XMD11-85h KiNativ -- single dose experiment - Dataset (ID:20098)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD11-85h | PC-3 | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | 10.7 | 10 | uM |
XMD11-85h | PC-3 | RSK2_domain2 | SkRDPTEEIEILLR | Protein Kinase Domain | -2.2 | 10 | uM |
XMD11-85h | HeLa | RSK2_domain2 | SkRDPTEEIEILLR | Protein Kinase Domain | -7.8 | 10 | uM |
XMD11-85h | HeLa | IRAK3 | SHLEHQSCTINMTSSSSkHLWYMPEEYIR | Protein Kinase Domain | -3.2 | 10 | uM |
XMD11-85h | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -28.6 | 10 | uM |
XMD11-85h | PC-3 | ILK | ISMADVkFSFQCPGR | Protein Kinase Domain | 21.9 | 10 | uM |
XMD11-85h | HeLa | KSR1,KSR2 | SkNVFYDNGK | Protein Kinase Domain | 1.9 | 10 | uM |
XMD11-85h | HeLa | RSKL1_domain1 | VLGVIDkVLLVMDTR | Protein Kinase Domain | 31.3 | 10 | uM |
XMD11-85h | HeLa | MK14 | QELNkTIWEVPER | Other | -2.2 | 10 | uM |
XMD11-85h | PC-3 | ROCK1 | kLQLELNQER | Other | 1.2 | 10 | uM |
XMD11-85h | PC-3 | MRCKb | NHHVHLYPWSSLDGAEGSFDIkLPETK | Other | 15.0 | 10 | uM |
XMD11-85h | PC-3 | MK14 | QELNkTIWEVPER | Other | 0.5 | 10 | uM |
XMD11-85h | HeLa | JAK1 | QLASALSYLEDKDLVHGNVCTkNLLLAR | Other | 31.1 | 10 | uM |
XMD11-85h | PC-3 | MK11 | QELNkTVWEVPQR | Other | -4.2 | 10 | uM |
XMD11-85h | HeLa | IKKA | DLkPENIVLQDVGGK | Lys2 | -4.4 | 10 | uM |
XMD11-85h | PC-3 | GSK3B | DIkPQNLLLDPDTAVLK | Lys2 | 9.4 | 10 | uM |
XMD11-85h | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | -46.4 | 10 | uM |
XMD11-85h | PC-3 | GCN2_domain2 | DLkPVNIFLDSDDHVK | Lys2 | 2.0 | 10 | uM |
XMD11-85h | PC-3 | KC1A | DIkPDNFLMGIGR | Lys2 | 17.3 | 10 | uM |
XMD11-85h | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | -7.2 | 10 | uM |
XMD11-85h | PC-3 | IKKE,TBK1 | DIkPGNIMR | Lys2 | 12.1 | 10 | uM |
XMD11-85h | HeLa | BRAF | DLkSNNIFLHEDLTVK | Lys2 | 15.0 | 10 | uM |
XMD11-85h | PC-3 | CDK9 | DMkAANVLITR | Lys2 | 3.3 | 10 | uM |
XMD11-85h | HeLa | MK03 | DLkPSNLLINTTCDLK | Lys2 | -6.6 | 10 | uM |
XMD11-85h | HeLa | CDK7 | DLkPNNLLLDENGVLK | Lys2 | -15.7 | 10 | uM |