Breast Cancer Profiling Project, Drug Sensitivity phase II: Fixed-cell GR measures of 33 breast cell lines and PDX lines to 16 small molecule perturbagens from library plate II. Dataset 2 of 2: Calculated dose response metrics - Dataset (ID:20355)
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Cell | Small Molecule | GR50 | GRmax | GR_AOC | GEC50 | GRinf | GR Hill Coefficient | GR r2 | pval_GR |
---|---|---|---|---|---|---|---|---|---|
MCF7 | AZD5363 | 12.4103884 | 0.4782 | 0.2060 | 1.1629 | 0.3135 | 0.4165 | 0.8201 | 4.86e-10 |
HCC1395 | RO-3306 | 0.479643325 | -0.1494 | 0.4249 | 6.7176 | -1.0000 | 0.4162 | 0.8546 | 3.39e-11 |
HCC1395 | BMS-265246 | 0.005815242 | -0.2349 | 0.7953 | 0.0151 | -0.2416 | 0.4121 | 0.9312 | 3e-15 |
HCC1937 | BMS-265246 | 0.000340758 | -0.0634 | 0.9143 | 0.0005 | -0.0734 | 0.4108 | 0.8462 | 6.89e-11 |
HCC1419 | AZD2014 | 0.000451019 | -0.1328 | 0.9581 | 0.0009 | -0.1553 | 0.4080 | 0.8343 | 1.75e-10 |
HCC38 | BMS-265246 | 0.00394749 | -0.0214 | 0.7767 | 0.0054 | -0.0686 | 0.4043 | 0.9575 | 1.11e-16 |
MDA-MB-436 | Ulixertinib | 34.76507133 | 0.5719 | 0.1213 | 534.6670 | -1.0000 | 0.4020 | 0.5984 | 1.11e-05 |
HCC1806 | Senexin B | inf | 0.8083 | 0.1042 | 0.1453 | 0.7979 | 0.4002 | 0.4857 | 0.000245355132328 |
CAL-51 | MK 1775 | 0.310910353 | -0.1886 | 0.4395 | 4.9452 | -1.0000 | 0.3971 | 0.9792 | 1.11e-16 |
MCF7 | Ribociclib | 0.189284804 | 0.2285 | 0.4067 | 0.0345 | 0.2453 | 0.3959 | 0.8429 | 8.95e-11 |
AU565 | MK 1775 | 0.223405816 | -0.4543 | 0.4894 | 3.6482 | -1.0000 | 0.3933 | 0.8692 | 9.09e-12 |
CAMA-1 | Ulixertinib | 2.566161953 | 0.1288 | 0.2586 | 42.4009 | -1.0000 | 0.3917 | 0.5616 | 3.34e-05 |
HCC1143 | BMS-265246 | 0.001767259 | -0.0571 | 0.8227 | 0.0030 | -0.1138 | 0.3912 | 0.9074 | 1.21e-13 |
Hs 578T | MK 1775 | 0.014507078 | -0.3462 | 0.7648 | 0.0762 | -0.4564 | 0.3909 | 0.9740 | 1.11e-16 |
CAL-85-1 | MK 1775 | 0.182874423 | -0.5298 | 0.5409 | 3.0854 | -1.0000 | 0.3888 | 0.7205 | 1.2e-07 |
HCC1937 | AZD5363 | 12.85319785 | 0.4773 | 0.3596 | 0.0112 | 0.4671 | 0.3863 | 0.5345 | 7.07e-05 |
HCC38 | Senexin B | 15.63810324 | 0.5236 | 0.1411 | 269.9088 | -0.9985 | 0.3853 | 0.5885 | 1.51e-05 |
HCC1954 | AZD5363 | 2.96992805185 | 0.2599 | 0.2385 | 51.5317 | -1.0000 | 0.3850 | 0.8789 | 3.45068418284e-12 |
HCC1419 | GSK2334470 | 7.272032069 | 0.4604 | 0.2878 | 0.7439 | 0.2916 | 0.3838 | 0.5825 | 1.81e-05 |
Hs 578T | Ulixertinib | 1.12758771 | 0.2421 | 0.3284 | 1.7251 | -0.0883 | 0.3825 | 0.9567 | 1.11e-16 |
MDA-MB-453 | GSK2334470 | 2.045052119 | 0.1203 | 0.2628 | 36.8285 | -1.0000 | 0.3800 | 0.7865 | 4.15e-09 |
SUM149PT | BMS-265246 | 0.016950371 | 0.0738 | 0.6317 | 0.0171 | -0.0015 | 0.3767 | 0.9526 | 1.11e-16 |
SUM1315MO2 | SHP099 | 22.32790504 | 0.4783 | 0.1197 | 419.3194 | -1.0000 | 0.3746 | 0.3197 | 0.008107411 |
Hs 578T | AZD2014 | 0.068067431 | 0.2555 | 0.5090 | 0.0201 | 0.1834 | 0.3744 | 0.9704 | 1.11e-16 |
CAL-85-1 | Ulixertinib | 3.83746694 | 0.2311 | 0.2960 | 72.1557 | -1.0000 | 0.3744 | 0.3008 | 0.011412092 |