QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| QL-XII-47 | MWCL.1 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | -4.6555368 | 1 | uM |
| QL-XII-47 | MWCL.1 | ABL,ARG | YSLTVAVKTLKEDTMEVEEFLK | Lys1 | 19.0495645 | 1 | uM |
| QL-XII-47 | MWCL.1 | ACK | TVSVAVKCLKPDVLSQPEAMDDFIR | Lys1 | 10.48021172 | 1 | uM |
| QL-XII-47 | MWCL.1 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | 7.862213435 | 1 | uM |
| QL-XII-47 | MWCL.1 | ARAF | DLKSNNIFLHEGLTVK | Lys2 | -8.125226322 | 1 | uM |
| QL-XII-47 | MWCL.1 | ATR | FYIMMCKPK | ATP | 26.45300257 | 1 | uM |
| QL-XII-47 | MWCL.1 | AurA | FILALKVLFK | Lys1 | 11.33219394 | 1 | uM |
| QL-XII-47 | MWCL.1 | AurB | SHFIVALKVLFK | Lys1 | -12.60176386 | 1 | uM |
| QL-XII-47 | MWCL.1 | BARK1 | DLKPANILLDEHGHVR | Lys2 | -11.39063633 | 1 | uM |
| QL-XII-47 | MWCL.1 | BRAF | DLKSNNIFLHEDLTVK | Lys2 | 22.55132673 | 1 | uM |
| QL-XII-47 | MWCL.1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | 73.49216218 | 1 | uM |
| QL-XII-47 | MWCL.1 | CAMK1D | LFAVKCIPK | Lys1 | -13.81029327 | 1 | uM |
| QL-XII-47 | MWCL.1 | CaMK2g | TSTQEYAAKIINTK | Lys1 | -11.28758926 | 1 | uM |
| QL-XII-47 | MWCL.1 | CaMKK2 | DIKPSNLLVGEDGHIK | Lys2 | 11.9973621 | 1 | uM |
| QL-XII-47 | MWCL.1 | CASK | ETGQQFAVKIVDVAK | Lys1 | 20.5361767 | 1 | uM |
| QL-XII-47 | MWCL.1 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | -11.26471968 | 1 | uM |
| QL-XII-47 | MWCL.1 | CDK11,CDK8 | DLKPANILVMGEGPER | Lys2 | 4.501665604 | 1 | uM |
| QL-XII-47 | MWCL.1 | CDK2 | DLKPQNLLINTEGAIK | Lys2 | -3.151747592 | 1 | uM |
| QL-XII-47 | MWCL.1 | CDK4 | DLKPENILVTSGGTVK | Lys2 | -6.2228303 | 1 | uM |
| QL-XII-47 | MWCL.1 | CDK5 | DLKPQNLLINR | Lys2 | -8.984027957 | 1 | uM |
| QL-XII-47 | MWCL.1 | CDK6 | DLKPQNILVTSSGQIK | Lys2 | 3.69039298 | 1 | uM |
| QL-XII-47 | MWCL.1 | CDK7 | DLKPNNLLLDENGVLK | Lys2 | 17.57459374 | 1 | uM |
| QL-XII-47 | MWCL.1 | CDK9 | DMKAANVLITR | Lys2 | -0.188182157 | 1 | uM |
| QL-XII-47 | MWCL.1 | CHK1 | DIKPENLLLDER | Lys2 | -6.099115594 | 1 | uM |
| QL-XII-47 | MWCL.1 | CHK2 | DLKPENVLLSSQEEDCLIK | Lys2 | 18.70101594 | 1 | uM |