5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| 5z-7-oxozeaenol | BCWM.1 | CHK2 | DLKPENVLLSSQEEDCLIK | Lys2 | -12.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CK1d,CK1e | DVKPDNFLMGLGKK | Lys2 | 11.9 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CK2a2 | DVKPHNVMIDHQQK | Lys2 | 16.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CLK3 | YEIVGNLGEGTFGKVVECLDHAR | ATP Loop | 1 | uM | |
| 5z-7-oxozeaenol | BCWM.1 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | 3.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | DGKA | IDPVPNTHPLLVFVNPKSGGK | ATP | -5.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | DNAPK | EHPFLVKGGEDLR | ATP | 19.2 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | DNAPK | KGGSWIQEINVAEK | ATP | -26.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | eEF2K | YIKYNSNSGFVR | ATP | -19.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | EPHB1 | YLQDDTSDPTYTSSLGGKIPVR | Activation Loop | 7.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | EPHB2 | FLEDDTSDPTYTSALGGKIPIR | Activation Loop | 8.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | MK03 | DLKPSNLLINTTCDLK | Lys2 | 4.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | MK01 | DLKPSNLLLNTTCDLK | Lys2 | 4.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | Erk5 | DLKPSNLLVNENCELK | Lys2 | 21.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | FER | TSVAVKTCKEDLPQELK | Lys1 | 1.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | FES | LRADNTLVAVKSCR | Lys1 | -9.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | FGR | LIKDDEYNPCQGSKFPIK | Activation Loop | 12.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | FRK | HEIKLPVK | Activation Loop | 18.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | FYN,SRC,YES | QGAKFPIKWTAPEAALYGR | Activation Loop | 5.4 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | GCK | DIKGANLLLTLQGDVK | Lys2 | -5.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | GSK3A | DIKPQNLLVDPDTAVLK | Lys2 | 10.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | GSK3B | DIKPQNLLLDPDTAVLK | Lys2 | 5.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | HPK1 | DIKGANILINDAGEVR | Lys2 | -2.9 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | IKKA | DLKPENIVLQDVGGK | Lys2 | -1.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | IKKB | DLKPENIVLQQGEQR | Lys2 | -8.8 | 1 | uM |