HG-6-64-01 KiNativ -- single dose experiment - Dataset (ID:20093)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| HG-6-64-01 | A-375 | KKCC1 | LAYNESEDRHYAMKVLSK | K1 | 10 | uM | |
| HG-6-64-01 | A-375 | CDC2 | VLHRDLKPQNLLIDDK | K2 | 10 | uM | |
| HG-6-64-01 | A-375 | CDK5, PRKX/Y | DLKPENILLDR | K2 | -12.1 | 10 | uM |
| HG-6-64-01 | A-375 | CDK8 | DGKDDKDYALKQIEGTGISMSACR | K1 | 10 | uM | |
| HG-6-64-01 | A-375 | CDK13 | DIKCSNILLNNRGQIK | K2 | 14.2 | 10 | uM |
| HG-6-64-01 | A-375 | CHK1 | LSKGDGLEFK | nonKD (autoinhibition domain) | 30.0 | 10 | uM |
| HG-6-64-01 | A-375 | CK1g1/2/3 | KIGCGNFGELR | ATP | 10 | uM | |
| HG-6-64-01 | A-375 | CK2a2 | LIDTVKDPVSK | KD | 10 | uM | |
| HG-6-64-01 | A-375 | CLK3 | YEIVGNLGEGTFGKVVECLDHAR | ATP | 10 | uM | |
| HG-6-64-01 | A-375 | COT | GAFGKVYLAQDIK | ATP | 10 | uM | |
| HG-6-64-01 | A-375 | CRK7 | DIKCSNILLNNSGQIK | K2 | 10 | uM | |
| HG-6-64-01 | A-375 | EPHB1 | LKLPGKREIYVAIK | K1 | 10 | uM | |
| HG-6-64-01 | A-375 | EPHB4 | FLEENSSDPTYTSSLGGKIPIR | ACT | -1.0 | 10 | uM |
| HG-6-64-01 | A-375 | Erk4 | DLKPANIFISTEDLVLK | K2 | -28.1 | 10 | uM |
| HG-6-64-01 | A-375 | FRAP1 | IQSIAPSLQVITSKQRPR | LIP | ~NI | 10 | uM |
| HG-6-64-01 | A-375 | FYN | VAIKTLKPGTMSPESFLEEAQIMK | K1 | 10 | uM | |
| HG-6-64-01 | A-375 | HGK (ZC1) | TGQLAAIKVMDVTEDEEEEIKLEINMLKK | K1 | 10 | uM | |
| HG-6-64-01 | A-375 | IGF1R | VAIKTVNEAASMR | K1 | 10 | uM | |
| HG-6-64-01 | A-375 | IKKB | WHNQETGEQIAIKQCR | K1 | 5.1 | 10 | uM |
| HG-6-64-01 | A-375 | INSR | VAVKTVNESASLR | K1 | 10 | uM | |
| HG-6-64-01 | A-375 | LATS2 | VDTHALYAMKTLR | K1 | 10 | uM | |
| HG-6-64-01 | A-375 | LYN | VAVKTLKPGTMSVQAFLEEANLMK | K1 | 96.8 | 10 | uM |
| HG-6-64-01 | A-375 | MAP3K5 | DIKGDNVLINTYSGVLK | K2 | -9.4 | 10 | uM |
| HG-6-64-01 | A-375 | MARK1 | HVLTGREVAVKIIDKTQLNPTSLQK | K1 | 10 | uM | |
| HG-6-64-01 | A-375 | MASTL | LYAVKVVK | K1 | -4.2 | 10 | uM |