HG-6-64-01 KiNativ -- single dose experiment - Dataset (ID:20093)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| HG-6-64-01 | A-375 | TLK1/2 | YLNEIKPPIIHYDLKPGNILLVNGTACGEIK | K2 | 10 | uM | |
| HG-6-64-01 | A-375 | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | K2 | 10 | uM | |
| HG-6-64-01 | A-375 | eEF2K | YIKYNSNSGFVR | ATP | 26.2 | 10 | uM |
| HG-6-64-01 | A-375 | WEE1 | YIHSMSLVHMDIKPSNIFISR | K2 | 13.1 | 10 | uM |
| HG-6-64-01 | A-375 | CLK3 | YEIVGNLGEGTFGKVVECLDHAR | ATP | 10 | uM | |
| HG-6-64-01 | A-375 | JAK1_domain2 | YDPEGDNTGEQVAVKSLKPESGGNHIADLKK | K1 | 10 | uM | |
| HG-6-64-01 | A-375 | ILK | WQGNDIVVKVLK | K1 | 12.3 | 10 | uM |
| HG-6-64-01 | A-375 | MLTK | WISQDKEVAVKK | K1 | 89.2 | 10 | uM |
| HG-6-64-01 | A-375 | IKKB | WHNQETGEQIAIKQCR | K1 | 5.1 | 10 | uM |
| HG-6-64-01 | A-375 | CSK | VSDFGLTKEASSTQDTGKLPVK | ACT | 97.0 | 10 | uM |
| HG-6-64-01 | A-375 | PIK4CB | VPHTQAVVLNSKDKAPYLIYVEVLECENFDTTSVPARIPENR | nonKD | -58.2 | 10 | uM |
| HG-6-64-01 | A-375 | PAN3 | VMDPTKILITGK | KD | 10 | uM | |
| HG-6-64-01 | A-375 | TIF1b | VLVNDAQKVTEGQQER | ~NI | 10 | uM | |
| HG-6-64-01 | A-375 | CDC2 | VLHRDLKPQNLLIDDK | K2 | 10 | uM | |
| HG-6-64-01 | A-375 | MSK1,MSK2_domain1 | VLGTGAYGKVFLVR | ATP | 28.0 | 10 | uM |
| HG-6-64-01 | A-375 | PKCh | VLGKGSFGKVMLAR | ATP | 10 | uM | |
| HG-6-64-01 | A-375 | EPHA2 | VLEDDPEATYTTSGGKIPIR | ACT | 66.8 | 10 | uM |
| HG-6-64-01 | A-375 | PI42C | VKELPTLKDMDFLNK | LIP (PI5K) | -4.7 | 10 | uM |
| HG-6-64-01 | A-375 | PIK3C2B | VIFKCGDDLRQDMLTLQMIR | LIP (PI3K/PI4K) | 16.5 | 10 | uM |
| HG-6-64-01 | A-375 | AMPKa1 | VGKHELTGHKVAVKILNR | K1 | 10 | uM | |
| HG-6-64-01 | A-375 | PIK3CB | VFGEDSVGVIFKNGDDLRQDMLTLQMLR | LIP (PI3K/PI4K) | 10 | uM | |
| HG-6-64-01 | A-375 | LATS2 | VDTHALYAMKTLR | K1 | 10 | uM | |
| HG-6-64-01 | A-375 | INSR | VAVKTVNESASLR | K1 | 10 | uM | |
| HG-6-64-01 | A-375 | LYN | VAVKTLKPGTMSVQAFLEEANLMK | K1 | 96.8 | 10 | uM |
| HG-6-64-01 | A-375 | IGF1R | VAIKTVNEAASMR | K1 | 10 | uM |