HG-6-64-01 KiNativ -- single dose experiment - Dataset (ID:20093)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
HG-6-64-01 | A-375 | MET | DMYDKEYYSVHNK | ACT | -0.9 | 10 | uM |
HG-6-64-01 | A-375 | MRCKb | NHHVHLYPWSSLDGAEGSFDIKLPETK | K2 | -6.0 | 10 | uM |
HG-6-64-01 | A-375 | MSK1 (Domain 1) | LYAMKVLK | K1 | 10 | uM | |
HG-6-64-01 | A-375 | NEK3 | SKNIFLTQNGK | ACT | 10 | uM | |
HG-6-64-01 | A-375 | NEK4 | DLKTQNVFLTR | K2 | 0.2 | 10 | uM |
HG-6-64-01 | A-375 | p38a | DLKPSNLAVNEDCELK | K2 | 70.7 | 10 | uM |
HG-6-64-01 | A-375 | MK14 | QELNKTIWEVPER | Other (MAPKAP2/3 active site in p38a complex) | 97.3 | 10 | uM |
HG-6-64-01 | A-375 | PAN3 | VMDPTKILITGK | KD | 10 | uM | |
HG-6-64-01 | A-375 | PCTAIRE2 | DLKPQNLLINEKGELKLADFGLAR | K2 | 10 | uM | |
HG-6-64-01 | A-375 | PDK1 | ELATSREYAIKILEKR | K1 | NI | 10 | uM |
HG-6-64-01 | A-375 | PEK | DLKPSNIFFTMDDVVK | K2 | -1.7 | 10 | uM |
HG-6-64-01 | A-375 | CDK15 | PQNLLISHLGELKLADFGLARAKSIPSQTYSSEVVTLWYR | 10 | uM | ||
HG-6-64-01 | A-375 | PIK3C2B | VIFKCGDDLRQDMLTLQMIR | LIP (PI3K/PI4K) | 16.5 | 10 | uM |
HG-6-64-01 | A-375 | PIK4CB | VPHTQAVVLNSKDKAPYLIYVEVLECENFDTTSVPARIPENR | nonKD | -58.2 | 10 | uM |
HG-6-64-01 | A-375 | PIP4K2B | AKDLPTFKDNDFLNEGQK | LIP (PI5K) | -37.8 | 10 | uM |
HG-6-64-01 | A-375 | PKCd | GRGEYFAIKALKK | K1 | 10 | uM | |
HG-6-64-01 | A-375 | PKCh | VLGKGSFGKVMLAR | ATP | 10 | uM | |
HG-6-64-01 | A-375 | PKCz | NDQIYAMKVVK | K1 | 10 | uM | |
HG-6-64-01 | A-375 | PKD2 | DVAVKVIDK(LR)? | K1 | 10 | uM | |
HG-6-64-01 | A-375 | PKD3 | DVAIKVIDK | K1 | 10 | uM | |
HG-6-64-01 | A-375 | PKN1 | GHFGKVLLSEFRPSGELFAIK | K1 | 19.0 | 10 | uM |
HG-6-64-01 | A-375 | PLK1 | DLKLGNIFLDENLEVK | K2 | -0.4 | 10 | uM |
HG-6-64-01 | A-375 | PLK1 like (splice variant or novel kinase) | CFEISDADNKVVFAGKIVPK | K1 | 10 | uM | |
HG-6-64-01 | A-375 | PLK2 | DLKLGNFFINEAMELK | K2 | 10 | uM | |
HG-6-64-01 | A-375 | PRKX/Y | HFFALKVMSIPDVIR | K1 | 10 | uM |