XMD11-85h KiNativ -- single dose experiment - Dataset (ID:20098)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD11-85h PC-3 eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
10.7
10
uM
XMD11-85h PC-3 RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
-2.2
10
uM
XMD11-85h HeLa RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
-7.8
10
uM
XMD11-85h HeLa IRAK3
SHLEHQSCTINMTSSSSkHLWYMPEEYIR
Protein Kinase Domain
-3.2
10
uM
XMD11-85h HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-28.6
10
uM
XMD11-85h PC-3 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
21.9
10
uM
XMD11-85h HeLa KSR1,KSR2
SkNVFYDNGK
Protein Kinase Domain
1.9
10
uM
XMD11-85h HeLa RSKL1_domain1
VLGVIDkVLLVMDTR
Protein Kinase Domain
31.3
10
uM
XMD11-85h HeLa MK14
QELNkTIWEVPER
Other
-2.2
10
uM
XMD11-85h PC-3 ROCK1
kLQLELNQER
Other
1.2
10
uM
XMD11-85h PC-3 MRCKb
NHHVHLYPWSSLDGAEGSFDIkLPETK
Other
15.0
10
uM
XMD11-85h PC-3 MK14
QELNkTIWEVPER
Other
0.5
10
uM
XMD11-85h HeLa JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Other
31.1
10
uM
XMD11-85h PC-3 MK11
QELNkTVWEVPQR
Other
-4.2
10
uM
XMD11-85h HeLa IKKA
DLkPENIVLQDVGGK
Lys2
-4.4
10
uM
XMD11-85h PC-3 GSK3B
DIkPQNLLLDPDTAVLK
Lys2
9.4
10
uM
XMD11-85h HeLa IKKE,TBK1
DIkPGNIMR
Lys2
-46.4
10
uM
XMD11-85h PC-3 GCN2_domain2
DLkPVNIFLDSDDHVK
Lys2
2.0
10
uM
XMD11-85h PC-3 KC1A
DIkPDNFLMGIGR
Lys2
17.3
10
uM
XMD11-85h HeLa GSK3A
DIkPQNLLVDPDTAVLK
Lys2
-7.2
10
uM
XMD11-85h PC-3 IKKE,TBK1
DIkPGNIMR
Lys2
12.1
10
uM
XMD11-85h HeLa BRAF
DLkSNNIFLHEDLTVK
Lys2
15.0
10
uM
XMD11-85h PC-3 CDK9
DMkAANVLITR
Lys2
3.3
10
uM
XMD11-85h HeLa MK03
DLkPSNLLINTTCDLK
Lys2
-6.6
10
uM
XMD11-85h HeLa CDK7
DLkPNNLLLDENGVLK
Lys2
-15.7
10
uM
  • Page 1 of 10
  • 1 to 25 of 241 records