Evaluation of the sensitivities of six triple-negative breast cancer (TNBC) cell lines to 23 different PI3K/AKT/mTOR inhibitors or to a MEK inhibitor (trametinib). Dataset 1 of 2: GR values. - Dataset (ID:20364)

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Cell line Drug name Experimental replicate Timepoint Drug concentration Live cell count Average live cell count, DMSO control Average live cell count (time = 0) Log10(drug concentration) GR value Relative cell count (treatment versus DMSO) Cell doublings (DMSO control) Experiment name
Hs 578T Dactolisib 2 72
0.1
1055.0 3555.0 624.7
-1.0
0.232 0.297 2.509
Hs578T BEZ235 2
Hs 578T Dactolisib 2 72
0.32
829.8 3555.0 624.7
-0.495
0.120 0.233 2.509
Hs578T BEZ235 2
Hs 578T Dactolisib 2 72
1.0
728.5 3555.0 624.7
0.0
0.063 0.205 2.509
Hs578T BEZ235 2
Hs 578T Dactolisib 2 72
3.2
532.5 3555.0 624.7
0.505
-0.062 0.150 2.509
Hs578T BEZ235 2
Hs 578T Buparlisib 2 72
0.001
3710.0 3566.8 624.7
-3.0
1.030 1.040 2.513
Hs578T BKM120 2
Hs 578T Buparlisib 2 72
0.0032
3593.8 3566.8 624.7
-2.49
1.010 1.010 2.513
Hs578T BKM120 2
Hs 578T Buparlisib 2 72
0.01
3527.8 3566.8 624.7
-2.0
0.991 0.989 2.513
Hs578T BKM120 2
Hs 578T Buparlisib 2 72
0.032
3475.3 3566.8 624.7
-1.49
0.979 0.974 2.513
Hs578T BKM120 2
Hs 578T Buparlisib 2 72
0.1
3150.3 3566.8 624.7
-1.0
0.904 0.883 2.513
Hs578T BKM120 2
Hs 578T Buparlisib 2 72
0.32
2526.5 3566.8 624.7
-0.495
0.744 0.708 2.513
Hs578T BKM120 2
Hs 578T Buparlisib 2 72
1.0
1255.0 3566.8 624.7
0.0
0.320 0.352 2.513
Hs578T BKM120 2
Hs 578T Buparlisib 2 72
3.2
158.8 3566.8 624.7
0.505
-0.420 0.045 2.513
Hs578T BKM120 2
Hs 578T BX-912 2 72
0.001
3521.3 3632.8 624.7
-3.0
0.976 0.969 2.540
Hs578T BX912 2
Hs 578T BX-912 2 72
0.0032
3582.0 3632.8 624.7
-2.49
0.989 0.986 2.540
Hs578T BX912 2
Hs 578T BX-912 2 72
0.01
3561.8 3632.8 624.7
-2.0
0.985 0.980 2.540
Hs578T BX912 2
Hs 578T BX-912 2 72
0.032
3564.0 3632.8 624.7
-1.49
0.985 0.981 2.540
Hs578T BX912 2
Hs 578T BX-912 2 72
0.1
3390.3 3632.8 624.7
-1.0
0.946 0.933 2.540
Hs578T BX912 2
Hs 578T BX-912 2 72
0.32
3091.5 3632.8 624.7
-0.495
0.877 0.851 2.540
Hs578T BX912 2
Hs 578T BX-912 2 72
1.0
1822.8 3632.8 624.7
0.0
0.524 0.502 2.540
Hs578T BX912 2
Hs 578T BX-912 2 72
3.2
595.0 3632.8 624.7
0.505
-0.019 0.164 2.540
Hs578T BX912 2
Hs 578T Alpelisib 2 72
0.001
2972.3 3566.3 624.7
-3.0
0.860 0.833 2.513
Hs578T BYL719 2
Hs 578T Alpelisib 2 72
0.0032
2946.5 3566.3 624.7
-2.49
0.854 0.826 2.513
Hs578T BYL719 2
Hs 578T Alpelisib 2 72
0.01
3462.0 3566.3 624.7
-2.0
0.977 0.971 2.513
Hs578T BYL719 2
Hs 578T Alpelisib 2 72
0.032
3302.8 3566.3 624.7
-1.49
0.940 0.926 2.513
Hs578T BYL719 2
Hs 578T Alpelisib 2 72
0.1
3269.8 3566.3 624.7
-1.0
0.932 0.917 2.513
Hs578T BYL719 2