Breast Cancer Profiling Project, Drug Sensitivity phase I: Fixed-cell GR measures of 35 breast cell lines to 34 small molecule perturbagens from library plate I. Dataset 1 of 2: Normalized growth rate inhibition values - Dataset (ID:20343)
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Cell | Small Molecule | Small Mol Concentration (uM) | Primary Target | Pathway | Mean Normalized Growth Rate Inhibition Value | Increased Fraction Dead |
---|---|---|---|---|---|---|
BT-20 | Saracatinib | 1.0 | SRC | MAPK/nRTK | 0.7638 | 0.04930 |
BT-20 | Saracatinib | 3.1623 | SRC | MAPK/nRTK | 0.6128 | 0.07032 |
BT-20 | Saracatinib | 10.0 | SRC | MAPK/nRTK | 0.3103 | 0.12644 |
BT-20 | ABT-737 | 0.001 | Bcl2/XL | Misc | 1.0936 | 0.00187 |
BT-20 | ABT-737 | 0.0031623 | Bcl2/XL | Misc | 1.0529 | 0.00292 |
BT-20 | ABT-737 | 0.01 | Bcl2/XL | Misc | 1.0586 | 0.00276 |
BT-20 | ABT-737 | 0.031623 | Bcl2/XL | Misc | 1.0481 | 0.01277 |
BT-20 | ABT-737 | 0.1 | Bcl2/XL | Misc | 1.0162 | 0.01978 |
BT-20 | ABT-737 | 0.31623 | Bcl2/XL | Misc | 0.9870 | 0.02911 |
BT-20 | ABT-737 | 1.0 | Bcl2/XL | Misc | 0.9351 | 0.04831 |
BT-20 | ABT-737 | 3.1623 | Bcl2/XL | Misc | 0.8923 | 0.07580 |
BT-20 | ABT-737 | 10.0 | Bcl2/XL | Misc | 0.5926 | 0.16414 |
BT-20 | Vorinostat | 0.001 | HDAC | Misc | 1.0736 | -0.00774 |
BT-20 | Vorinostat | 0.0031623 | HDAC | Misc | 1.0276 | -0.00162 |
BT-20 | Vorinostat | 0.01 | HDAC | Misc | 1.0801 | -0.00840 |
BT-20 | Vorinostat | 0.031623 | HDAC | Misc | 1.0906 | 0.00068 |
BT-20 | Vorinostat | 0.1 | HDAC | Misc | 1.0164 | 0.00615 |
BT-20 | Vorinostat | 0.31623 | HDAC | Misc | 0.9768 | 0.01830 |
BT-20 | Vorinostat | 1.0 | HDAC | Misc | 0.7991 | 0.05872 |
BT-20 | Vorinostat | 3.1623 | HDAC | Misc | 0.3234 | 0.21206 |
BT-20 | Vorinostat | 10.0 | HDAC | Misc | -0.1134 | 0.35615 |
BT-20 | Luminespib | 0.0001 | HSP90 | Misc | 1.0515 | 0.00266 |
BT-20 | Luminespib | 0.00031623 | HSP90 | Misc | 1.0678 | -0.00788 |
BT-20 | Luminespib | 0.001 | HSP90 | Misc | 1.0553 | 0.00563 |
BT-20 | Luminespib | 0.0031623 | HSP90 | Misc | 0.9463 | 0.00717 |