HG-6-64-01 KiNativ -- single dose experiment - Dataset (ID:20093)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
HG-6-64-01 A-375 PKN2
DLKLDNLLLDTEGFVK
K2
-29.8
10
uM
HG-6-64-01 A-375 PKR
DLKPSNIFLVDTK
K2
-1.4
10
uM
HG-6-64-01 A-375 PLK1
CFEISDADTKEVFAGKIVPK
K1
3.4
10
uM
HG-6-64-01 A-375 PRPK
FLSGLELVKQGAEAR
ATP
6.3
10
uM
HG-6-64-01 A-375 ROCK1,ROCK2
DVKPDNMLLDK
K2
0.2
10
uM
HG-6-64-01 A-375 RSK1,RSK2,RSK3_domain1
DLKPENILLDEEGHIK
K2
9.7
10
uM
HG-6-64-01 A-375 RSK1_domain1
KVTRPDSGHLYAMKVLK
K1
10
uM
HG-6-64-01 A-375 RSK1_domain2
DLKPSNILYVDESGNPECLR
K2
2.9
10
uM
HG-6-64-01 A-375 RSK2_domain2
DLKPSNILYVDESGNPESIR
K2
4.3
10
uM
HG-6-64-01 A-375 SGK3
FYAVKVLQK
K1
6.8
10
uM
HG-6-64-01 A-375 SLK
DLKAGNILFTLDGDIK
-1.1
10
uM
HG-6-64-01 A-375 SMG1
DTVTIHSVGGTITILPTKTKPK
LIP
12.2
10
uM
HG-6-64-01 A-375 TAO1,TAOK3
DIKAGNILLTEPGQVK
K2
ND
10
uM
HG-6-64-01 A-375 TAOK2
DVKAGNILLSEPGLVK
K2
21.1
10
uM
HG-6-64-01 A-375 TLK1
YLNEIKPPIIHYDLKPGNILLVDGTACGEIK
K2
10
uM
HG-6-64-01 A-375 ULK3
NISHLDLKPQNILLSSLEKPHLK
K2
-7.7
10
uM
HG-6-64-01 A-375 WEE1
YIHSMSLVHMDIKPSNIFISR
K2
13.1
10
uM
HG-6-64-01 A-375 Wnk1,Wnk2,Wnk3
DLKCDNIFITGPTGSVK
K2
-12.9
10
uM
HG-6-64-01 A-375 Wnk1,Wnk2,Wnk4
IGDLGLATLKR
ACT
0.6
10
uM
HG-6-64-01 A-375 MLTK
WISQDKEVAVKK
K1
89.2
10
uM
HG-6-64-01 A-375 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIKGQNVLLTENAEVK
K2
60.3
10
uM
HG-6-64-01 A-375 AMPKa1
VGKHELTGHKVAVKILNR
K1
10
uM
HG-6-64-01 A-375 AMPKa2
IGEHQLTGHKVAVKILNR
K1
10
uM
HG-6-64-01 A-375 AXL
KIYNGDYYR
ACT
10
uM
HG-6-64-01 A-375 CAMK1D
LFAVKCIPK
K1
-5.5
10
uM