5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| 5z-7-oxozeaenol | BCWM.1 | TYK2(Kin.Dom.2) | IGDFGLAKAVPEGHEYYR | Activation Loop | 11.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | -3.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | SYK | ISDFGLSKALR | Activation Loop | -0.4 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | FAK2 | YIEDEDYYKASVTR | Activation Loop | 27.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | -1.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | MER,TYRO3 | KIYSGDYYR | Activation Loop | 14.0 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | STLK5 | YSVKVLPWLSPEVLQQNLQGYDAK | Activation Loop | -31.2 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | KSR1 | SKNVFYDNGKVVITDFGLFGISGVVR | Activation Loop | 51.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | JAK1_domain2 | IGDFGLTKAIETDKEYYTVK | Activation Loop | 5.9 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | EPHB2 | FLEDDTSDPTYTSALGGKIPIR | Activation Loop | 8.8 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | 25.9 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | FGR | LIKDDEYNPCQGSKFPIK | Activation Loop | 12.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | FRK | HEIKLPVK | Activation Loop | 18.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | NEK3 | SKNIFLTQNGK | Activation Loop | -6.9 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | 25.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | LCK | EGAKFPIKWTAPEAINYGTFTIK | Activation Loop | 15.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | 3.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | JAK3 domain2 | IADFGLAKLLPLDKDYYVVR | Activation Loop | 21.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | KSR1,KSR2 | SKNVFYDNGK | Activation Loop | 59.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | TEC | YVLDDQYTSSSGAKFPVK | Activation Loop | 16.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | -2.2 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | EPHB1 | YLQDDTSDPTYTSSLGGKIPVR | Activation Loop | 7.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | FYN,SRC,YES | QGAKFPIKWTAPEAALYGR | Activation Loop | 5.4 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | EPHB2 | FLEDDTSDPTYTSALGGKIPIR | Activation Loop | 1 | uM | |
| 5z-7-oxozeaenol | MWCL.1 | EPHB1 | YLQDDTSDPTYTSSLGGKIPVR | Activation Loop | 12.7 | 1 | uM |