QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| QL-XII-47 | MWCL.1 | ZC2/TNIK | TGQLAAIKVMDVTGDEEEEIKQEINMLKK | Lys1 | -2.724092946 | 1 | uM |
| QL-XII-47 | BCWM.1 | ZC2/TNIK | TGQLAAIKVMDVTGDEEEEIKQEINMLKK | Lys1 | 4.081055995 | 1 | uM |
| QL-XII-47 | MWCL.1 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIKGQNVLLTENAEVK | Lys2 | -26.32668943 | 1 | uM |
| QL-XII-47 | BCWM.1 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIKGQNVLLTENAEVK | Lys2 | -19.55134985 | 1 | uM |
| QL-XII-47 | BCWM.1 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | Lys2 | -6.796460792 | 1 | uM |
| QL-XII-47 | MWCL.1 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | Lys2 | -10.55702775 | 1 | uM |
| QL-XII-47 | BCWM.1 | Wnk1,Wnk2 | GSFKTVYK | ATP Loop | -23.10912536 | 1 | uM |
| QL-XII-47 | MWCL.1 | Wnk1,Wnk2 | GSFKTVYK | ATP Loop | -0.603873492 | 1 | uM |
| QL-XII-47 | BCWM.1 | WEE1 | YIHSMSLVHMDIKPSNIFISR | Lys2 | 0.899795474 | 1 | uM |
| QL-XII-47 | MWCL.1 | WEE1 | YIHSMSLVHMDIKPSNIFISR | Lys2 | -37.77693454 | 1 | uM |
| QL-XII-47 | BCWM.1 | VRK2 | MLDVLEYIHENEYVHGDIKAANLLLGYK | Lys2 | -1.787209636 | 1 | uM |
| QL-XII-47 | MWCL.1 | VRK2 | MLDVLEYIHENEYVHGDIKAANLLLGYK | Lys2 | 22.7412435 | 1 | uM |
| QL-XII-47 | BCWM.1 | ULK3 | NISHLDLKPQNILLSSLEKPHLK | Lys2 | 10.43573458 | 1 | uM |
| QL-XII-47 | MWCL.1 | ULK3 | NISHLDLKPQNILLSSLEKPHLK | Lys2 | 2.928063615 | 1 | uM |
| QL-XII-47 | BCWM.1 | ULK1 | DLKPQNILLSNPAGR | Lys2 | 10.00533539 | 1 | uM |
| QL-XII-47 | MWCL.1 | ULK1 | DLKPQNILLSNPAGR | Lys2 | -14.58312377 | 1 | uM |
| QL-XII-47 | BCWM.1 | TYK2(Kin.Dom.2) | IGDFGLAKAVPEGHEYYR | Activation Loop | 0.574708889 | 1 | uM |
| QL-XII-47 | MWCL.1 | TYK2(Kin.Dom.2) | IGDFGLAKAVPEGHEYYR | Activation Loop | -4.184361 | 1 | uM |
| QL-XII-47 | MWCL.1 | TLK1/2 | YLNEIKPPIIHYDLKPGNILLVNGTACGEIK | Lys2 | -2.951577221 | 1 | uM |
| QL-XII-47 | BCWM.1 | TLK1/2 | YLNEIKPPIIHYDLKPGNILLVNGTACGEIK | Lys2 | -3.9573695 | 1 | uM |
| QL-XII-47 | BCWM.1 | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | Lys2 | 11.52268187 | 1 | uM |
| QL-XII-47 | MWCL.1 | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | Lys2 | -1.435121129 | 1 | uM |
| QL-XII-47 | BCWM.1 | TEC | YVLDDQYTSSSGAKFPVK | Activation Loop | 70.24556535 | 1 | uM |
| QL-XII-47 | MWCL.1 | TEC | YVLDDQYTSSSGAKFPVK | Activation Loop | 60.11680682 | 1 | uM |
| QL-XII-47 | MWCL.1 | TBK1 | TGDLFAIKVFNNISFLRPVDVQMR | Lys1 | 0.073270679 | 1 | uM |