5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
5z-7-oxozeaenol | BCWM.1 | MAP3K1 | DVKGANLLIDSTGQR | Lys2 | 24.7 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MAP3K3 | ELASKQVQFDPDSPETSKEVSALECEIQLLK | Lys1 | -2.8 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MAP3K4 | DIKGANIFLTSSGLIK | Lys2 | -2.1 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MAP3K5 | DIKGDNVLINTYSGVLK | Lys2 | 1.5 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | M3K6 | DIKGDNVLINTFSGLLK | Lys2 | -32.1 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MARK2,MARK3 | DLKAENLLLDADMNIK | Lys2 | 22.1 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MARK3 | EVAIKIIDKTQLNPTSLQK | Lys1 | 11.5 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MARK3,MARK4 | EVAIKIIDK | Lys1 | 2.1 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MARK4 | DLKAENLLLDAEANIK | Lys2 | -5.7 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MAST1,MAST2 | DLKPDNLLITSMGHIK | Lys2 | 39.2 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MAST3 | DLKPDNLLITSLGHIK | Lys2 | 8.3 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MASTL | GAFGKVYLGQK | ATP Loop | 7.9 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MASTL | LYAVKVVK | Lys1 | 11.4 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MELK | DLKPENLLFDEYHK | Lys2 | 14.1 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MER,TYRO3 | KIYSGDYYR | Activation Loop | 14.0 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MLK3 | DLKSNNILLLQPIESDDMEHK | Lys2 | 17.1 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MLK4 | DLKSSNILLLEK | Lys2 | 5.7 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MLKL | APVAIKVFK | Lys1 | 2.5 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MSK2 domain1 | DLKLENVLLDSEGHIVLTDFGLSK | Lys2 | 15.4 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MST1 | ETGQIVAIKQVPVESDLQEIIK | Lys1 | -10.7 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MST2 | ESGQVVAIKQVPVESDLQEIIK | Lys1 | -6.0 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MST3 | DIKAANVLLSEHGEVK | Lys2 | 16.7 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MST4 | TQQVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSSYVTK | Lys1 | 37.3 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MST4,YSK1 | DIKAANVLLSEQGDVK | Lys2 | 13.8 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MYO3A,MYO3B | DVKGNNILLTTEGGVK | Lys2 | 7.7 | 1 | uM |