Evaluation of the sensitivities of six triple-negative breast cancer (TNBC) cell lines to 23 different PI3K/AKT/mTOR inhibitors or to a MEK inhibitor (trametinib). Dataset 1 of 2: GR values. - Dataset (ID:20364)

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Cell line Drug name Experimental replicate Timepoint Drug concentration Live cell count Average live cell count, DMSO control Average live cell count (time = 0) Log10(drug concentration) GR value Relative cell count (treatment versus DMSO) Cell doublings (DMSO control) Experiment name
Hs 578T AZD8055 1 72
0.1
1406.0 3514.5 873.1
-1.0
0.268 0.400 2.009
Hs578T AZD8055 1
Hs 578T AZD8055 1 72
0.32
1141.3 3514.5 873.1
-0.495
0.143 0.325 2.009
Hs578T AZD8055 1
Hs 578T AZD8055 1 72
1.0
1056.5 3514.5 873.1
0.0
0.100 0.301 2.009
Hs578T AZD8055 1
Hs 578T AZD8055 1 72
3.2
1005.8 3514.5 873.1
0.505
0.073 0.286 2.009
Hs578T AZD8055 1
Hs 578T Dactolisib 1 72
0.001
3257.3 3608.8 873.1
-3.0
0.902 0.903 2.047
Hs578T BEZ235 1
Hs 578T Dactolisib 1 72
0.0032
2819.5 3608.8 873.1
-2.49
0.773 0.781 2.047
Hs578T BEZ235 1
Hs 578T Dactolisib 1 72
0.01
1815.0 3608.8 873.1
-2.0
0.430 0.503 2.047
Hs578T BEZ235 1
Hs 578T Dactolisib 1 72
0.032
1346.5 3608.8 873.1
-1.49
0.236 0.373 2.047
Hs578T BEZ235 1
Hs 578T Dactolisib 1 72
0.1
1208.5 3608.8 873.1
-1.0
0.172 0.335 2.047
Hs578T BEZ235 1
Hs 578T Dactolisib 1 72
0.32
1095.0 3608.8 873.1
-0.495
0.117 0.303 2.047
Hs578T BEZ235 1
Hs 578T Dactolisib 1 72
1.0
899.5 3608.8 873.1
0.0
0.015 0.249 2.047
Hs578T BEZ235 1
Hs 578T Dactolisib 1 72
3.2
768.3 3608.8 873.1
0.505
-0.061 0.213 2.047
Hs578T BEZ235 1
Hs 578T Buparlisib 1 72
0.001
3598.5 3651.8 873.1
-3.0
0.986 0.985 2.064
Hs578T BKM120 1
Hs 578T Buparlisib 1 72
0.0032
3416.3 3651.8 873.1
-2.49
0.936 0.936 2.064
Hs578T BKM120 1
Hs 578T Buparlisib 1 72
0.01
3506.0 3651.8 873.1
-2.0
0.961 0.960 2.064
Hs578T BKM120 1
Hs 578T Buparlisib 1 72
0.032
3520.3 3651.8 873.1
-1.49
0.965 0.964 2.064
Hs578T BKM120 1
Hs 578T Buparlisib 1 72
0.1
3235.0 3651.8 873.1
-1.0
0.886 0.886 2.064
Hs578T BKM120 1
Hs 578T Buparlisib 1 72
0.32
2526.8 3651.8 873.1
-0.495
0.673 0.692 2.064
Hs578T BKM120 1
Hs 578T Buparlisib 1 72
1.0
1329.3 3651.8 873.1
0.0
0.226 0.364 2.064
Hs578T BKM120 1
Hs 578T Buparlisib 1 72
3.2
146.5 3651.8 873.1
0.505
-0.579 0.040 2.064
Hs578T BKM120 1
Hs 578T BX-912 1 72
0.001
3608.5 3493.8 873.1
-3.0
1.030 1.030 2.001
Hs578T BX912 1
Hs 578T BX-912 1 72
0.0032
3647.8 3493.8 873.1
-2.49
1.040 1.040 2.001
Hs578T BX912 1
Hs 578T BX-912 1 72
0.01
3559.8 3493.8 873.1
-2.0
1.020 1.020 2.001
Hs578T BX912 1
Hs 578T BX-912 1 72
0.032
3582.3 3493.8 873.1
-1.49
1.030 1.030 2.001
Hs578T BX912 1
Hs 578T BX-912 1 72
0.1
3418.5 3493.8 873.1
-1.0
0.978 0.978 2.001
Hs578T BX912 1