XMD11-85h KiNativ -- single dose experiment - Dataset (ID:20098)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD11-85h | PC-3 | MAP3K4 | DIkGANIFLTSSGLIK | Lys2 | -9.9 | 10 | uM |
| XMD11-85h | PC-3 | CASK | ETGQQFAVkIVDVAK | Lys1 | -9.9 | 10 | uM |
| XMD11-85h | PC-3 | p38a | DLkPSNLAVNEDCELK | Lys2 | 9.8 | 10 | uM |
| XMD11-85h | HeLa | RSK1,RSK2_domain1 | DLkPENILLDEEGHIKLTDFGLSK | Lys2 | 9.6 | 10 | uM |
| XMD11-85h | HeLa | ULK3 | EVVAIkCVAK | Lys1 | -9.6 | 10 | uM |
| XMD11-85h | HeLa | MST1 | ETGQIVAIkQVPVESDLQEIIK | Lys1 | 9.4 | 10 | uM |
| XMD11-85h | PC-3 | GSK3B | DIkPQNLLLDPDTAVLK | Lys2 | 9.4 | 10 | uM |
| XMD11-85h | HeLa | MAP3K1 | DVkGANLLIDSTGQR | Lys2 | -9.3 | 10 | uM |
| XMD11-85h | HeLa | MST2 | ESGQVVAIkQVPVESDLQEIIK | Lys1 | 9.2 | 10 | uM |
| XMD11-85h | HeLa | RSK1,RSK4 domain1 | VLGQGSFGkVFLVR | ATP Loop | 9.0 | 10 | uM |
| XMD11-85h | HeLa | CAMK1D | LFAVkCIPK | Lys1 | -8.9 | 10 | uM |
| XMD11-85h | HeLa | ATR | FYIMMCkPK | ATP | -8.9 | 10 | uM |
| XMD11-85h | PC-3 | MARK2 | EVAVkIIDKTQLNSSSLQK | Lys1 | 8.8 | 10 | uM |
| XMD11-85h | HeLa | Erk5 | DLkPSNLLVNENCELK | Lys2 | -8.8 | 10 | uM |
| XMD11-85h | PC-3 | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | 8.6 | 10 | uM |
| XMD11-85h | PC-3 | KHS1 | NVHTGELAAVkIIK | Lys1 | -8.6 | 10 | uM |
| XMD11-85h | PC-3 | MLTK | WISQDKEVAVKk | Lys1 | 8.5 | 10 | uM |
| XMD11-85h | HeLa | IKKE | SGELVAVkVFNTTSYLRPR | Lys1 | -8.5 | 10 | uM |
| XMD11-85h | HeLa | FES | LRADNTLVAVkSCR | Lys1 | -8.4 | 10 | uM |
| XMD11-85h | PC-3 | PIK3CB | VFGEDSVGVIFkNGDDLRQDMLTLQMLR | ATP | -82.1 | 10 | uM |
| XMD11-85h | PC-3 | SRPK1/2 | FVAMkVVK | Lys1 | 8.1 | 10 | uM |
| XMD11-85h | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -8.0 | 10 | uM |
| XMD11-85h | HeLa | HPK1 | DKVSGDLVALkMVK | Lys1 | -8.0 | 10 | uM |
| XMD11-85h | PC-3 | NEK9 | LGDYGLAkK | Activation Loop | 7.8 | 10 | uM |
| XMD11-85h | HeLa | RSK2_domain2 | SkRDPTEEIEILLR | Protein Kinase Domain | -7.8 | 10 | uM |