan | KINOMEscan |
| 20146 | BMS-345541 KINOMEscan | KINOMEscan |
| 20147 | AC220 KINOMEscan | KINOMEscan |
| 20148 | R406 KINOMEscan-2 | KINOMEscan |
| 20149 | BI-2536 KINOMEscan-2 | KINOMEscan |
| 20150 | AMG-706 KINOMEscan | KINOMEscan |
| 20151 | BIRB-796 KINOMEscan | KINOMEscan |
| 20152 | GDC-0941 KINOMEscan-2 | KINOMEscan |
| 20153 | CI-1040 KINOMEscan | KINOMEscan |
| 20154 | PLX-4720 KINOMEscan-2 | KINOMEscan |
| 20155 | Lapatinib KINOMEscan-2 | KINOMEscan |
| 20156 | AZD-6244 KINOMEscan | KINOMEscan |
| 20157 | MLN-8054 KINOMEscan | KINOMEscan |
| 20158 | AZD-1152HQPA KINOMEscan-2 | KINOMEscan |
| 20159 | LY-317615 KINOMEscan | KINOMEscan |
| 20160 | Erlotinib KINOMEscan | KINOMEscan |
| 20161 | Gefitinib KINOMEscan | KINOMEscan |
| 20162 | Nilotinib KINOMEscan | KINOMEscan |
| 20163 | Pazopanib KINOMEscan | KINOMEscan |
| 20164 | CI-1033 KINOMEscan-2 | KINOMEscan |
| 20165 | SGX-523 KINOMEscan | KINOMEscan |
| 20166 | PHA-665752 KINOMEscan | KINOMEscan |
| 20167 | PI-103 KINOMEscan | KINOMEscan |
| 20168 | TKI-258 KINOMEscan | KINOMEscan |
| 20169 | GSK-690693 KINOMEscan | KINOMEscan |
| 20170 | AB-1010 KINOMEscan | KINOMEscan |
| 20171 | BMS-387032 KINOMEscan | KINOMEscan |
| 20172 | BIBW-2992 KINOMEscan | KINOMEscan |
| 20173 | INCB018424 KINOMEscan | KINOMEscan |
| 20174 | TG-101348 KINOMEscan | KINOMEscan |
| 20175 | BIBF-1120 KINOMEscan | KINOMEscan |
| 20176 | GSK-1363089 KINOMEscan | KINOMEscan |
| 20177 | SB-203580 KINOMEscan | KINOMEscan |
| 20178 | VX-745 KINOMEscan | KINOMEscan |
| 20179 | Sunitinib KINOMEscan | KINOMEscan |
| 20180 | BMS-540215 KINOMEscan | KINOMEscan |
| 20181 | GDC-0879 KINOMEscan | KINOMEscan |
| 20182 | ABT-869 KINOMEscan | KINOMEscan |
| 20183 | Ki-20227 KINOMEscan | KINOMEscan |
| 20184 | SKI-606 KINOMEscan | KINOMEscan |
| 20185 | KW-2449 KINOMEscan | KINOMEscan |
| 20186 | Vandetanib KINOMEscan | KINOMEscan |
| 20187 | PKC-412 KINOMEscan | KINOMEscan |
| 20188 | CP-690550 KINOMEscan | KINOMEscan |
| 20189 | CEP-701 KINOMEscan | KINOMEscan |
| 20190 | GSK-1838705A KINOMEscan | KINOMEscan |
| 20191 | AT-7519 KINOMEscan | KINOMEscan |
| 20192 | Sorafenib KINOMEscan-2 | KINOMEscan |
| 20193 | Flavopiridol KINOMEscan | KINOMEscan |
| 20194 | GSK-461364A KINOMEscan | KINOMEscan |
| 20195 | HKI-272 KINOMEscan-2 | KINOMEscan |
| 20196 | Dasatinib KINOMEscan | KINOMEscan |
| 20197 | VX-680 KINOMEscan | KINOMEscan |
| 20198 | Imatinib KINOMEscan | KINOMEscan |
| 20199 | TAE-684 KINOMEscan | KINOMEscan |
| 20200 | Crizotinib KINOMEscan-2 | KINOMEscan |
| 20201 | RAF-265 KINOMEscan | KINOMEscan |
| 20202 | RO-3306 KINOMEscan | KINOMEscan |
| 20203 | CGP74514A KINOMEscan | KINOMEscan |
| 20211 | 5z-7-oxozeaenol KINOMEscan | KINOMEscan |
| 20212 | JNK-IN-8 KINOMEscan | KINOMEscan |
| 20222 | Ibrutinib KINOMEscan | KINOMEscan |
| 20224 | BGJ398 KINOMEscan | KINOMEscan |
| 20227 | Baricitinib KINOMEscan | KINOMEscan |
| 20228 | MRT67307 KINOMEscan | KINOMEscan |
| 20261 | GDC-0941 KINOMEscan-3 | KINOMEscan |
| 20262 | Buparlisib KINOMEscan | KINOMEscan |
| 20263 | BYL719 KINOMEscan | KINOMEscan |
| 20264 | Taselisib KINOMEscan | KINOMEscan |
| 20326 | CH5424802 KINOMEscan | KINOMEscan |
| 20327 | BI-D1870 KINOMEscan | KINOMEscan |
| 20328 | Torkinib KINOMEscan | KINOMEscan |
| 20329 | Ceritinib KINOMEscan | KINOMEscan |
| 20330 | Ribociclib KINOMEscan | KINOMEscan |
| 20332 | BMX-IN-1 KINOMEscan | KINOMEscan |
| 20333 | SCH772984 KINOMEscan | KINOMEscan |
| 20334 | THZ1 KINOMEscan | KINOMEscan |
| 20335 | JNK-IN-11 KINOMEscan | KINOMEscan |
| 20337 | ERK5-IN-1 KINOMEscan | KINOMEscan |
| 20338 | Abemaciclib KINOMEscan | KINOMEscan |
| 20339 | Palbociclib KINOMEscan | KINOMEscan |
| 20340 | QL-XII-47 KINOMEscan | KINOMEscan |
| 20342 | (s)-CR8 KINOMEscan | KINOMEscan |