5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
5z-7-oxozeaenol BCWM.1 MAP3K1
DVKGANLLIDSTGQR
Lys2
24.7
1
uM
5z-7-oxozeaenol BCWM.1 MAP3K3
ELASKQVQFDPDSPETSKEVSALECEIQLLK
Lys1
-2.8
1
uM
5z-7-oxozeaenol BCWM.1 MAP3K4
DIKGANIFLTSSGLIK
Lys2
-2.1
1
uM
5z-7-oxozeaenol BCWM.1 MAP3K5
DIKGDNVLINTYSGVLK
Lys2
1.5
1
uM
5z-7-oxozeaenol BCWM.1 M3K6
DIKGDNVLINTFSGLLK
Lys2
-32.1
1
uM
5z-7-oxozeaenol BCWM.1 MARK2,MARK3
DLKAENLLLDADMNIK
Lys2
22.1
1
uM
5z-7-oxozeaenol BCWM.1 MARK3
EVAIKIIDKTQLNPTSLQK
Lys1
11.5
1
uM
5z-7-oxozeaenol BCWM.1 MARK3,MARK4
EVAIKIIDK
Lys1
2.1
1
uM
5z-7-oxozeaenol BCWM.1 MARK4
DLKAENLLLDAEANIK
Lys2
-5.7
1
uM
5z-7-oxozeaenol BCWM.1 MAST1,MAST2
DLKPDNLLITSMGHIK
Lys2
39.2
1
uM
5z-7-oxozeaenol BCWM.1 MAST3
DLKPDNLLITSLGHIK
Lys2
8.3
1
uM
5z-7-oxozeaenol BCWM.1 MASTL
GAFGKVYLGQK
ATP Loop
7.9
1
uM
5z-7-oxozeaenol BCWM.1 MASTL
LYAVKVVK
Lys1
11.4
1
uM
5z-7-oxozeaenol BCWM.1 MELK
DLKPENLLFDEYHK
Lys2
14.1
1
uM
5z-7-oxozeaenol BCWM.1 MER,TYRO3
KIYSGDYYR
Activation Loop
14.0
1
uM
5z-7-oxozeaenol BCWM.1 MLK3
DLKSNNILLLQPIESDDMEHK
Lys2
17.1
1
uM
5z-7-oxozeaenol BCWM.1 MLK4
DLKSSNILLLEK
Lys2
5.7
1
uM
5z-7-oxozeaenol BCWM.1 MLKL
APVAIKVFK
Lys1
2.5
1
uM
5z-7-oxozeaenol BCWM.1 MSK2 domain1
DLKLENVLLDSEGHIVLTDFGLSK
Lys2
15.4
1
uM
5z-7-oxozeaenol BCWM.1 MST1
ETGQIVAIKQVPVESDLQEIIK
Lys1
-10.7
1
uM
5z-7-oxozeaenol BCWM.1 MST2
ESGQVVAIKQVPVESDLQEIIK
Lys1
-6.0
1
uM
5z-7-oxozeaenol BCWM.1 MST3
DIKAANVLLSEHGEVK
Lys2
16.7
1
uM
5z-7-oxozeaenol BCWM.1 MST4
TQQVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSSYVTK
Lys1
37.3
1
uM
5z-7-oxozeaenol BCWM.1 MST4,YSK1
DIKAANVLLSEQGDVK
Lys2
13.8
1
uM
5z-7-oxozeaenol BCWM.1 MYO3A,MYO3B
DVKGNNILLTTEGGVK
Lys2
7.7
1
uM