QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| QL-XII-47 | BCWM.1 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | -4.884271122 | 1 | uM |
| QL-XII-47 | MWCL.1 | ABL,ARG | YSLTVAVKTLKEDTMEVEEFLK | Lys1 | 19.0495645 | 1 | uM |
| QL-XII-47 | MWCL.1 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | -4.6555368 | 1 | uM |
| QL-XII-47 | BCWM.1 | ABL,ARG | YSLTVAVKTLKEDTMEVEEFLK | Lys1 | 23.94636209 | 1 | uM |
| QL-XII-47 | BCWM.1 | ACK | TVSVAVKCLKPDVLSQPEAMDDFIR | Lys1 | 16.75144083 | 1 | uM |
| QL-XII-47 | MWCL.1 | ACK | TVSVAVKCLKPDVLSQPEAMDDFIR | Lys1 | 10.48021172 | 1 | uM |
| QL-XII-47 | MWCL.1 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | 7.862213435 | 1 | uM |
| QL-XII-47 | BCWM.1 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | 18.43323382 | 1 | uM |
| QL-XII-47 | MWCL.1 | ARAF | DLKSNNIFLHEGLTVK | Lys2 | -8.125226322 | 1 | uM |
| QL-XII-47 | BCWM.1 | ARAF | DLKSNNIFLHEGLTVK | Lys2 | 4.534711447 | 1 | uM |
| QL-XII-47 | MWCL.1 | ATR | FYIMMCKPK | ATP | 26.45300257 | 1 | uM |
| QL-XII-47 | BCWM.1 | ATR | FYIMMCKPK | ATP | 0.044349501 | 1 | uM |
| QL-XII-47 | MWCL.1 | AurA | FILALKVLFK | Lys1 | 11.33219394 | 1 | uM |
| QL-XII-47 | BCWM.1 | AurA | FILALKVLFK | Lys1 | 19.31283508 | 1 | uM |
| QL-XII-47 | MWCL.1 | AurB | SHFIVALKVLFK | Lys1 | -12.60176386 | 1 | uM |
| QL-XII-47 | BCWM.1 | AurB | SHFIVALKVLFK | Lys1 | 7.861261294 | 1 | uM |
| QL-XII-47 | BCWM.1 | BARK1 | DLKPANILLDEHGHVR | Lys2 | -22.46332421 | 1 | uM |
| QL-XII-47 | MWCL.1 | BARK1 | DLKPANILLDEHGHVR | Lys2 | -11.39063633 | 1 | uM |
| QL-XII-47 | BCWM.1 | BLK | IIDSEYTAQEGAKFPIK | Activation Loop | 47.0732956 | 1 | uM |
| QL-XII-47 | MWCL.1 | BLK | IIDSEYTAQEGAKFPIK | Activation Loop | ND | 1 | uM |
| QL-XII-47 | BCWM.1 | BRAF | DLKSNNIFLHEDLTVK | Lys2 | 17.78977881 | 1 | uM |
| QL-XII-47 | MWCL.1 | BRAF | DLKSNNIFLHEDLTVK | Lys2 | 22.55132673 | 1 | uM |
| QL-XII-47 | MWCL.1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | 73.49216218 | 1 | uM |
| QL-XII-47 | BCWM.1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | 70.55327861 | 1 | uM |
| QL-XII-47 | BCWM.1 | CAMK1D | LFAVKCIPK | Lys1 | 0.033712822 | 1 | uM |