5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
5z-7-oxozeaenol MWCL.1 LKB1
DIKPGNLLLTTGGTLK
Lys2
0.0
1
uM
5z-7-oxozeaenol MWCL.1 FER
TSVAVKTCKEDLPQELK
Lys1
0.2
1
uM
5z-7-oxozeaenol MWCL.1 PLK1
CFEISDADTKEVFAGKIVPK
Lys1
0.2
1
uM
5z-7-oxozeaenol MWCL.1 PIK3CD
VNWLAHNVSKDNRQ
ATP
-0.3
1
uM
5z-7-oxozeaenol MWCL.1 STLK6
HTPTGTLVTIKITNLENCNEER
Lys1
0.3
1
uM
5z-7-oxozeaenol BCWM.1 SYK
ISDFGLSKALR
Activation Loop
-0.4
1
uM
5z-7-oxozeaenol MWCL.1 PRP4
CNILHADIKPDNILVNESK
Lys2
0.6
1
uM
5z-7-oxozeaenol BCWM.1 p38d,p38g
DLKPGNLAVNEDCELK
Lys2
-0.7
1
uM
5z-7-oxozeaenol BCWM.1 KHS1
NVHTGELAAVKIIK
Lys1
-0.7
1
uM
5z-7-oxozeaenol MWCL.1 Wnk1,Wnk2,Wnk3
DLKCDNIFITGPTGSVK
Lys2
-0.7
1
uM
5z-7-oxozeaenol MWCL.1 GSK3B
DIKPQNLLLDPDTAVLK
Lys2
0.7
1
uM
5z-7-oxozeaenol BCWM.1 ULK1
DLKPQNILLSNPAGR
Lys2
-0.8
1
uM
5z-7-oxozeaenol BCWM.1 SRPK1
IIHTDIKPENILLSVNEQYIR
Lys2
-1.0
1
uM
5z-7-oxozeaenol MWCL.1 ILK
WQGNDIVVKVLK
Lys1
-10.0
1
uM
5z-7-oxozeaenol BCWM.1 ULK3
NISHLDLKPQNILLSSLEKPHLK
Lys2
-10.1
1
uM
5z-7-oxozeaenol BCWM.1 CDK6
DLKPQNILVTSSGQIK
Lys2
10.3
1
uM
5z-7-oxozeaenol MWCL.1 PI4KB
VPHTQAVVLNSKDK
ATP
-10.4
1
uM
5z-7-oxozeaenol MWCL.1 PI42C
TLVIKEVSSEDIADMHSNLSNYHQYIVK
ATP
-10.6
1
uM
5z-7-oxozeaenol MWCL.1 SYK
ISDFGLSKALR
Activation Loop
10.6
1
uM
5z-7-oxozeaenol BCWM.1 MST1
ETGQIVAIKQVPVESDLQEIIK
Lys1
-10.7
1
uM
5z-7-oxozeaenol BCWM.1 LOK
DLKAGNVLMTLEGDIR
Lys2
10.7
1
uM
5z-7-oxozeaenol BCWM.1 CDK16
SKLTDNLVALKEIR
Lys1
-10.8
1
uM
5z-7-oxozeaenol BCWM.1 GSK3A
DIKPQNLLVDPDTAVLK
Lys2
10.8
1
uM
5z-7-oxozeaenol MWCL.1 MASTL
LYAVKVVK
Lys1
1.1
1
uM
5z-7-oxozeaenol MWCL.1 MK01
DLKPSNLLLNTTCDLK
Lys2
1.1
1
uM
  • Page 1 of 16
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