XMD11-85h KiNativ -- single dose experiment - Dataset (ID:20098)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD11-85h | PC-3 | EphA1 | LLDDFDGTYETQGGkIPIR | Activation Loop | -1.4 | 10 | uM |
XMD11-85h | HeLa | SYK | ISDFGLSkALR | Activation Loop | -11.5 | 10 | uM |
XMD11-85h | PC-3 | MET | DMYDkEYYSVHNK | Activation Loop | 27.6 | 10 | uM |
XMD11-85h | PC-3 | EGFR | ITDFGLAkLLGAEEK | Activation Loop | 11.4 | 10 | uM |
XMD11-85h | HeLa | JAK2 domain2 | IGDFGLTkVLPQDKEYYK | Activation Loop | -1.1 | 10 | uM |
XMD11-85h | HeLa | RSK1 domain1 | LTDFGLSkEAIDHEK | Activation Loop | -23.5 | 10 | uM |
XMD11-85h | PC-3 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | 4.0 | 10 | uM |
XMD11-85h | PC-3 | EPHB4 | FLEENSSDPTYTSSLGGkIPIR | Activation Loop | 0.4 | 10 | uM |
XMD11-85h | PC-3 | EGFR | LLGAEEKEYHAEGGkVPIK | Activation Loop | 4.3 | 10 | uM |
XMD11-85h | PC-3 | NEK9 | LGDYGLAkK | Activation Loop | 7.8 | 10 | uM |
XMD11-85h | PC-3 | EphA7 | VIEDDPEAVYTTTGGkIPVR | Activation Loop | 4.1 | 10 | uM |
XMD11-85h | PC-3 | EPHB2 | FLEDDTSDPTYTSALGGkIPIR | Activation Loop | -37.3 | 10 | uM |
XMD11-85h | HeLa | JAK3 domain2 | IADFGLAkLLPLDKDYYVVR | Activation Loop | -13.7 | 10 | uM |
XMD11-85h | PC-3 | MET | DMYDKEYYSVHNkTGAK | Activation Loop | 38.6 | 10 | uM |
XMD11-85h | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | -38.1 | 10 | uM |
XMD11-85h | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -8.0 | 10 | uM |
XMD11-85h | HeLa | STLK5 | YSVkVLPWLSPEVLQQNLQGYDAK | Activation Loop | -30.0 | 10 | uM |
XMD11-85h | PC-3 | Wnk1,Wnk2,Wnk4 | IGDLGLATLkR | Activation Loop | -5.1 | 10 | uM |
XMD11-85h | HeLa | JAK1_domain2 | IGDFGLTkAIETDKEYYTVK | Activation Loop | -6.3 | 10 | uM |
XMD11-85h | PC-3 | FYN,SRC,YES | QGAkFPIKWTAPEAALYGR | Activation Loop | 6.7 | 10 | uM |
XMD11-85h | PC-3 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | -0.5 | 10 | uM |
XMD11-85h | HeLa | NEK9 | LGDYGLAkK | Activation Loop | -20.3 | 10 | uM |
XMD11-85h | HeLa | RSK2_domain1 | LTDFGLSkESIDHEKK | Activation Loop | -10.3 | 10 | uM |
XMD11-85h | HeLa | TEC | YVLDDQYTSSSGAkFPVK | Activation Loop | -11.8 | 10 | uM |
XMD11-85h | HeLa | PIK3C3 | TEDGGKYPVIFkHGDDLR | ATP | -5.7 | 10 | uM |