5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| 5z-7-oxozeaenol | MWCL.1 | MARK3,MARK4 | EVAIKIIDK | Lys1 | -16.7 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MARK4 | DLKAENLLLDAEANIK | Lys2 | 1 | uM | |
| 5z-7-oxozeaenol | MWCL.1 | MAST1,MAST2 | DLKPDNLLITSMGHIK | Lys2 | 41.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MAST3 | DLKPDNLLITSLGHIK | Lys2 | -1.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MASTL | GAFGKVYLGQK | ATP Loop | -3.7 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MASTL | LYAVKVVK | Lys1 | 1.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MELK | DLKPENLLFDEYHK | Lys2 | 12.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MER,TYRO3 | KIYSGDYYR | Activation Loop | 1 | uM | |
| 5z-7-oxozeaenol | MWCL.1 | MLK3 | DLKSNNILLLQPIESDDMEHK | Lys2 | 20.0 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MLK4 | DLKSSNILLLEK | Lys2 | 1 | uM | |
| 5z-7-oxozeaenol | MWCL.1 | MLKL | APVAIKVFK | Lys1 | -13.8 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MSK2 domain1 | DLKLENVLLDSEGHIVLTDFGLSK | Lys2 | 36.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MST1 | ETGQIVAIKQVPVESDLQEIIK | Lys1 | -11.0 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MST2 | ESGQVVAIKQVPVESDLQEIIK | Lys1 | -12.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MST3 | DIKAANVLLSEHGEVK | Lys2 | -2.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MST4 | TQQVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSSYVTK | Lys1 | 31.2 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MST4,YSK1 | DIKAANVLLSEQGDVK | Lys2 | 9.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | MYO3A,MYO3B | DVKGNNILLTTEGGVK | Lys2 | 2.9 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | NDR1 | DIKPDNLLLDSK | Lys2 | -6.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | NDR2 | DIKPDNLLLDAK | Lys2 | -3.9 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | NEK1 | DIKSQNIFLTK | Lys2 | -11.9 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | NEK2 | DLKPANVFLDGK | Lys2 | -8.2 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | NEK3 | SKNIFLTQNGK | Activation Loop | 18.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | NEK4 | DLKTQNVFLTR | Lys2 | -6.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | NEK6,NEK7 | DIKPANVFITATGVVK | Lys2 | -3.6 | 1 | uM |