5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| 5z-7-oxozeaenol | BCWM.1 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | 25.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | 25.9 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | ACK | TVSVAVKCLKPDVLSQPEAMDDFIR | Lys1 | 18.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ACK | TVSVAVKCLKPDVLSQPEAMDDFIR | Lys1 | 17.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | AGK | ATVFLNPAACKGK | Other | 1 | uM | |
| 5z-7-oxozeaenol | BCWM.1 | AGK | ATVFLNPAACKGK | Other | 4.9 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | 23.0 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | 14.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | ARAF | DLKSNNIFLHEGLTVK | Lys2 | -81.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ARAF | DLKSNNIFLHEGLTVK | Lys2 | -120.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | ATR | FYIMMCKPK | ATP | 28.8 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ATR | FYIMMCKPK | ATP | 28.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | AurA | FILALKVLFK | Lys1 | -15.2 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | AurA | FILALKVLFK | Lys1 | -4.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | AurB | SHFIVALKVLFK | Lys1 | -23.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | AurB | SHFIVALKVLFK | Lys1 | -12.9 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | BARK1 | DLKPANILLDEHGHVR | Lys2 | 31.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | BARK1 | DLKPANILLDEHGHVR | Lys2 | 25.8 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | BRAF | DLKSNNIFLHEDLTVK | Lys2 | -9.2 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | BRAF | DLKSNNIFLHEDLTVK | Lys2 | 2.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | -1.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | -2.2 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CAMK1D | LFAVKCIPK | Lys1 | 2.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CAMK1D | LFAVKCIPK | Lys1 | 11.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CaMK2g | TSTQEYAAKIINTK | Lys1 | 20.7 | 1 | uM |