QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| QL-XII-47 | BCWM.1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | 70.55327861 | 1 | uM |
| QL-XII-47 | BCWM.1 | KSR1,KSR2 | SKNVFYDNGK | Activation Loop | -18.43797163 | 1 | uM |
| QL-XII-47 | MWCL.1 | SYK | ISDFGLSKALR | Activation Loop | 9.937407948 | 1 | uM |
| QL-XII-47 | BCWM.1 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | -4.884271122 | 1 | uM |
| QL-XII-47 | BCWM.1 | FGR | LIKDDEYNPCQGSKFPIK | Activation Loop | -59.65168038 | 1 | uM |
| QL-XII-47 | BCWM.1 | JAK3 domain2 | IADFGLAKLLPLDKDYYVVR | Activation Loop | -55.6912494 | 1 | uM |
| QL-XII-47 | MWCL.1 | FYN,SRC,YES | QGAKFPIKWTAPEAALYGR | Activation Loop | -8.174014716 | 1 | uM |
| QL-XII-47 | MWCL.1 | STLK5 | YSVKVLPWLSPEVLQQNLQGYDAK | Activation Loop | -1.488167509 | 1 | uM |
| QL-XII-47 | MWCL.1 | TEC | YVLDDQYTSSSGAKFPVK | Activation Loop | 60.11680682 | 1 | uM |
| QL-XII-47 | MWCL.1 | JAK1_domain2 | IGDFGLTKAIETDKEYYTVK | Activation Loop | -9.341503001 | 1 | uM |
| QL-XII-47 | BCWM.1 | EPHB2 | FLEDDTSDPTYTSALGGKIPIR | Activation Loop | -24.56149352 | 1 | uM |
| QL-XII-47 | MWCL.1 | NEK3 | SKNIFLTQNGK | Activation Loop | 9.919741065 | 1 | uM |
| QL-XII-47 | BCWM.1 | FYN,SRC,YES | QGAKFPIKWTAPEAALYGR | Activation Loop | 2.746888981 | 1 | uM |
| QL-XII-47 | BCWM.1 | JAK1_domain2 | IGDFGLTKAIETDKEYYTVK | Activation Loop | -18.81736377 | 1 | uM |
| QL-XII-47 | MWCL.1 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | -4.6555368 | 1 | uM |
| QL-XII-47 | MWCL.1 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | -1.027450805 | 1 | uM |
| QL-XII-47 | MWCL.1 | KSR1,KSR2 | SKNVFYDNGK | Activation Loop | -17.85533882 | 1 | uM |
| QL-XII-47 | MWCL.1 | FAK2 | YIEDEDYYKASVTR | Activation Loop | -31.93905936 | 1 | uM |
| QL-XII-47 | MWCL.1 | JAK3 domain2 | IADFGLAKLLPLDKDYYVVR | Activation Loop | -87.4730226 | 1 | uM |
| QL-XII-47 | MWCL.1 | EPHB2 | FLEDDTSDPTYTSALGGKIPIR | Activation Loop | ND | 1 | uM |
| QL-XII-47 | MWCL.1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | 73.49216218 | 1 | uM |
| QL-XII-47 | MWCL.1 | FGR | LIKDDEYNPCQGSKFPIK | Activation Loop | -18.8674785 | 1 | uM |
| QL-XII-47 | BCWM.1 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | 0.583601186 | 1 | uM |
| QL-XII-47 | BCWM.1 | FAK2 | YIEDEDYYKASVTR | Activation Loop | -37.08301629 | 1 | uM |
| QL-XII-47 | BCWM.1 | NEK3 | SKNIFLTQNGK | Activation Loop | -10.13654488 | 1 | uM |