Evaluation of the sensitivities of six triple-negative breast cancer (TNBC) cell lines to 23 different PI3K/AKT/mTOR inhibitors or to a MEK inhibitor (trametinib). Dataset 1 of 2: GR values. - Dataset (ID:20364)
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Cell line | Drug name | Experimental replicate | Timepoint | Drug concentration | Live cell count | Average live cell count, DMSO control | Average live cell count (time = 0) | Log10(drug concentration) | GR value | Relative cell count (treatment versus DMSO) | Cell doublings (DMSO control) | Experiment name |
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Hs 578T | Dactolisib | 2 | 72 | 0.1 | 1055.0 | 3555.0 | 624.7 | -1.0 | 0.232 | 0.297 | 2.509 | Hs578T BEZ235 2 |
Hs 578T | Dactolisib | 2 | 72 | 0.32 | 829.8 | 3555.0 | 624.7 | -0.495 | 0.120 | 0.233 | 2.509 | Hs578T BEZ235 2 |
Hs 578T | Dactolisib | 2 | 72 | 1.0 | 728.5 | 3555.0 | 624.7 | 0.0 | 0.063 | 0.205 | 2.509 | Hs578T BEZ235 2 |
Hs 578T | Dactolisib | 2 | 72 | 3.2 | 532.5 | 3555.0 | 624.7 | 0.505 | -0.062 | 0.150 | 2.509 | Hs578T BEZ235 2 |
Hs 578T | Buparlisib | 2 | 72 | 0.001 | 3710.0 | 3566.8 | 624.7 | -3.0 | 1.030 | 1.040 | 2.513 | Hs578T BKM120 2 |
Hs 578T | Buparlisib | 2 | 72 | 0.0032 | 3593.8 | 3566.8 | 624.7 | -2.49 | 1.010 | 1.010 | 2.513 | Hs578T BKM120 2 |
Hs 578T | Buparlisib | 2 | 72 | 0.01 | 3527.8 | 3566.8 | 624.7 | -2.0 | 0.991 | 0.989 | 2.513 | Hs578T BKM120 2 |
Hs 578T | Buparlisib | 2 | 72 | 0.032 | 3475.3 | 3566.8 | 624.7 | -1.49 | 0.979 | 0.974 | 2.513 | Hs578T BKM120 2 |
Hs 578T | Buparlisib | 2 | 72 | 0.1 | 3150.3 | 3566.8 | 624.7 | -1.0 | 0.904 | 0.883 | 2.513 | Hs578T BKM120 2 |
Hs 578T | Buparlisib | 2 | 72 | 0.32 | 2526.5 | 3566.8 | 624.7 | -0.495 | 0.744 | 0.708 | 2.513 | Hs578T BKM120 2 |
Hs 578T | Buparlisib | 2 | 72 | 1.0 | 1255.0 | 3566.8 | 624.7 | 0.0 | 0.320 | 0.352 | 2.513 | Hs578T BKM120 2 |
Hs 578T | Buparlisib | 2 | 72 | 3.2 | 158.8 | 3566.8 | 624.7 | 0.505 | -0.420 | 0.045 | 2.513 | Hs578T BKM120 2 |
Hs 578T | BX-912 | 2 | 72 | 0.001 | 3521.3 | 3632.8 | 624.7 | -3.0 | 0.976 | 0.969 | 2.540 | Hs578T BX912 2 |
Hs 578T | BX-912 | 2 | 72 | 0.0032 | 3582.0 | 3632.8 | 624.7 | -2.49 | 0.989 | 0.986 | 2.540 | Hs578T BX912 2 |
Hs 578T | BX-912 | 2 | 72 | 0.01 | 3561.8 | 3632.8 | 624.7 | -2.0 | 0.985 | 0.980 | 2.540 | Hs578T BX912 2 |
Hs 578T | BX-912 | 2 | 72 | 0.032 | 3564.0 | 3632.8 | 624.7 | -1.49 | 0.985 | 0.981 | 2.540 | Hs578T BX912 2 |
Hs 578T | BX-912 | 2 | 72 | 0.1 | 3390.3 | 3632.8 | 624.7 | -1.0 | 0.946 | 0.933 | 2.540 | Hs578T BX912 2 |
Hs 578T | BX-912 | 2 | 72 | 0.32 | 3091.5 | 3632.8 | 624.7 | -0.495 | 0.877 | 0.851 | 2.540 | Hs578T BX912 2 |
Hs 578T | BX-912 | 2 | 72 | 1.0 | 1822.8 | 3632.8 | 624.7 | 0.0 | 0.524 | 0.502 | 2.540 | Hs578T BX912 2 |
Hs 578T | BX-912 | 2 | 72 | 3.2 | 595.0 | 3632.8 | 624.7 | 0.505 | -0.019 | 0.164 | 2.540 | Hs578T BX912 2 |
Hs 578T | Alpelisib | 2 | 72 | 0.001 | 2972.3 | 3566.3 | 624.7 | -3.0 | 0.860 | 0.833 | 2.513 | Hs578T BYL719 2 |
Hs 578T | Alpelisib | 2 | 72 | 0.0032 | 2946.5 | 3566.3 | 624.7 | -2.49 | 0.854 | 0.826 | 2.513 | Hs578T BYL719 2 |
Hs 578T | Alpelisib | 2 | 72 | 0.01 | 3462.0 | 3566.3 | 624.7 | -2.0 | 0.977 | 0.971 | 2.513 | Hs578T BYL719 2 |
Hs 578T | Alpelisib | 2 | 72 | 0.032 | 3302.8 | 3566.3 | 624.7 | -1.49 | 0.940 | 0.926 | 2.513 | Hs578T BYL719 2 |
Hs 578T | Alpelisib | 2 | 72 | 0.1 | 3269.8 | 3566.3 | 624.7 | -1.0 | 0.932 | 0.917 | 2.513 | Hs578T BYL719 2 |