5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| 5z-7-oxozeaenol | BCWM.1 | ZC2/TNIK | TGQLAAIKVMDVTGDEEEEIKQEINMLKK | Lys1 | 40.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ZC2/TNIK | TGQLAAIKVMDVTGDEEEEIKQEINMLKK | Lys1 | 47.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIKGQNVLLTENAEVK | Lys2 | 16.0 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIKGQNVLLTENAEVK | Lys2 | 12.4 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | Lys2 | 14.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | Lys2 | -0.7 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | Wnk1,Wnk2 | GSFKTVYK | ATP Loop | -19.3 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | Wnk1,Wnk2 | GSFKTVYK | ATP Loop | 7.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | WEE1 | YIHSMSLVHMDIKPSNIFISR | Lys2 | 23.0 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | WEE1 | YIHSMSLVHMDIKPSNIFISR | Lys2 | 1 | uM | |
| 5z-7-oxozeaenol | BCWM.1 | VRK2 | MLDVLEYIHENEYVHGDIKAANLLLGYK | Lys2 | 24.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | VRK2 | MLDVLEYIHENEYVHGDIKAANLLLGYK | Lys2 | 18.6 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | ULK3 | NISHLDLKPQNILLSSLEKPHLK | Lys2 | -10.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ULK3 | NISHLDLKPQNILLSSLEKPHLK | Lys2 | -3.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | ULK1 | DLKPQNILLSNPAGR | Lys2 | -0.8 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ULK1 | DLKPQNILLSNPAGR | Lys2 | 9.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | TYK2(Kin.Dom.2) | IGDFGLAKAVPEGHEYYR | Activation Loop | 19.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | TYK2(Kin.Dom.2) | IGDFGLAKAVPEGHEYYR | Activation Loop | 11.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | TLK1/2 | YLNEIKPPIIHYDLKPGNILLVNGTACGEIK | Lys2 | -25.0 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | TLK1/2 | YLNEIKPPIIHYDLKPGNILLVNGTACGEIK | Lys2 | 2.4 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | Lys2 | 5.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | Lys2 | -2.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | TEC | YVLDDQYTSSSGAKFPVK | Activation Loop | 19.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | TEC | YVLDDQYTSSSGAKFPVK | Activation Loop | 16.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | TBK1 | TGDLFAIKVFNNISFLRPVDVQMR | Lys1 | 9.9 | 1 | uM |