XMD11-85h KiNativ -- single dose experiment - Dataset (ID:20098)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD11-85h | PC-3 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLkPENLLLASK | Lys2 | -0.1 | 10 | uM |
| XMD11-85h | PC-3 | PRP4 | CNILHADIkPDNILVNESK | Lys2 | 0.1 | 10 | uM |
| XMD11-85h | PC-3 | M3K2 | ELAVkQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | 0.1 | 10 | uM |
| XMD11-85h | HeLa | PKR | DLkPSNIFLVDTK | Lys2 | -0.2 | 10 | uM |
| XMD11-85h | PC-3 | EPHB4 | FLEENSSDPTYTSSLGGkIPIR | Activation Loop | 0.4 | 10 | uM |
| XMD11-85h | PC-3 | MST1 | ETGQIVAIkQVPVESDLQEIIK | Lys1 | 0.4 | 10 | uM |
| XMD11-85h | PC-3 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | -0.5 | 10 | uM |
| XMD11-85h | PC-3 | MK14 | QELNkTIWEVPER | Other | 0.5 | 10 | uM |
| XMD11-85h | PC-3 | M3K2,MAP3K3 | DIkGANILR | Lys2 | -0.6 | 10 | uM |
| XMD11-85h | PC-3 | CDK5 | DLkPQNLLINR | Lys2 | 0.6 | 10 | uM |
| XMD11-85h | PC-3 | CHK2 | VAIkIISK | Lys1 | 0.6 | 10 | uM |
| XMD11-85h | PC-3 | SLK | ETSVLAAAkVIDTK | Lys1 | -0.8 | 10 | uM |
| XMD11-85h | PC-3 | PKR | DLkPSNIFLVDTK | Lys2 | 0.8 | 10 | uM |
| XMD11-85h | PC-3 | CLK2 | LTHTDLkPENILFVNSDYELTYNLEK | Lys2 | -1.0 | 10 | uM |
| XMD11-85h | HeLa | JNK1,JNK2,JNK3 | DLkPSNIVVK | Lys2 | -10.1 | 10 | uM |
| XMD11-85h | HeLa | RSK2_domain1 | LTDFGLSkESIDHEKK | Activation Loop | -10.3 | 10 | uM |
| XMD11-85h | HeLa | KPCI | IYAMkVVK | Lys1 | -10.5 | 10 | uM |
| XMD11-85h | PC-3 | RON | IQCAIkSLSR | Lys1 | 10.5 | 10 | uM |
| XMD11-85h | HeLa | CaMK1a | LVAIkCIAK | Lys1 | -10.7 | 10 | uM |
| XMD11-85h | HeLa | PAN3 | VMDPTkILITGK | -10.7 | 10 | uM | |
| XMD11-85h | PC-3 | SLK | DLkAGNILFTLDGDIK | Lys2 | -10.7 | 10 | uM |
| XMD11-85h | PC-3 | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | 10.7 | 10 | uM |
| XMD11-85h | PC-3 | ROCK1,ROCK2 | DVkPDNMLLDK | Lys2 | 10.7 | 10 | uM |
| XMD11-85h | HeLa | JAK2 domain2 | IGDFGLTkVLPQDKEYYK | Activation Loop | -1.1 | 10 | uM |
| XMD11-85h | HeLa | CHK1 | DIkPENLLLDER | Lys2 | -11.0 | 10 | uM |