5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| 5z-7-oxozeaenol | MWCL.1 | VRK2 | MLDVLEYIHENEYVHGDIKAANLLLGYK | Lys2 | 18.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | WEE1 | YIHSMSLVHMDIKPSNIFISR | Lys2 | 1 | uM | |
| 5z-7-oxozeaenol | MWCL.1 | Wnk1,Wnk2 | GSFKTVYK | ATP Loop | -19.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | Lys2 | -0.7 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIKGQNVLLTENAEVK | Lys2 | 12.4 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ZC2/TNIK | TGQLAAIKVMDVTGDEEEEIKQEINMLKK | Lys1 | 47.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | KCC2D | IPTGQEYAAKIINTKK | Lys1 | 4.0 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | KC1A | DIKPDNFLMGIGR | Lys2 | 26.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | KC1G2 | DVKPENFLVGRPGTK | Lys2 | 6.9 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | FRAP1 | IQSIAPSLQVITSKQRPR | ATP | -3.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | GCN2_domain2 | DLKPVNIFLDSDDHVK | Lys2 | 4.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | JAK1_domain2 | IGDFGLTKAIETDKEYYTVK | Activation Loop | 22.9 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | M4K3 | NVNTGELAAIKVIK | Lys1 | 1 | uM | |
| 5z-7-oxozeaenol | MWCL.1 | MP2K7 | DVKPSNILLDER | Lys2 | 28.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | M3K2 | ELAVKQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | -16.8 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | M3K2,MAP3K3 | DIKGANILR | Lys2 | -4.7 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MSK1_domain1 | DIKLENILLDSNGHVVLTDFGLSK | Lys2 | 7.7 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MK14 | QELNKTIWEVPER | Other | 16.7 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MK11 | QELNKTVWEVPQR | Other | 17.4 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | KS6B1 | DLKPENIMLNHQGHVK | Lys2 | 15.7 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | KS6B2 | DLKPENIMLSSQGHIK | Lys2 | 26.0 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CDK16 | SKLTDNLVALKEIR | Lys1 | 1 | uM | |
| 5z-7-oxozeaenol | MWCL.1 | CDK14 | LVALKVIR | Lys1 | -17.9 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | PI42C | TLVIKEVSSEDIADMHSNLSNYHQYIVK | ATP | -10.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | FAK2 | YIEDEDYYKASVTR | Activation Loop | -9.5 | 1 | uM |