Evaluation of the sensitivities of six triple-negative breast cancer (TNBC) cell lines to 23 different PI3K/AKT/mTOR inhibitors or to a MEK inhibitor (trametinib). Dataset 1 of 2: GR values. - Dataset (ID:20364)

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Cell line Drug name Experimental replicate Timepoint Drug concentration Live cell count Average live cell count, DMSO control Average live cell count (time = 0) Log10(drug concentration) GR value Relative cell count (treatment versus DMSO) Cell doublings (DMSO control) Experiment name
Hs 578T Buparlisib 3 72
0.1
3869.5 4235.0 571.3
-1.0
0.939 0.914 2.890
Hs578T BKM120 3
Hs 578T Buparlisib 3 72
0.32
3143.5 4235.0 571.3
-0.495
0.804 0.742 2.890
Hs578T BKM120 3
Hs 578T Buparlisib 3 72
1.0
1442.8 4235.0 571.3
0.0
0.378 0.341 2.890
Hs578T BKM120 3
Hs 578T Buparlisib 3 72
3.2
115.3 4235.0 571.3
0.505
-0.425 0.027 2.890
Hs578T BKM120 3
Hs 578T BX-912 3 72
0.001
4175.8 3993.8 571.3
-3.0
1.030 1.050 2.805
Hs578T BX912 3
Hs 578T BX-912 3 72
0.0032
4202.0 3993.8 571.3
-2.49
1.040 1.050 2.805
Hs578T BX912 3
Hs 578T BX-912 3 72
0.01
4285.5 3993.8 571.3
-2.0
1.050 1.070 2.805
Hs578T BX912 3
Hs 578T BX-912 3 72
0.032
4271.3 3993.8 571.3
-1.49
1.050 1.070 2.805
Hs578T BX912 3
Hs 578T BX-912 3 72
0.1
4017.5 3993.8 571.3
-1.0
1.000 1.010 2.805
Hs578T BX912 3
Hs 578T BX-912 3 72
0.32
3679.8 3993.8 571.3
-0.495
0.942 0.921 2.805
Hs578T BX912 3
Hs 578T BX-912 3 72
1.0
1860.5 3993.8 571.3
0.0
0.523 0.466 2.805
Hs578T BX912 3
Hs 578T BX-912 3 72
3.2
591.0 3993.8 571.3
0.505
0.012 0.148 2.805
Hs578T BX912 3
Hs 578T Alpelisib 3 72
0.001
4208.5 4137.8 571.3
-3.0
1.010 1.020 2.856
Hs578T BYL719 3
Hs 578T Alpelisib 3 72
0.0032
4164.3 4137.8 571.3
-2.49
1.000 1.010 2.856
Hs578T BYL719 3
Hs 578T Alpelisib 3 72
0.01
4273.3 4137.8 571.3
-2.0
1.020 1.030 2.856
Hs578T BYL719 3
Hs 578T Alpelisib 3 72
0.032
3790.5 4137.8 571.3
-1.49
0.940 0.916 2.856
Hs578T BYL719 3
Hs 578T Alpelisib 3 72
0.1
3935.8 4137.8 571.3
-1.0
0.965 0.951 2.856
Hs578T BYL719 3
Hs 578T Alpelisib 3 72
0.32
3419.0 4137.8 571.3
-0.495
0.871 0.826 2.856
Hs578T BYL719 3
Hs 578T Alpelisib 3 72
1.0
3087.3 4137.8 571.3
0.0
0.805 0.746 2.856
Hs578T BYL719 3
Hs 578T Alpelisib 3 72
3.2
2652.0 4137.8 571.3
0.505
0.712 0.641 2.856
Hs578T BYL719 3
Hs 578T CAL-101 3 72
0.001
4189.5 4189.5 571.3
-3.0
1.000 1.000 2.874
Hs578T CAL101 3
Hs 578T CAL-101 3 72
0.0032
4192.0 4189.5 571.3
-2.49
1.000 1.000 2.874
Hs578T CAL101 3
Hs 578T CAL-101 3 72
0.01
4238.3 4189.5 571.3
-2.0
1.010 1.010 2.874
Hs578T CAL101 3
Hs 578T CAL-101 3 72
0.032
4226.0 4189.5 571.3
-1.49
1.010 1.010 2.874
Hs578T CAL101 3
Hs 578T CAL-101 3 72
0.1
4231.8 4189.5 571.3
-1.0
1.010 1.010 2.874
Hs578T CAL101 3