5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| 5z-7-oxozeaenol | BCWM.1 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | 25.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | ACK | TVSVAVKCLKPDVLSQPEAMDDFIR | Lys1 | 18.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | AGK | ATVFLNPAACKGK | Other | 4.9 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | 14.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | ARAF | DLKSNNIFLHEGLTVK | Lys2 | -81.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | ATR | FYIMMCKPK | ATP | 28.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | AurA | FILALKVLFK | Lys1 | -4.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | AurB | SHFIVALKVLFK | Lys1 | -12.9 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | BARK1 | DLKPANILLDEHGHVR | Lys2 | 25.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | BRAF | DLKSNNIFLHEDLTVK | Lys2 | 2.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | -2.2 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CAMK1D | LFAVKCIPK | Lys1 | 11.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CaMK2g | TSTQEYAAKIINTK | Lys1 | 20.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | KCC4 | DLKPENLLYATPAPDAPLK | Lys2 | 16.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CaMKK2 | DIKPSNLLVGEDGHIK | Lys2 | 8.9 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CASK | ETGQQFAVKIVDVAK | Lys1 | -20.9 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | 9.4 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CDK11,CDK8 | DLKPANILVMGEGPER | Lys2 | 7.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CDK2 | DLKPQNLLINTEGAIK | Lys2 | 5.0 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CDK4 | DLKPENILVTSGGTVK | Lys2 | 21.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CDK5 | DLKPQNLLINR | Lys2 | 9.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CDK6 | DLKPQNILVTSSGQIK | Lys2 | 10.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CDK7 | DLKPNNLLLDENGVLK | Lys2 | -3.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CDK9 | DMKAANVLITR | Lys2 | 25.0 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CHK1 | DIKPENLLLDER | Lys2 | 13.3 | 1 | uM |