HG-6-64-01 KiNativ -- single dose experiment - Dataset (ID:20093)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
HG-6-64-01 | A-375 | MST4,YSK1 | DIKAANVLLSEQGDVK | K2 | -26.0 | 10 | uM |
HG-6-64-01 | A-375 | NDR1 | DTGHVYAMKILR | K1 | 3.3 | 10 | uM |
HG-6-64-01 | A-375 | NDR2 | DTGHIYAMKILR | K1 | 10 | uM | |
HG-6-64-01 | A-375 | NEK1 | DIKSQNIFLTK | K2 | -0.7 | 10 | uM |
HG-6-64-01 | A-375 | NEK6,NEK7 | DIKPANVFITATGVVK | K2 | 20.3 | 10 | uM |
HG-6-64-01 | A-375 | NEK7 | AACLLDGVPVALKK | K1 | -26.1 | 10 | uM |
HG-6-64-01 | A-375 | NEK8 | DLKTQNILLDK | K2 | 10 | uM | |
HG-6-64-01 | A-375 | NEK9 | DIKTLNIFLTK | K2 | -4.0 | 10 | uM |
HG-6-64-01 | A-375 | p38d,p38g | DLKPGNLAVNEDCELK | K2 | 10.2 | 10 | uM |
HG-6-64-01 | A-375 | KS6B1 | DLKPENIMLNHQGHVK | K2 | -1.0 | 10 | uM |
HG-6-64-01 | A-375 | KS6B2 | DLKPENIMLSSQGHIK | K2 | 4.2 | 10 | uM |
HG-6-64-01 | A-375 | CDK16 | LTDNLVALKEIR | K1 | 10 | uM | |
HG-6-64-01 | A-375 | PCTAIRE2,PCTAIRE3 | SKLTENLVALKEIR | K1 | 10 | uM | |
HG-6-64-01 | A-375 | PHKg2 | ATGHEFAVKIMEVTAER | K1 | 2.7 | 10 | uM |
HG-6-64-01 | A-375 | PI4KA,PI4KAP2 | SGTPMQSAAKAPYLAK | LIP | 13.7 | 10 | uM |
HG-6-64-01 | A-375 | PIK3C3 | TEDGGKYPVIFKHGDDLR | LIP (PI3K/PI4K) | 16.3 | 10 | uM |
HG-6-64-01 | A-375 | PIK3CB | VFGEDSVGVIFKNGDDLRQDMLTLQMLR | LIP (PI3K/PI4K) | 10 | uM | |
HG-6-64-01 | A-375 | PIP4K2A | AKELPTLKDNDFINEGQK | LIP (PI5K) | -2.6 | 10 | uM |
HG-6-64-01 | A-375 | PI42C | VKELPTLKDMDFLNK | LIP (PI5K) | -4.7 | 10 | uM |
HG-6-64-01 | A-375 | PI42C | TLVIKEVSSEDIADMHSNLSNYHQYIVK | LIP (PI5K) | 9.6 | 10 | uM |
HG-6-64-01 | A-375 | FYV1 | GGKSGAAFYATEDDRFILK | LIP (PI5K) | -22.6 | 10 | uM |
HG-6-64-01 | A-375 | PITSLRE | DLKTSNLLLSHAGILK | K2 | 3.2 | 10 | uM |
HG-6-64-01 | A-375 | PKCa,PKCb | DLKLDNVMLDSEGHIK | K2 | 1.5 | 10 | uM |
HG-6-64-01 | A-375 | KPCT | DLKLDNILLDK | K2 | -7.2 | 10 | uM |
HG-6-64-01 | A-375 | PKD1,PKD2 | NIVHCDLKPENVLLASADPFPQVK | K2 | 8.4 | 10 | uM |