HG-6-64-01 KiNativ -- single dose experiment - Dataset (ID:20093)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
HG-6-64-01 A-375 MET
DMYDKEYYSVHNK
ACT
-0.9
10
uM
HG-6-64-01 A-375 MRCKb
NHHVHLYPWSSLDGAEGSFDIKLPETK
K2
-6.0
10
uM
HG-6-64-01 A-375 MSK1 (Domain 1)
LYAMKVLK
K1
10
uM
HG-6-64-01 A-375 NEK3
SKNIFLTQNGK
ACT
10
uM
HG-6-64-01 A-375 NEK4
DLKTQNVFLTR
K2
0.2
10
uM
HG-6-64-01 A-375 p38a
DLKPSNLAVNEDCELK
K2
70.7
10
uM
HG-6-64-01 A-375 MK14
QELNKTIWEVPER
Other (MAPKAP2/3 active site in p38a complex)
97.3
10
uM
HG-6-64-01 A-375 PAN3
VMDPTKILITGK
KD
10
uM
HG-6-64-01 A-375 PCTAIRE2
DLKPQNLLINEKGELKLADFGLAR
K2
10
uM
HG-6-64-01 A-375 PDK1
ELATSREYAIKILEKR
K1
NI
10
uM
HG-6-64-01 A-375 PEK
DLKPSNIFFTMDDVVK
K2
-1.7
10
uM
HG-6-64-01 A-375 CDK15
PQNLLISHLGELKLADFGLARAKSIPSQTYSSEVVTLWYR
10
uM
HG-6-64-01 A-375 PIK3C2B
VIFKCGDDLRQDMLTLQMIR
LIP (PI3K/PI4K)
16.5
10
uM
HG-6-64-01 A-375 PIK4CB
VPHTQAVVLNSKDKAPYLIYVEVLECENFDTTSVPARIPENR
nonKD
-58.2
10
uM
HG-6-64-01 A-375 PIP4K2B
AKDLPTFKDNDFLNEGQK
LIP (PI5K)
-37.8
10
uM
HG-6-64-01 A-375 PKCd
GRGEYFAIKALKK
K1
10
uM
HG-6-64-01 A-375 PKCh
VLGKGSFGKVMLAR
ATP
10
uM
HG-6-64-01 A-375 PKCz
NDQIYAMKVVK
K1
10
uM
HG-6-64-01 A-375 PKD2
DVAVKVIDK(LR)?
K1
10
uM
HG-6-64-01 A-375 PKD3
DVAIKVIDK
K1
10
uM
HG-6-64-01 A-375 PKN1
GHFGKVLLSEFRPSGELFAIK
K1
19.0
10
uM
HG-6-64-01 A-375 PLK1
DLKLGNIFLDENLEVK
K2
-0.4
10
uM
HG-6-64-01 A-375 PLK1 like (splice variant or novel kinase)
CFEISDADNKVVFAGKIVPK
K1
10
uM
HG-6-64-01 A-375 PLK2
DLKLGNFFINEAMELK
K2
10
uM
HG-6-64-01 A-375 PRKX/Y
HFFALKVMSIPDVIR
K1
10
uM