Breast Cancer Profiling Project, Drug Sensitivity phase I: Fixed-cell GR measures of 35 breast cell lines to 34 small molecule perturbagens from library plate I. Dataset 1 of 2: Normalized growth rate inhibition values - Dataset (ID:20343)
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Cell | Small Molecule | Small Mol Concentration (uM) | Primary Target | Pathway | Mean Normalized Growth Rate Inhibition Value | Increased Fraction Dead |
---|---|---|---|---|---|---|
BT-20 | Etoposide | 10.0 | Topo II | Chemotherapy | -0.3834 | 0.56500 |
BT-20 | Dasatinib | 0.001 | BCR/ABL | MAPK/nRTK | 0.9136 | 0.01008 |
BT-20 | Dasatinib | 0.0031623 | BCR/ABL | MAPK/nRTK | 0.9090 | 0.01661 |
BT-20 | Dasatinib | 0.01 | BCR/ABL | MAPK/nRTK | 0.9134 | 0.02789 |
BT-20 | Dasatinib | 0.031623 | BCR/ABL | MAPK/nRTK | 0.8598 | 0.04190 |
BT-20 | Dasatinib | 0.1 | BCR/ABL | MAPK/nRTK | 0.6781 | 0.07382 |
BT-20 | Dasatinib | 0.31623 | BCR/ABL | MAPK/nRTK | 0.5595 | 0.11968 |
BT-20 | Dasatinib | 1.0 | BCR/ABL | MAPK/nRTK | 0.4638 | 0.14107 |
BT-20 | Dasatinib | 3.1623 | BCR/ABL | MAPK/nRTK | 0.3868 | 0.16072 |
BT-20 | Dasatinib | 10.0 | BCR/ABL | MAPK/nRTK | 0.2835 | 0.16347 |
BT-20 | Trametinib | 0.0001 | MEK | MAPK/nRTK | 1.0624 | 0.00127 |
BT-20 | Trametinib | 0.00031623 | MEK | MAPK/nRTK | 1.0401 | 0.00439 |
BT-20 | Trametinib | 0.001 | MEK | MAPK/nRTK | 0.9545 | 0.01412 |
BT-20 | Trametinib | 0.0031623 | MEK | MAPK/nRTK | 0.8965 | 0.02484 |
BT-20 | Trametinib | 0.01 | MEK | MAPK/nRTK | 0.8643 | 0.03949 |
BT-20 | Trametinib | 0.031623 | MEK | MAPK/nRTK | 0.7406 | 0.06874 |
BT-20 | Trametinib | 0.1 | MEK | MAPK/nRTK | 0.6938 | 0.08108 |
BT-20 | Trametinib | 0.31623 | MEK | MAPK/nRTK | 0.6192 | 0.11389 |
BT-20 | Trametinib | 1.0 | MEK | MAPK/nRTK | 0.5034 | 0.13365 |
BT-20 | Saracatinib | 0.001 | SRC | MAPK/nRTK | 1.0364 | 0.01093 |
BT-20 | Saracatinib | 0.0031623 | SRC | MAPK/nRTK | 0.9942 | 0.00784 |
BT-20 | Saracatinib | 0.01 | SRC | MAPK/nRTK | 0.9466 | 0.01489 |
BT-20 | Saracatinib | 0.031623 | SRC | MAPK/nRTK | 0.9467 | 0.02156 |
BT-20 | Saracatinib | 0.1 | SRC | MAPK/nRTK | 0.8930 | 0.02961 |
BT-20 | Saracatinib | 0.31623 | SRC | MAPK/nRTK | 0.8970 | 0.03479 |