5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| 5z-7-oxozeaenol | MWCL.1 | PKN1 | VLLSEFRPSGELFAIKALK | Lys1 | -9.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | PKR | DLKPSNIFLVDTK | Lys2 | -4.4 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | PLK1 | CFEISDADTKEVFAGKIVPK | Lys1 | 0.2 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | PRP4 | CNILHADIKPDNILVNESK | Lys2 | 0.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | PRPK | FLSGLELVKQGAEAR | ATP Loop | 22.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | RIPK2 | VQVAVKHLHIHTPLLDSER | Lys1 | 1 | uM | |
| 5z-7-oxozeaenol | MWCL.1 | RIPK3 | DLKPSNVLLDPELHVK | Lys2 | 20.0 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ROCK1,ROCK2 | DVKPDNMLLDK | Lys2 | 16.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | RSK1 domain1 | DLKPENILLDEEGHIKLTDFGLSKEAIDHEK | Lys2 | 24.4 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | RSK2 domain1 | DLKPENILLDEEGHIKLTDFGLSKESIDHEK | Lys2 | 32.7 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | RSK4 domain1 | DLKPENILLDEIGHIK | Lys2 | 1 | uM | |
| 5z-7-oxozeaenol | MWCL.1 | SGK3 | FYAVKVLQK | Lys1 | -20.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | SLK | DLKAGNILFTLDGDIK | Lys2 | 3.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | SMG1 | DTVTIHSVGGTITILPTKTKPK | ATP | 2.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | SNRK | DLKPENVVFFEK | Lys2 | -5.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | SRPK1 | IIHTDIKPENILLSVNEQYIR | Lys2 | -1.2 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | STK33 | DLKLENIMVK | Lys2 | 18.0 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | STLK5 | YSVKVLPWLSPEVLQQNLQGYDAK | Activation Loop | 2.7 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | STLK6 | HTPTGTLVTIKITNLENCNEER | Lys1 | 0.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | SYK | ISDFGLSKALR | Activation Loop | 10.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | TBK1 | TGDLFAIKVFNNISFLRPVDVQMR | Lys1 | 32.9 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | TEC | YVLDDQYTSSSGAKFPVK | Activation Loop | 19.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | Lys2 | 5.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ULK1 | DLKPQNILLSNPAGR | Lys2 | 9.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ULK3 | NISHLDLKPQNILLSSLEKPHLK | Lys2 | -3.7 | 1 | uM |