XMD11-85h KiNativ -- single dose experiment - Dataset (ID:20098)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD11-85h | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | -38.1 | 10 | uM |
| XMD11-85h | HeLa | ACK | TVSVAVkCLKPDVLSQPEAMDDFIR | Lys1 | -2.4 | 10 | uM |
| XMD11-85h | PC-3 | AGK | ATVFLNPAACkGK | ATP | -1.4 | 10 | uM |
| XMD11-85h | HeLa | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | -34.6 | 10 | uM |
| XMD11-85h | PC-3 | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 16.2 | 10 | uM |
| XMD11-85h | HeLa | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | -16.3 | 10 | uM |
| XMD11-85h | PC-3 | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | -2.4 | 10 | uM |
| XMD11-85h | PC-3 | ANPb | GMAFLHNSIISSHGSLkSSNCVVDSR | Lys2 | 11.0 | 10 | uM |
| XMD11-85h | HeLa | ARAF | DLkSNNIFLHEGLTVK | Lys2 | 4.5 | 10 | uM |
| XMD11-85h | PC-3 | ATR | FYIMMCkPK | ATP | 21.6 | 10 | uM |
| XMD11-85h | HeLa | ATR | FYIMMCkPK | ATP | -8.9 | 10 | uM |
| XMD11-85h | HeLa | AurB | SHFIVALkVLFK | Lys1 | 41.7 | 10 | uM |
| XMD11-85h | HeLa | BARK1 | DLkPANILLDEHGHVR | Lys2 | -33.3 | 10 | uM |
| XMD11-85h | HeLa | BRAF | DLkSNNIFLHEDLTVK | Lys2 | 15.0 | 10 | uM |
| XMD11-85h | HeLa | BTK | GQYDVAIkMIK | Lys1 | -35.0 | 10 | uM |
| XMD11-85h | HeLa | CaMK1a | LVAIkCIAK | Lys1 | -10.7 | 10 | uM |
| XMD11-85h | HeLa | CAMK1D | LFAVkCIPK | Lys1 | -8.9 | 10 | uM |
| XMD11-85h | PC-3 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLkPENLLLASK | Lys2 | -0.1 | 10 | uM |
| XMD11-85h | PC-3 | CaMK2g | TSTQEYAAkIINTK | Lys1 | -2.6 | 10 | uM |
| XMD11-85h | HeLa | CaMK2g | TSTQEYAAkIINTK | Lys1 | -16.1 | 10 | uM |
| XMD11-85h | PC-3 | CASK | ETGQQFAVkIVDVAK | Lys1 | -9.9 | 10 | uM |
| XMD11-85h | PC-3 | CDK10 | DLkVSNLLMTDK | Lys2 | 14.6 | 10 | uM |
| XMD11-85h | PC-3 | CDK11,CDK8 | DLkPANILVMGEGPER | Lys2 | 16.3 | 10 | uM |
| XMD11-85h | PC-3 | CDK14 | LVALkVIR | Lys1 | -22.4 | 10 | uM |
| XMD11-85h | PC-3 | CDK16 | LTDNLVALkEIR | Lys1 | -12.2 | 10 | uM |