5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
5z-7-oxozeaenol MWCL.1 RSK1_domain2
DLKPSNILYVDESGNPECLR
Lys2
8.1
1
uM
5z-7-oxozeaenol MWCL.1 RSK1,RSK2,RSK3_domain1
DLKPENILLDEEGHIK
Lys2
3.3
1
uM
5z-7-oxozeaenol MWCL.1 RSK2_domain2
DLKPSNILYVDESGNPESIR
Lys2
-2.4
1
uM
5z-7-oxozeaenol MWCL.1 RSK3_domain1
DLKPENILLDEEGHIKITDFGLSK
Lys2
11.6
1
uM
5z-7-oxozeaenol MWCL.1 RSKL1_domain1
VLGVIDKVLLVMDTR
Protein Kinase Domain
1.7
1
uM
5z-7-oxozeaenol MWCL.1 SRPK1/2
FVAMKVVK
Lys1
32.2
1
uM
5z-7-oxozeaenol MWCL.1 MAP3K7,TAK1
DLKPPNLLLVAGGTVLK
Lys2
> 81
1
uM
5z-7-oxozeaenol MWCL.1 TAO1,TAOK3
DIKAGNILLTEPGQVK
Lys2
25.6
1
uM
5z-7-oxozeaenol MWCL.1 TAOK2
DVKAGNILLSEPGLVK
Lys2
31.8
1
uM
5z-7-oxozeaenol MWCL.1 TLK1/2
YLNEIKPPIIHYDLKPGNILLVNGTACGEIK
Lys2
-25.0
1
uM
5z-7-oxozeaenol MWCL.1 TYK2(Kin.Dom.2)
IGDFGLAKAVPEGHEYYR
Activation Loop
19.1
1
uM