5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
5z-7-oxozeaenol | MWCL.1 | LKB1 | DIKPGNLLLTTGGTLK | Lys2 | 0.0 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | FER | TSVAVKTCKEDLPQELK | Lys1 | 0.2 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PLK1 | CFEISDADTKEVFAGKIVPK | Lys1 | 0.2 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PIK3CD | VNWLAHNVSKDNRQ | ATP | -0.3 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | STLK6 | HTPTGTLVTIKITNLENCNEER | Lys1 | 0.3 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | SYK | ISDFGLSKALR | Activation Loop | -0.4 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PRP4 | CNILHADIKPDNILVNESK | Lys2 | 0.6 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | p38d,p38g | DLKPGNLAVNEDCELK | Lys2 | -0.7 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | KHS1 | NVHTGELAAVKIIK | Lys1 | -0.7 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | Lys2 | -0.7 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | GSK3B | DIKPQNLLLDPDTAVLK | Lys2 | 0.7 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | ULK1 | DLKPQNILLSNPAGR | Lys2 | -0.8 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | SRPK1 | IIHTDIKPENILLSVNEQYIR | Lys2 | -1.0 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | ILK | WQGNDIVVKVLK | Lys1 | -10.0 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | ULK3 | NISHLDLKPQNILLSSLEKPHLK | Lys2 | -10.1 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | CDK6 | DLKPQNILVTSSGQIK | Lys2 | 10.3 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PI4KB | VPHTQAVVLNSKDK | ATP | -10.4 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | PI42C | TLVIKEVSSEDIADMHSNLSNYHQYIVK | ATP | -10.6 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | SYK | ISDFGLSKALR | Activation Loop | 10.6 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | MST1 | ETGQIVAIKQVPVESDLQEIIK | Lys1 | -10.7 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | LOK | DLKAGNVLMTLEGDIR | Lys2 | 10.7 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | CDK16 | SKLTDNLVALKEIR | Lys1 | -10.8 | 1 | uM |
5z-7-oxozeaenol | BCWM.1 | GSK3A | DIKPQNLLVDPDTAVLK | Lys2 | 10.8 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | MASTL | LYAVKVVK | Lys1 | 1.1 | 1 | uM |
5z-7-oxozeaenol | MWCL.1 | MK01 | DLKPSNLLLNTTCDLK | Lys2 | 1.1 | 1 | uM |