HG-6-64-01 KiNativ -- single dose experiment - Dataset (ID:20093)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
HG-6-64-01 A-375 NEK7
AACLLDGVPVALKK
K1
-26.1
10
uM
HG-6-64-01 A-375 PRP4
AAGIGKDFKENPNLR
10.8
10
uM
HG-6-64-01 A-375 IRAK1
AIQFLHQDSPSLIHGDIKSSNVLLDER
K2
49.4
10
uM
HG-6-64-01 A-375 PIP4K2B
AKDLPTFKDNDFLNEGQK
LIP (PI5K)
-37.8
10
uM
HG-6-64-01 A-375 PIP4K2A
AKELPTLKDNDFINEGQK
LIP (PI5K)
-2.6
10
uM
HG-6-64-01 A-375 LATS1
ALYATKTLR
K1
15.4
10
uM
HG-6-64-01 A-375 MLKL
APVAIKVFK
K1
-7.5
10
uM
HG-6-64-01 A-375 PHKg2
ATGHEFAVKIMEVTAER
K1
2.7
10
uM
HG-6-64-01 A-375 RSK1 (Domain 2)
ATNMEYAVKVIDK
K1
10
uM
HG-6-64-01 A-375 AGK
ATVFLNPAACKGK
LIP
~NI
10
uM
HG-6-64-01 A-375 PLK1 like (splice variant or novel kinase)
CFEISDADNKVVFAGKIVPK
K1
10
uM
HG-6-64-01 A-375 PLK1
CFEISDADTKEVFAGKIVPK
K1
3.4
10
uM
HG-6-64-01 A-375 FAK
CIGEGQFGDVHQGIYMSPENPALAVAIKTCK
K1
10
uM
HG-6-64-01 A-375 CDK8
DGKDDKDYALKQIEGTGISMSACR
K1
10
uM
HG-6-64-01 A-375 MST3
DIKAANVLLSEHGEVK
K2
-5.1
10
uM
HG-6-64-01 A-375 MST4,YSK1
DIKAANVLLSEQGDVK
K2
-26.0
10
uM
HG-6-64-01 A-375 MST1,MST2
DIKAGNILLNTEGHAK
K2
18.3
10
uM
HG-6-64-01 A-375 TAO1,TAOK3
DIKAGNILLTEPGQVK
K2
ND
10
uM
HG-6-64-01 A-375 CDK13
DIKCSNILLNNRGQIK
K2
14.2
10
uM
HG-6-64-01 A-375 CRK7
DIKCSNILLNNSGQIK
K2
10
uM
HG-6-64-01 A-375 MAP3K4
DIKGANIFLTSSGLIK
K2
-21.8
10
uM
HG-6-64-01 A-375 KHS1
DIKGANILLTDHGDVK
K2
35.0
10
uM
HG-6-64-01 A-375 M3K2,MAP3K3
DIKGANILR
K2
11.7
10
uM
HG-6-64-01 A-375 GCK
DIKGANLLLTLQGDVK
K2
10
uM
HG-6-64-01 A-375 MAP3K5
DIKGDNVLINTYSGVLK
K2
-9.4
10
uM
  • Page 1 of 8
  • 1 to 25 of 194 records