HG-6-64-01 KiNativ -- single dose experiment - Dataset (ID:20093)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
HG-6-64-01 | A-375 | PKN2 | DLKLDNLLLDTEGFVK | K2 | -29.8 | 10 | uM |
HG-6-64-01 | A-375 | PKR | DLKPSNIFLVDTK | K2 | -1.4 | 10 | uM |
HG-6-64-01 | A-375 | PLK1 | CFEISDADTKEVFAGKIVPK | K1 | 3.4 | 10 | uM |
HG-6-64-01 | A-375 | PRPK | FLSGLELVKQGAEAR | ATP | 6.3 | 10 | uM |
HG-6-64-01 | A-375 | ROCK1,ROCK2 | DVKPDNMLLDK | K2 | 0.2 | 10 | uM |
HG-6-64-01 | A-375 | RSK1,RSK2,RSK3_domain1 | DLKPENILLDEEGHIK | K2 | 9.7 | 10 | uM |
HG-6-64-01 | A-375 | RSK1_domain1 | KVTRPDSGHLYAMKVLK | K1 | 10 | uM | |
HG-6-64-01 | A-375 | RSK1_domain2 | DLKPSNILYVDESGNPECLR | K2 | 2.9 | 10 | uM |
HG-6-64-01 | A-375 | RSK2_domain2 | DLKPSNILYVDESGNPESIR | K2 | 4.3 | 10 | uM |
HG-6-64-01 | A-375 | SGK3 | FYAVKVLQK | K1 | 6.8 | 10 | uM |
HG-6-64-01 | A-375 | SLK | DLKAGNILFTLDGDIK | -1.1 | 10 | uM | |
HG-6-64-01 | A-375 | SMG1 | DTVTIHSVGGTITILPTKTKPK | LIP | 12.2 | 10 | uM |
HG-6-64-01 | A-375 | TAO1,TAOK3 | DIKAGNILLTEPGQVK | K2 | ND | 10 | uM |
HG-6-64-01 | A-375 | TAOK2 | DVKAGNILLSEPGLVK | K2 | 21.1 | 10 | uM |
HG-6-64-01 | A-375 | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | K2 | 10 | uM | |
HG-6-64-01 | A-375 | ULK3 | NISHLDLKPQNILLSSLEKPHLK | K2 | -7.7 | 10 | uM |
HG-6-64-01 | A-375 | WEE1 | YIHSMSLVHMDIKPSNIFISR | K2 | 13.1 | 10 | uM |
HG-6-64-01 | A-375 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | K2 | -12.9 | 10 | uM |
HG-6-64-01 | A-375 | Wnk1,Wnk2,Wnk4 | IGDLGLATLKR | ACT | 0.6 | 10 | uM |
HG-6-64-01 | A-375 | MLTK | WISQDKEVAVKK | K1 | 89.2 | 10 | uM |
HG-6-64-01 | A-375 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIKGQNVLLTENAEVK | K2 | 60.3 | 10 | uM |
HG-6-64-01 | A-375 | AMPKa1 | VGKHELTGHKVAVKILNR | K1 | 10 | uM | |
HG-6-64-01 | A-375 | AMPKa2 | IGEHQLTGHKVAVKILNR | K1 | 10 | uM | |
HG-6-64-01 | A-375 | AXL | KIYNGDYYR | ACT | 10 | uM | |
HG-6-64-01 | A-375 | CAMK1D | LFAVKCIPK | K1 | -5.5 | 10 | uM |