HG-6-64-01 KiNativ -- single dose experiment - Dataset (ID:20093)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| HG-6-64-01 | A-375 | ABL,ARG | LMTGDTYTAHAGAKFPIK | ACT | 96.2 | 10 | uM |
| HG-6-64-01 | A-375 | ACK | TVSVAVKCLKPDVLSQPEAMDDFIR | K1 | 10 | uM | |
| HG-6-64-01 | A-375 | AGK | ATVFLNPAACKGK | LIP | ~NI | 10 | uM |
| HG-6-64-01 | A-375 | AKT1 | GTFGKVILVK | ATP | 3.8 | 10 | uM |
| HG-6-64-01 | A-375 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | K2 | 8.8 | 10 | uM |
| HG-6-64-01 | A-375 | ARAF | DLKSNNIFLHEGLTVK | K2 | 24.0 | 10 | uM |
| HG-6-64-01 | A-375 | ATM | QLVKGRDDLRQDAVMQQVFQMCNTLLQR | LIP | 10 | uM | |
| HG-6-64-01 | A-375 | ATR | FYIMMCKPK | LIP | 9.7 | 10 | uM |
| HG-6-64-01 | A-375 | AurA | DIKPENLLLGSAGELK | K2 | 5.1 | 10 | uM |
| HG-6-64-01 | A-375 | AurA,AurB,AurC | GKFGNVYLAR | ATP | 9.6 | 10 | uM |
| HG-6-64-01 | A-375 | BRAF | DLKSNNIFLHEDLTVK | K2 | 27.1 | 10 | uM |
| HG-6-64-01 | A-375 | KCC2D | IPTGQEYAAKIINTK | K1 | 33.7 | 10 | uM |
| HG-6-64-01 | A-375 | CaMK2g | TSTQEYAAKIINTK | K1 | 2.5 | 10 | uM |
| HG-6-64-01 | A-375 | CaMKK2 | LAYNENDNTYYAMKVLSK | K1 | 10 | uM | |
| HG-6-64-01 | A-375 | CASK | ETGQQFAVKIVDVAK | K1 | 10 | uM | |
| HG-6-64-01 | A-375 | CDK10 | DLKVSNLLMTDK | K2 | 6.5 | 10 | uM |
| HG-6-64-01 | A-375 | CDK11,CDK8 | DLKPANILVMGEGPER | K2 | -2.7 | 10 | uM |
| HG-6-64-01 | A-375 | CDK2 | NKLTGEVVALKK | K1 | -19.9 | 10 | uM |
| HG-6-64-01 | A-375 | CDK2 | DLKPQNLLINTEGAIK | K2 | -2.1 | 10 | uM |
| HG-6-64-01 | A-375 | CDK5 | NVLHRDLKPQNLLINR | K2 | -13.8 | 10 | uM |
| HG-6-64-01 | A-375 | CDK7 | DLKPNNLLLDENGVLK | K2 | 23.5 | 10 | uM |
| HG-6-64-01 | A-375 | CDK9 | DMKAANVLITR | K2 | -19.4 | 10 | uM |
| HG-6-64-01 | A-375 | CHK1 | DIKPENLLLDERDNLK | K2 | 6.3 | 10 | uM |
| HG-6-64-01 | A-375 | CHK2 | VAIKIISK | K1 | 10 | uM | |
| HG-6-64-01 | A-375 | KC1A | DIKPDNFLMGIGR | K2 | -2.0 | 10 | uM |