5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| 5z-7-oxozeaenol | BCWM.1 | IKKE | SGELVAVKVFNTTSYLRPR | Lys1 | 7.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | ILK | WQGNDIVVKVLK | Lys1 | 3.0 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | IRAK1 | AIQFLHQDSPSLIHGDIKSSNVLLDER | Lys2 | -31.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | IRAK4 | DIKSANILLDEAFTAK | Lys2 | -1.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | IRE1 | DLKPHNILISMPNAHGK | Lys2 | 19.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | ITPK1 | ESIFFNSHNVSKPESSSVLTELDKIEGVFERPSDEVIR | Other | -37.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | JAK1 | QLASALSYLEDKDLVHGNVCTKNLLLAR | Other | 24.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | JAK3 domain2 | IADFGLAKLLPLDKDYYVVR | Activation Loop | 21.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | JNK1,JNK2,JNK3 | DLKPSNIVVK | Lys2 | 3.2 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | KHS1 | NVHTGELAAVKIIK | Lys1 | -0.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | KSR1 | SKNVFYDNGKVVITDFGLFGISGVVR | Activation Loop | 51.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | KSR1,KSR2 | SKNVFYDNGK | Activation Loop | 59.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | LATS1 | ALYATKTLR | Lys1 | 11.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | LATS2 | DIKPDNILIDLDGHIK | Lys2 | -11.0 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | LCK | EGAKFPIKWTAPEAINYGTFTIK | Activation Loop | 15.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | LKB1 | DIKPGNLLLTTGGTLK | Lys2 | 9.4 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | LOK | DLKAGNVLMTLEGDIR | Lys2 | 10.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | LRRK2 | DLKPHNVLLFTLYPNAAIIAK | Lys2 | -19.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | LYN | VAVKTLKPGTMSVQAFLEEANLMK | Lys1 | 21.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | MAP2K1 | IMHRDVKPSNILVNSR | Lys2 | > 98 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | MAP2K1,MAP2K2 | DVKPSNILVNSR | Lys2 | 97.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | MAP2K3 | DVKPSNVLINK | Lys2 | 51.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | MAP2K4 | DIKPSNILLDR | Lys2 | -6.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | MAP2K5 | DVKPSNMLVNTR | Lys2 | > 98 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | MAP2K6 | DVKPSNVLINALGQVK | Lys2 | 91.8 | 1 | uM |