XMD11-85h KiNativ -- single dose experiment - Dataset (ID:20098)

Filter results: >>>>
  • Page 1 of 10
  • 1 to 25 of 241 records
Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD11-85h PC-3 EphA1
LLDDFDGTYETQGGkIPIR
Activation Loop
-1.4
10
uM
XMD11-85h HeLa SYK
ISDFGLSkALR
Activation Loop
-11.5
10
uM
XMD11-85h PC-3 MET
DMYDkEYYSVHNK
Activation Loop
27.6
10
uM
XMD11-85h PC-3 EGFR
ITDFGLAkLLGAEEK
Activation Loop
11.4
10
uM
XMD11-85h HeLa JAK2 domain2
IGDFGLTkVLPQDKEYYK
Activation Loop
-1.1
10
uM
XMD11-85h HeLa RSK1 domain1
LTDFGLSkEAIDHEK
Activation Loop
-23.5
10
uM
XMD11-85h PC-3 CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
4.0
10
uM
XMD11-85h PC-3 EPHB4
FLEENSSDPTYTSSLGGkIPIR
Activation Loop
0.4
10
uM
XMD11-85h PC-3 EGFR
LLGAEEKEYHAEGGkVPIK
Activation Loop
4.3
10
uM
XMD11-85h PC-3 NEK9
LGDYGLAkK
Activation Loop
7.8
10
uM
XMD11-85h PC-3 EphA7
VIEDDPEAVYTTTGGkIPVR
Activation Loop
4.1
10
uM
XMD11-85h PC-3 EPHB2
FLEDDTSDPTYTSALGGkIPIR
Activation Loop
-37.3
10
uM
XMD11-85h HeLa JAK3 domain2
IADFGLAkLLPLDKDYYVVR
Activation Loop
-13.7
10
uM
XMD11-85h PC-3 MET
DMYDKEYYSVHNkTGAK
Activation Loop
38.6
10
uM
XMD11-85h HeLa ABL,ARG
LMTGDTYTAHAGAkFPIK
Activation Loop
-38.1
10
uM
XMD11-85h HeLa CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-8.0
10
uM
XMD11-85h HeLa STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
-30.0
10
uM
XMD11-85h PC-3 Wnk1,Wnk2,Wnk4
IGDLGLATLkR
Activation Loop
-5.1
10
uM
XMD11-85h HeLa JAK1_domain2
IGDFGLTkAIETDKEYYTVK
Activation Loop
-6.3
10
uM
XMD11-85h PC-3 FYN,SRC,YES
QGAkFPIKWTAPEAALYGR
Activation Loop
6.7
10
uM
XMD11-85h PC-3 EPHA2
VLEDDPEATYTTSGGkIPIR
Activation Loop
-0.5
10
uM
XMD11-85h HeLa NEK9
LGDYGLAkK
Activation Loop
-20.3
10
uM
XMD11-85h HeLa RSK2_domain1
LTDFGLSkESIDHEKK
Activation Loop
-10.3
10
uM
XMD11-85h HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
-11.8
10
uM
XMD11-85h HeLa PIK3C3
TEDGGKYPVIFkHGDDLR
ATP
-5.7
10
uM
  • Page 1 of 10
  • 1 to 25 of 241 records