5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| 5z-7-oxozeaenol | BCWM.1 | NDR1 | DIKPDNLLLDSK | Lys2 | -5.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | NDR2 | DIKPDNLLLDAK | Lys2 | 2.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | NEK1 | DIKSQNIFLTK | Lys2 | 9.4 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | NEK2 | DLKPANVFLDGK | Lys2 | 15.9 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | NEK3 | SKNIFLTQNGK | Activation Loop | -6.9 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | NEK4 | DLKTQNVFLTR | Lys2 | 8.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | NEK6,NEK7 | DIKPANVFITATGVVK | Lys2 | 7.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | NEK7 | AACLLDGVPVALKK | Lys1 | 16.2 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | NEK8 | DLKTQNILLDK | Lys2 | -1.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | NEK9 | DIKTLNIFLTK | Lys2 | 15.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | OSR1 | DVKAGNILLGEDGSVQIADFGVSAFLATGGDITR | Lys2 | 9.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | p38a | DLKPSNLAVNEDCELK | Lys2 | 13.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | p38d,p38g | DLKPGNLAVNEDCELK | Lys2 | -0.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | PAN3 | VMDPTKILITGK | ATP | 5.9 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | PCTAIRE2,PCTAIRE3 | SKLTENLVALKEIR | Lys1 | -11.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | PDHK1 | SPGQPIQVVYVPSHLYHMVFELFKNAMR | Other | 1 | uM | |
| 5z-7-oxozeaenol | BCWM.1 | PDK1 | EYAIKILEK | Lys1 | -15.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | PEK | DLKPSNIFFTMDDVVK | Lys2 | 17.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | PHKg1 | DLKPENILLDDNMNIK | Lys2 | -1.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | PHKg2 | ATGHEFAVKIMEVTAER | Lys1 | 4.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | PI4KA,PI4KAP2 | SGTPMQSAAKAPYLAK | ATP | 32.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | PI4KB | VPHTQAVVLNSKDK | ATP | 19.2 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | PIK3C2B | VIFKCGDDLRQDMLTLQMIR | ATP | 13.0 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | PIK3C3 | TEDGGKYPVIFKHGDDLR | ATP | 14.2 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | PIK3CB | VFGEDSVGVIFKNGDDLRQDMLTLQMLR | ATP | 38.0 | 1 | uM |