QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
QL-XII-47 | BCWM.1 | CAMK1D | LFAVKCIPK | Lys1 | 0.033712822 | 1 | uM |
QL-XII-47 | MWCL.1 | NEK1 | DIKSQNIFLTK | Lys2 | 0.042103767 | 1 | uM |
QL-XII-47 | BCWM.1 | ATR | FYIMMCKPK | ATP | 0.044349501 | 1 | uM |
QL-XII-47 | MWCL.1 | TBK1 | TGDLFAIKVFNNISFLRPVDVQMR | Lys1 | 0.073270679 | 1 | uM |
QL-XII-47 | BCWM.1 | MASTL | GAFGKVYLGQK | ATP Loop | -0.133762637 | 1 | uM |
QL-XII-47 | BCWM.1 | NEK2 | DLKPANVFLDGK | Lys2 | 0.142322043 | 1 | uM |
QL-XII-47 | MWCL.1 | CDK9 | DMKAANVLITR | Lys2 | -0.188182157 | 1 | uM |
QL-XII-47 | MWCL.1 | KC1G2 | DVKPENFLVGRPGTK | Lys2 | 0.240956147 | 1 | uM |
QL-XII-47 | BCWM.1 | IKKE | SGELVAVKVFNTTSYLRPR | Lys1 | 0.341218516 | 1 | uM |
QL-XII-47 | BCWM.1 | SRPK1 | IIHTDIKPENILLSVNEQYIR | Lys2 | 0.388055572 | 1 | uM |
QL-XII-47 | BCWM.1 | MK01 | DLKPSNLLLNTTCDLK | Lys2 | 0.422779704 | 1 | uM |
QL-XII-47 | MWCL.1 | M3K2 | ELAVKQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | -0.459368027 | 1 | uM |
QL-XII-47 | MWCL.1 | MST4,YSK1 | DIKAANVLLSEQGDVK | Lys2 | -0.541351906 | 1 | uM |
QL-XII-47 | BCWM.1 | CDK6 | DLKPQNILVTSSGQIK | Lys2 | -0.544166997 | 1 | uM |
QL-XII-47 | MWCL.1 | FER | TSVAVKTCKEDLPQELK | Lys1 | 0.548717854 | 1 | uM |
QL-XII-47 | BCWM.1 | TYK2(Kin.Dom.2) | IGDFGLAKAVPEGHEYYR | Activation Loop | 0.574708889 | 1 | uM |
QL-XII-47 | BCWM.1 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | 0.583601186 | 1 | uM |
QL-XII-47 | MWCL.1 | Wnk1,Wnk2 | GSFKTVYK | ATP Loop | -0.603873492 | 1 | uM |
QL-XII-47 | MWCL.1 | NDR1 | DIKPDNLLLDSK | Lys2 | 0.686324454 | 1 | uM |
QL-XII-47 | BCWM.1 | MAP2K4 | DIKPSNILLDR | Lys2 | -0.827779834 | 1 | uM |
QL-XII-47 | BCWM.1 | KCC2D | IPTGQEYAAKIINTKK | Lys1 | 0.853020424 | 1 | uM |
QL-XII-47 | MWCL.1 | IKKB | DLKPENIVLQQGEQR | Lys2 | 0.88441842 | 1 | uM |
QL-XII-47 | BCWM.1 | WEE1 | YIHSMSLVHMDIKPSNIFISR | Lys2 | 0.899795474 | 1 | uM |
QL-XII-47 | MWCL.1 | IKKE | SGELVAVKVFNTTSYLRPR | Lys1 | 0.982360401 | 1 | uM |
QL-XII-47 | BCWM.1 | ULK1 | DLKPQNILLSNPAGR | Lys2 | 10.00533539 | 1 | uM |