QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
QL-XII-47 BCWM.1 CAMK1D
LFAVKCIPK
Lys1
0.033712822
1
uM
QL-XII-47 MWCL.1 NEK1
DIKSQNIFLTK
Lys2
0.042103767
1
uM
QL-XII-47 BCWM.1 ATR
FYIMMCKPK
ATP
0.044349501
1
uM
QL-XII-47 MWCL.1 TBK1
TGDLFAIKVFNNISFLRPVDVQMR
Lys1
0.073270679
1
uM
QL-XII-47 BCWM.1 MASTL
GAFGKVYLGQK
ATP Loop
-0.133762637
1
uM
QL-XII-47 BCWM.1 NEK2
DLKPANVFLDGK
Lys2
0.142322043
1
uM
QL-XII-47 MWCL.1 CDK9
DMKAANVLITR
Lys2
-0.188182157
1
uM
QL-XII-47 MWCL.1 KC1G2
DVKPENFLVGRPGTK
Lys2
0.240956147
1
uM
QL-XII-47 BCWM.1 IKKE
SGELVAVKVFNTTSYLRPR
Lys1
0.341218516
1
uM
QL-XII-47 BCWM.1 SRPK1
IIHTDIKPENILLSVNEQYIR
Lys2
0.388055572
1
uM
QL-XII-47 BCWM.1 MK01
DLKPSNLLLNTTCDLK
Lys2
0.422779704
1
uM
QL-XII-47 MWCL.1 M3K2
ELAVKQVQFDPDSPETSKEVNALECEIQLLK
Lys1
-0.459368027
1
uM
QL-XII-47 MWCL.1 MST4,YSK1
DIKAANVLLSEQGDVK
Lys2
-0.541351906
1
uM
QL-XII-47 BCWM.1 CDK6
DLKPQNILVTSSGQIK
Lys2
-0.544166997
1
uM
QL-XII-47 MWCL.1 FER
TSVAVKTCKEDLPQELK
Lys1
0.548717854
1
uM
QL-XII-47 BCWM.1 TYK2(Kin.Dom.2)
IGDFGLAKAVPEGHEYYR
Activation Loop
0.574708889
1
uM
QL-XII-47 BCWM.1 CSK
VSDFGLTKEASSTQDTGKLPVK
Activation Loop
0.583601186
1
uM
QL-XII-47 MWCL.1 Wnk1,Wnk2
GSFKTVYK
ATP Loop
-0.603873492
1
uM
QL-XII-47 MWCL.1 NDR1
DIKPDNLLLDSK
Lys2
0.686324454
1
uM
QL-XII-47 BCWM.1 MAP2K4
DIKPSNILLDR
Lys2
-0.827779834
1
uM
QL-XII-47 BCWM.1 KCC2D
IPTGQEYAAKIINTKK
Lys1
0.853020424
1
uM
QL-XII-47 MWCL.1 IKKB
DLKPENIVLQQGEQR
Lys2
0.88441842
1
uM
QL-XII-47 BCWM.1 WEE1
YIHSMSLVHMDIKPSNIFISR
Lys2
0.899795474
1
uM
QL-XII-47 MWCL.1 IKKE
SGELVAVKVFNTTSYLRPR
Lys1
0.982360401
1
uM
QL-XII-47 BCWM.1 ULK1
DLKPQNILLSNPAGR
Lys2
10.00533539
1
uM
  • Page 1 of 16
  • 1 to 25 of 378 records