XMD11-85h KiNativ -- single dose experiment - Dataset (ID:20098)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD11-85h | HeLa | GCK | DTVTSELAAVkIVK | Lys1 | -2.7 | 10 | uM |
| XMD11-85h | HeLa | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | -16.3 | 10 | uM |
| XMD11-85h | HeLa | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | -21.2 | 10 | uM |
| XMD11-85h | HeLa | FER | TSVAVkTCKEDLPQELK | Lys1 | -20.4 | 10 | uM |
| XMD11-85h | HeLa | IKKA | DLkPENIVLQDVGGK | Lys2 | -4.4 | 10 | uM |
| XMD11-85h | HeLa | ILK | WQGNDIVVkVLK | Lys1 | -7.3 | 10 | uM |
| XMD11-85h | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -8.0 | 10 | uM |
| XMD11-85h | HeLa | DMPK | DIkPDNILLDR | Lys2 | 16.5 | 10 | uM |
| XMD11-85h | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -28.6 | 10 | uM |
| XMD11-85h | HeLa | Erk5 | DLkPSNLLVNENCELK | Lys2 | -8.8 | 10 | uM |
| XMD11-85h | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | -7.2 | 10 | uM |
| XMD11-85h | HeLa | CaMK2g | TSTQEYAAkIINTK | Lys1 | -16.1 | 10 | uM |
| XMD11-85h | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | -38.1 | 10 | uM |
| XMD11-85h | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | -46.4 | 10 | uM |
| XMD11-85h | HeLa | ARAF | DLkSNNIFLHEGLTVK | Lys2 | 4.5 | 10 | uM |
| XMD11-85h | HeLa | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | -34.6 | 10 | uM |
| XMD11-85h | HeLa | CDK2 | DLkPQNLLINTEGAIK | Lys2 | -4.5 | 10 | uM |
| XMD11-85h | HeLa | ATR | FYIMMCkPK | ATP | -8.9 | 10 | uM |
| XMD11-85h | HeLa | ACK | TVSVAVkCLKPDVLSQPEAMDDFIR | Lys1 | -2.4 | 10 | uM |
| XMD11-85h | HeLa | CDK7 | DLkPNNLLLDENGVLK | Lys2 | -15.7 | 10 | uM |
| XMD11-85h | HeLa | BRAF | DLkSNNIFLHEDLTVK | Lys2 | 15.0 | 10 | uM |
| XMD11-85h | HeLa | MK03 | DLkPSNLLINTTCDLK | Lys2 | -6.6 | 10 | uM |
| XMD11-85h | HeLa | CaMK1a | LVAIkCIAK | Lys1 | -10.7 | 10 | uM |
| XMD11-85h | HeLa | IRE1 | DLkPHNILISMPNAHGK | Lys2 | -26.2 | 10 | uM |
| XMD11-85h | HeLa | IRAK4 | DIkSANILLDEAFTAK | Lys2 | 11.1 | 10 | uM |